YU52303A - Postupak karbamoilacije alkohola - Google Patents

Postupak karbamoilacije alkohola

Info

Publication number
YU52303A
YU52303A YU52303A YUP52303A YU52303A YU 52303 A YU52303 A YU 52303A YU 52303 A YU52303 A YU 52303A YU P52303 A YUP52303 A YU P52303A YU 52303 A YU52303 A YU 52303A
Authority
YU
Yugoslavia
Prior art keywords
carbamoylating
alcohol
moiety
alcohols
sulfenyl
Prior art date
Application number
YU52303A
Other languages
English (en)
Inventor
James Edward Ellis
Original Assignee
Warner-Lambert Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner-Lambert Company filed Critical Warner-Lambert Company
Publication of YU52303A publication Critical patent/YU52303A/sh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)

Abstract

Ovaj pronalazak se odnosi na postupke za karbamoilaciju alkohola sa natrijum cijanatom u prisustvu metansulfonske kiseline. Reakcija se može odigrati pod anhidrovanim uslovima. Ovaj postupak je pogodan za karbamoilaciju molekula sa alkoholnim delom i baznim delom i/ili molekulom koji sadrži i alkoholni deo i sulfenil deo, kao što je prekursor sulfenil alkohola antiviralnog agensa Capravirina.[The present invention includes a method for carbamoylating an alcohol with sodium cyanate in the presence of methanesulfonic acid. The reaction can be conducted under anhydrous conditions. This method is suitable for carbamoylating a molecule including both an alcohol moiety and a basic moiety and/or a molecule including both an alcohol moiety and a sulfenyl moiety, such as the sulfenyl alcohol precursor of the antiviral agent Capravirine.
YU52303A 2001-01-31 2002-01-11 Postupak karbamoilacije alkohola YU52303A (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US26550201P 2001-01-31 2001-01-31

Publications (1)

Publication Number Publication Date
YU52303A true YU52303A (sh) 2006-05-25

Family

ID=23010706

Family Applications (1)

Application Number Title Priority Date Filing Date
YU52303A YU52303A (sh) 2001-01-31 2002-01-11 Postupak karbamoilacije alkohola

Country Status (19)

Country Link
US (1) US6613908B2 (sh)
EP (1) EP1377568A1 (sh)
JP (1) JP2004518687A (sh)
KR (1) KR100567706B1 (sh)
CN (1) CN1243748C (sh)
AR (1) AR032419A1 (sh)
BR (1) BR0206806A (sh)
CA (1) CA2433364A1 (sh)
CZ (1) CZ20032001A3 (sh)
HK (1) HK1060573A1 (sh)
HU (1) HUP0303028A3 (sh)
IL (1) IL156363A0 (sh)
MX (1) MXPA03005403A (sh)
PL (1) PL363321A1 (sh)
RU (1) RU2256657C2 (sh)
TW (1) TWI228507B (sh)
WO (1) WO2002060893A1 (sh)
YU (1) YU52303A (sh)
ZA (1) ZA200304687B (sh)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA014685B1 (ru) 2003-04-25 2010-12-30 Джилид Сайэнс, Инк. Фосфонатсодержащие антивирусные соединения (варианты) и фармацевтическая композиция на их основе
AU2004260789B2 (en) * 2003-07-30 2011-06-30 Gilead Sciences, Inc. Nucleobase phosphonate analogs for antiviral treatment
WO2005016912A1 (en) * 2003-08-19 2005-02-24 Pfizer Inc. An efficient microbial preparation of capravirine metabolites m4 and m5
US20050080268A1 (en) * 2003-10-08 2005-04-14 Yong-Moon Choi Process of preparing O-carbamoyl compounds in the presence of active amine group
NZ552405A (en) * 2004-07-16 2011-04-29 Gilead Sciences Inc Pyrrolidine containing antiviral compounds
UA88313C2 (ru) 2004-07-27 2009-10-12 Гилиад Сайенсиз, Инк. Фосфонатные аналоги соединений ингибиторов вич
TW200738742A (en) * 2005-07-14 2007-10-16 Gilead Sciences Inc Antiviral compounds
TWI389908B (zh) * 2005-07-14 2013-03-21 Gilead Sciences Inc 抗病毒化合物類
EP1906971A2 (en) * 2005-07-27 2008-04-09 Gilead Sciences, Inc. Antiviral compounds
US7842672B2 (en) * 2006-07-07 2010-11-30 Gilead Sciences, Inc. Phosphonate inhibitors of HCV
EA018308B1 (ru) 2008-07-08 2013-07-30 Джилид Сайэнс, Инк. Соли соединений ингибиторов вич
US8810796B2 (en) 2009-04-21 2014-08-19 Michigan Aerospace Corporation Light processing system and method
PL3661937T3 (pl) 2017-08-01 2021-12-20 Gilead Sciences, Inc. Formy krystaliczne ((s)-((((2r,5r)-5-(6-amino-9h-puryn-9-ylo)-4-fluoro-2,5-dihydrofuran-2-ylo)oksy)metylo)(fenoksy)fosforylo)-l-alaninianu etylu (gs-9131) do leczenia zakażeń wirusowych

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2611695A1 (de) * 1976-03-19 1977-09-29 Hoechst Ag Herbizide mittel
CA2200316C (en) 1994-09-26 2004-09-21 Hirohiko Sugimoto Imidazole derivative

Also Published As

Publication number Publication date
HUP0303028A2 (hu) 2003-12-29
HK1060573A1 (en) 2004-08-13
CA2433364A1 (en) 2002-08-08
CN1243748C (zh) 2006-03-01
KR100567706B1 (ko) 2006-04-05
MXPA03005403A (es) 2003-09-25
IL156363A0 (en) 2004-01-04
CN1489584A (zh) 2004-04-14
US20020103378A1 (en) 2002-08-01
WO2002060893A1 (en) 2002-08-08
PL363321A1 (en) 2004-11-15
ZA200304687B (en) 2004-08-10
JP2004518687A (ja) 2004-06-24
BR0206806A (pt) 2004-02-03
AR032419A1 (es) 2003-11-05
TWI228507B (en) 2005-03-01
HUP0303028A3 (en) 2005-10-28
EP1377568A1 (en) 2004-01-07
KR20030069227A (ko) 2003-08-25
RU2256657C2 (ru) 2005-07-20
CZ20032001A3 (en) 2004-06-16
US6613908B2 (en) 2003-09-02
RU2003123791A (ru) 2005-02-27

Similar Documents

Publication Publication Date Title
YU52303A (sh) Postupak karbamoilacije alkohola
PL354050A1 (en) 8-(anilino)-1-naphthalenesulfonate analogs and their use in analyte detection assays
TW200514773A (en) Selective synthesis of CF3-substituted pyrimidines
HU0302444D0 (en) Process for monomethylation of nitrogen containing heterocyclic compounds
IL158249A (en) Process for the preparation of oxabispidines
TW200510285A (en) Method for purifying a fluoroalcohol
BR0117163A (pt) Método e equipamento para a preparação de hidrazodicarbonamida utilizando uréia como material de partida
BR0009453A (pt) Processo para a preparação de um composto
MXPA03002937A (es) Benzimidazoles n-alcoxialquil-substituidos y su uso como agentes contra protozoos parasitantes.
SE0101323D0 (sv) New process
ZA978492B (en) Process for amines.
GB9714302D0 (en) Process
BR0113944A (pt) Processo para a produção de compostos quirais
IL158785A0 (en) Uncatalysed addition reactions
BR9810687B1 (pt) processo para a preparação de um composto derivado de 2-alquiltiobenzonitrila.
BR0308297A (pt) Processo para a preparação de um composto
TH60482A (th) การปรับสภาพซับสเทรทชนิดแข็งเพื่อเสริมความทนทานของการปรับสภาพที่ประยุกต์ใช้บนที่นั้น
IL158530A0 (en) Method for producing 1,3-disubstituted 2-nitroguanidines
RS20100109A (en) Process for preparing 4-trifluoromethzlsulphinylpyrazole derivative
RS20100110A (en) Process for preparing 4- trifluoromethylsulphinylpyrazole derivative
UA67370A (en) A method for the preparation of bis (methylthio) methane
AR035928A1 (es) Procedimiento para la sintesis de antraciclinas opticamente activas e intermediarios de reaccion utilizados en dicho proceso