YU10396A - Postupak za proizvodnju l-aspartil-d-alanin-n-(tietan-3-il)-amida - Google Patents

Postupak za proizvodnju l-aspartil-d-alanin-n-(tietan-3-il)-amida

Info

Publication number
YU10396A
YU10396A YU10396A YU10396A YU10396A YU 10396 A YU10396 A YU 10396A YU 10396 A YU10396 A YU 10396A YU 10396 A YU10396 A YU 10396A YU 10396 A YU10396 A YU 10396A
Authority
YU
Yugoslavia
Prior art keywords
aspartyl
general formula
thietan
alanin
amides
Prior art date
Application number
YU10396A
Other languages
English (en)
Inventor
Karlheinz Drauz
Gunter Knaup
Stefan Retzow
Michael Schkarm
Christoph Weckbecker
Original Assignee
Degussa Aktiengesellchaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Degussa Aktiengesellchaft filed Critical Degussa Aktiengesellchaft
Publication of YU10396A publication Critical patent/YU10396A/sh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06104—Dipeptides with the first amino acid being acidic
    • C07K5/06113—Asp- or Asn-amino acid
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Seasonings (AREA)

Abstract

Postupak za proizvodnju L-aspartil-D-alanin-N-(tietan-3-il)-amida sa opštom formulom I pretvaranjem D-alanin-tietanamida opšte formule II sa jedinjenjima oksazolidinona opšte formule III u jednom inertnom organskom rastvaraču, u kojima R1 označava H ili jednu selektivno izdvojivu zaštitnu grupu, R2 - R5 medjusobno nezavisno su jednaki ili različiti: H, ili C1-C4-alkil, linearno ili razgranato, a R6 i R7 medjusobno nezavisno su jednaki ili različiti: H, C1-C4-alkil, linearno ili razgranato, aril ili jedan ostatak, koji aktivira karbonilnu grupu.
YU10396A 1995-02-21 1996-02-20 Postupak za proizvodnju l-aspartil-d-alanin-n-(tietan-3-il)-amida YU10396A (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19505933A DE19505933C2 (de) 1995-02-21 1995-02-21 Verfahren zur Herstellung von L-Aspartyl-D-alanin-N-(thietan-3-yl)-amiden

Publications (1)

Publication Number Publication Date
YU10396A true YU10396A (sh) 1998-09-18

Family

ID=7754609

Family Applications (1)

Application Number Title Priority Date Filing Date
YU10396A YU10396A (sh) 1995-02-21 1996-02-20 Postupak za proizvodnju l-aspartil-d-alanin-n-(tietan-3-il)-amida

Country Status (9)

Country Link
US (1) US5874121A (sh)
EP (1) EP0811012B1 (sh)
AU (1) AU4716496A (sh)
DE (2) DE19505933C2 (sh)
HR (1) HRP960083A2 (sh)
IL (1) IL117190A0 (sh)
WO (1) WO1996026213A1 (sh)
YU (1) YU10396A (sh)
ZA (1) ZA961343B (sh)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL1010867C2 (nl) * 1998-12-22 2000-06-23 Dsm Nv Werkwijze voor de bereiding van aminozuuramiden of derivaten daarvan.
DE10333368B4 (de) * 2003-07-23 2008-08-28 Universität Leipzig Oberflächenfunktionalisiertes Trägermaterial, Verfahren zu dessen Herstellung und dessen Verwendungen
FR2876102A1 (fr) * 2004-10-04 2006-04-07 Solvay Compose heterocyclique enantiopur
CN115093391B (zh) * 2022-06-28 2024-05-03 上海毕得医药科技股份有限公司 一种3-硫杂环丁胺盐酸盐的合成方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4411925A (en) * 1980-01-21 1983-10-25 Pfizer Inc. Branched amides of L-aspartyl-d-amino acid dipeptides
US4730076A (en) * 1985-12-18 1988-03-08 Nippon Kayaku Kabushiki Kaisha Process for producing α-aspartyl-phenylalanine ester
AT394854B (de) * 1986-06-12 1992-07-10 Biochemie Gmbh Verfahren zur herstellung von n-l-alpha-aspartyl-l-phenylalanin(nieder)alkylestern

Also Published As

Publication number Publication date
US5874121A (en) 1999-02-23
WO1996026213A1 (de) 1996-08-29
ZA961343B (en) 1996-08-26
IL117190A0 (en) 1996-06-18
AU4716496A (en) 1996-09-11
DE19505933C2 (de) 2000-09-21
EP0811012B1 (de) 1999-05-26
DE19505933A1 (de) 1996-08-22
EP0811012A1 (de) 1997-12-10
HRP960083A2 (en) 1997-08-31
DE59602002D1 (de) 1999-07-01

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