WO2015068171A1 - Nouveaux composés oxazolidinone - Google Patents

Nouveaux composés oxazolidinone Download PDF

Info

Publication number
WO2015068171A1
WO2015068171A1 PCT/IN2014/000018 IN2014000018W WO2015068171A1 WO 2015068171 A1 WO2015068171 A1 WO 2015068171A1 IN 2014000018 W IN2014000018 W IN 2014000018W WO 2015068171 A1 WO2015068171 A1 WO 2015068171A1
Authority
WO
WIPO (PCT)
Prior art keywords
compound
formula
methyl
oxooxazolidin
acetamide
Prior art date
Application number
PCT/IN2014/000018
Other languages
English (en)
Inventor
Raghu Mitra ALLA
Ajay Kumar DUBEY
Srinivas Reddy Mallepalli
Ramakrishna Reddy PONGILATI
Original Assignee
Lee Pharma Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lee Pharma Limited filed Critical Lee Pharma Limited
Publication of WO2015068171A1 publication Critical patent/WO2015068171A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

Nouveau composé oxazolidinone (S)-N-((3-(4-fluoro-3-morpholinophényl)-2-oxooxazolidin-5-yl)méthyl)acétamide de formule-I et procédé pour le préparer. Composé-I
PCT/IN2014/000018 2013-11-08 2014-01-08 Nouveaux composés oxazolidinone WO2015068171A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN5063CH2013 2013-11-08
IN5063/CHE/2013 2013-11-08

Publications (1)

Publication Number Publication Date
WO2015068171A1 true WO2015068171A1 (fr) 2015-05-14

Family

ID=53040990

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/IN2014/000018 WO2015068171A1 (fr) 2013-11-08 2014-01-08 Nouveaux composés oxazolidinone

Country Status (1)

Country Link
WO (1) WO2015068171A1 (fr)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9573910B2 (en) 2013-11-08 2017-02-21 Lee Pharma Limited Oxazolidinone antibacterial compound
CN108135887A (zh) * 2015-10-22 2018-06-08 默沙东公司 噁唑烷酮化合物及其作为抗菌剂的使用方法
RU2794494C2 (ru) * 2016-10-17 2023-04-19 МЕРК ШАРП И ДОУМ ЭлЭлСи Оксазолидиноновые соединения и способы их применения в качестве противобактериальных средств

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995007271A1 (fr) * 1993-09-09 1995-03-16 The Upjohn Company Agents antimicrobiens oxazolidinone a substitution oxazine et thiazine
WO1999037630A1 (fr) * 1998-01-23 1999-07-29 Versicor, Inc. Banques combinatoires d'oxazolidinones, compositions a base de tels composes et procedes de preparation
WO2003063862A1 (fr) * 2002-01-25 2003-08-07 Pharmacia & Upjohn Company Cotherapie avec une oxazolidinone et une vitamine b

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995007271A1 (fr) * 1993-09-09 1995-03-16 The Upjohn Company Agents antimicrobiens oxazolidinone a substitution oxazine et thiazine
WO1999037630A1 (fr) * 1998-01-23 1999-07-29 Versicor, Inc. Banques combinatoires d'oxazolidinones, compositions a base de tels composes et procedes de preparation
WO2003063862A1 (fr) * 2002-01-25 2003-08-07 Pharmacia & Upjohn Company Cotherapie avec une oxazolidinone et une vitamine b

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9573910B2 (en) 2013-11-08 2017-02-21 Lee Pharma Limited Oxazolidinone antibacterial compound
CN108135887A (zh) * 2015-10-22 2018-06-08 默沙东公司 噁唑烷酮化合物及其作为抗菌剂的使用方法
EP3364968A4 (fr) * 2015-10-22 2019-05-01 Merck Sharp & Dohme Corp. Composés d'oxazolidinone et procédés pour les utiliser comme agents antibactériens
US10947205B2 (en) 2015-10-22 2021-03-16 Merck Sharp & Dohme Corp. Oxazolidinone compounds and methods of use thereof as antibacterial agents
CN108135887B (zh) * 2015-10-22 2021-07-30 默沙东公司 噁唑烷酮化合物及其作为抗菌剂的使用方法
RU2794494C2 (ru) * 2016-10-17 2023-04-19 МЕРК ШАРП И ДОУМ ЭлЭлСи Оксазолидиноновые соединения и способы их применения в качестве противобактериальных средств

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