UY34150A - Cristal de compuesto heterociclico fusionado - Google Patents

Cristal de compuesto heterociclico fusionado

Info

Publication number
UY34150A
UY34150A UY0001034150A UY34150A UY34150A UY 34150 A UY34150 A UY 34150A UY 0001034150 A UY0001034150 A UY 0001034150A UY 34150 A UY34150 A UY 34150A UY 34150 A UY34150 A UY 34150A
Authority
UY
Uruguay
Prior art keywords
heterociclic
fused
composite crystal
composite
crystal
Prior art date
Application number
UY0001034150A
Other languages
English (en)
Inventor
Yamamoto Katsuhiko
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of UY34150A publication Critical patent/UY34150A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

La presente invención se refiere a un cristal de 1-etil-7-metil-3-{4-[(3-metil-3H-imidazo[4,5-b]piridin-2- il)oxi]fenil}-1,3-dihidro-2H-imidazo[4,5-b]piridin-2-ona útil como un agente profiláctico o terapéutico para la esquizofrenia y similares, qu e muestra un patrón de difracción de polvo por rayos X con picos característicos enespaciamientos interplanares (d) de 13,59±0,2 y 6,76±0,2 Angstroms en la difracción de polvo por rayos X.
UY0001034150A 2011-06-22 2012-06-21 Cristal de compuesto heterociclico fusionado UY34150A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2011138920 2011-06-22

Publications (1)

Publication Number Publication Date
UY34150A true UY34150A (es) 2013-01-31

Family

ID=46551819

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001034150A UY34150A (es) 2011-06-22 2012-06-21 Cristal de compuesto heterociclico fusionado

Country Status (26)

Country Link
US (1) US9512118B2 (es)
EP (1) EP2723738B1 (es)
JP (1) JP6025757B2 (es)
KR (1) KR20140040777A (es)
CN (1) CN103608348B (es)
AR (1) AR087004A1 (es)
AU (1) AU2012274292B2 (es)
BR (1) BR112013032052A2 (es)
CA (1) CA2839825C (es)
CL (1) CL2013003632A1 (es)
CO (1) CO6862150A2 (es)
CR (1) CR20140033A (es)
DO (1) DOP2013000311A (es)
EA (1) EA026137B1 (es)
EC (1) ECSP14013165A (es)
GE (1) GEP20166475B (es)
MA (1) MA35274B1 (es)
MX (1) MX342990B (es)
MY (1) MY163483A (es)
PE (1) PE20141030A1 (es)
TN (1) TN2013000510A1 (es)
TW (1) TWI570122B (es)
UA (1) UA112082C2 (es)
UY (1) UY34150A (es)
WO (1) WO2012176934A1 (es)
ZA (1) ZA201309611B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5973990B2 (ja) * 2011-03-16 2016-08-23 武田薬品工業株式会社 縮合複素環化合物
US10851076B2 (en) 2017-08-10 2020-12-01 Pratt Bethers Method for purifying crystals using solvent vapors
US10308626B1 (en) 2018-07-02 2019-06-04 Pratt Bethers Crystal purification in a glass or metal container
US10960322B2 (en) 2018-07-02 2021-03-30 Pratt Bethers Apparatus for purifying crystals using solvent vapors

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5597826A (en) * 1994-09-14 1997-01-28 Pfizer Inc. Compositions containing sertraline and a 5-HT1D receptor agonist or antagonist
WO2006038111A1 (en) * 2004-10-07 2006-04-13 Pfizer Products Inc. Benzoimidazole derivatives useful as antiproliferative agents
WO2007026664A1 (ja) 2005-08-30 2007-03-08 Asahi Kasei Pharma Corporation スルホンアミド化合物
FI20055498A0 (fi) 2005-09-16 2005-09-16 Biotie Therapies Corp Sulfonamidijohdannaisia
US7618982B2 (en) 2005-12-19 2009-11-17 Nerviano Medical Sciences S.R.L. Heteroarylpyrrolopyridinones active as kinase inhibitors
CA2636873A1 (en) * 2006-02-15 2007-08-23 Sanofi-Aventis Azacyclyl-substituted aryldihydroisoquinolinones, process for their preparation and their use as medicaments
US20080090834A1 (en) * 2006-07-06 2008-04-17 Pfizer Inc Selective azole pde10a inhibitor compounds
KR101524817B1 (ko) 2007-04-18 2015-06-01 깃세이 야쿠힌 고교 가부시키가이샤 질소 함유 축합환 유도체, 그것을 함유하는 의약 조성물 및 그 의약 용도
EP2276747A1 (en) 2008-03-11 2011-01-26 Cellzome Limited Sulfonamides as zap-70 inhibitors
TW201030001A (en) 2008-11-14 2010-08-16 Amgen Inc Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors
TWI396689B (zh) 2008-11-14 2013-05-21 Amgen Inc 作為磷酸二酯酶10抑制劑之吡衍生物
WO2010126002A1 (ja) 2009-04-28 2010-11-04 塩野義製薬株式会社 ヘテロ環スルホンアミド化合物を含有する医薬
EP2585462B1 (en) * 2010-06-24 2020-02-26 Takeda Pharmaceutical Company Limited Fused heterocyclic compounds as phosphodiesterases (pdes) inhibitors
US9029536B2 (en) 2010-08-04 2015-05-12 Takeda Pharmaceutical Company Limited Fused heterocyclic compounds
US9150588B2 (en) 2010-08-10 2015-10-06 Takeda Pharmaceutical Company Limited Substituted pyridazin-4(1H)-ones as phosphodiesterase 10A inhibitors
JP5973990B2 (ja) 2011-03-16 2016-08-23 武田薬品工業株式会社 縮合複素環化合物

Also Published As

Publication number Publication date
MX342990B (es) 2016-10-20
CO6862150A2 (es) 2014-02-10
EP2723738A1 (en) 2014-04-30
MY163483A (en) 2017-09-15
WO2012176934A1 (en) 2012-12-27
CR20140033A (es) 2014-03-12
AR087004A1 (es) 2014-02-05
MA35274B1 (fr) 2014-07-03
JP6025757B2 (ja) 2016-11-16
CL2013003632A1 (es) 2014-06-06
TN2013000510A1 (en) 2015-03-30
CN103608348B (zh) 2016-03-30
CA2839825A1 (en) 2012-12-27
CA2839825C (en) 2019-04-09
ECSP14013165A (es) 2014-02-28
UA112082C2 (uk) 2016-07-25
EP2723738B1 (en) 2018-03-14
JP2014516918A (ja) 2014-07-17
TW201313709A (zh) 2013-04-01
NZ618944A (en) 2015-08-28
ZA201309611B (en) 2014-08-27
PE20141030A1 (es) 2014-08-29
CN103608348A (zh) 2014-02-26
AU2012274292B2 (en) 2016-10-27
GEP20166475B (en) 2016-05-10
MX2013015354A (es) 2014-02-11
TWI570122B (zh) 2017-02-11
BR112013032052A2 (pt) 2016-12-13
US20140113932A1 (en) 2014-04-24
EA026137B1 (ru) 2017-03-31
DOP2013000311A (es) 2014-02-28
US9512118B2 (en) 2016-12-06
EA201490092A1 (ru) 2014-05-30
AU2012274292A1 (en) 2014-01-16
KR20140040777A (ko) 2014-04-03

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20201020