TN2013000510A1 - Crystal of fused heterocyclic compound - Google Patents

Crystal of fused heterocyclic compound

Info

Publication number
TN2013000510A1
TN2013000510A1 TNP2013000510A TN2013000510A TN2013000510A1 TN 2013000510 A1 TN2013000510 A1 TN 2013000510A1 TN P2013000510 A TNP2013000510 A TN P2013000510A TN 2013000510 A TN2013000510 A TN 2013000510A TN 2013000510 A1 TN2013000510 A1 TN 2013000510A1
Authority
TN
Tunisia
Prior art keywords
crystal
heterocyclic compound
fused heterocyclic
imidazo
pyridin
Prior art date
Application number
TNP2013000510A
Other languages
English (en)
Inventor
Katsuhiko Yamamoto
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of TN2013000510A1 publication Critical patent/TN2013000510A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
TNP2013000510A 2011-06-22 2013-12-06 Crystal of fused heterocyclic compound TN2013000510A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2011138920 2011-06-22
PCT/JP2012/066461 WO2012176934A1 (fr) 2011-06-22 2012-06-21 Cristal de composé hétérocyclique condensé

Publications (1)

Publication Number Publication Date
TN2013000510A1 true TN2013000510A1 (en) 2015-03-30

Family

ID=46551819

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2013000510A TN2013000510A1 (en) 2011-06-22 2013-12-06 Crystal of fused heterocyclic compound

Country Status (26)

Country Link
US (1) US9512118B2 (fr)
EP (1) EP2723738B1 (fr)
JP (1) JP6025757B2 (fr)
KR (1) KR20140040777A (fr)
CN (1) CN103608348B (fr)
AR (1) AR087004A1 (fr)
AU (1) AU2012274292B2 (fr)
BR (1) BR112013032052A2 (fr)
CA (1) CA2839825C (fr)
CL (1) CL2013003632A1 (fr)
CO (1) CO6862150A2 (fr)
CR (1) CR20140033A (fr)
DO (1) DOP2013000311A (fr)
EA (1) EA026137B1 (fr)
EC (1) ECSP14013165A (fr)
GE (1) GEP20166475B (fr)
MA (1) MA35274B1 (fr)
MX (1) MX342990B (fr)
MY (1) MY163483A (fr)
PE (1) PE20141030A1 (fr)
TN (1) TN2013000510A1 (fr)
TW (1) TWI570122B (fr)
UA (1) UA112082C2 (fr)
UY (1) UY34150A (fr)
WO (1) WO2012176934A1 (fr)
ZA (1) ZA201309611B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2012124782A1 (fr) * 2011-03-16 2012-09-20 武田薬品工業株式会社 Composé hétérocyclique condensé
US10308626B1 (en) 2018-07-02 2019-06-04 Pratt Bethers Crystal purification in a glass or metal container
US10960322B2 (en) 2018-07-02 2021-03-30 Pratt Bethers Apparatus for purifying crystals using solvent vapors
US10851076B2 (en) 2017-08-10 2020-12-01 Pratt Bethers Method for purifying crystals using solvent vapors

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5597826A (en) * 1994-09-14 1997-01-28 Pfizer Inc. Compositions containing sertraline and a 5-HT1D receptor agonist or antagonist
WO2006038111A1 (fr) * 2004-10-07 2006-04-13 Pfizer Products Inc. Derives de benzoimidazole utiles en tant qu'agents antiproliferatifs
JP5220414B2 (ja) 2005-08-30 2013-06-26 旭化成ファーマ株式会社 スルホンアミド化合物
FI20055498A0 (fi) 2005-09-16 2005-09-16 Biotie Therapies Corp Sulfonamidijohdannaisia
US7618982B2 (en) 2005-12-19 2009-11-17 Nerviano Medical Sciences S.R.L. Heteroarylpyrrolopyridinones active as kinase inhibitors
JP5175228B2 (ja) * 2006-02-15 2013-04-03 サノフイ 新規なアザシクリル置換アリールジヒドロイソキノリノン、それらの製造方法及び薬剤としてそれらの使用
US20080090834A1 (en) 2006-07-06 2008-04-17 Pfizer Inc Selective azole pde10a inhibitor compounds
KR101524817B1 (ko) 2007-04-18 2015-06-01 깃세이 야쿠힌 고교 가부시키가이샤 질소 함유 축합환 유도체, 그것을 함유하는 의약 조성물 및 그 의약 용도
US20110098288A1 (en) 2008-03-11 2011-04-28 Jeremy Major Sulfonamides as zap-70 inhibitors
AR074343A1 (es) 2008-11-14 2011-01-12 Amgen Inc Derivados de piridina y pirimidina como inhibidores de la fosfodiesterasa 10
TWI396689B (zh) 2008-11-14 2013-05-21 Amgen Inc 作為磷酸二酯酶10抑制劑之吡衍生物
WO2010126002A1 (fr) 2009-04-28 2010-11-04 塩野義製薬株式会社 Produit pharmaceutique contenant un composé sulfonamide hétérocyclique
BR112012032087A2 (pt) * 2010-06-24 2016-11-16 Takeda Pharmaceuticals Co composto, medicamento, e, uso de um composto
EP2601192B1 (fr) 2010-08-04 2017-03-01 Takeda Pharmaceutical Company Limited Composés hétérocycliques condensés
EP2604597B1 (fr) 2010-08-10 2017-01-04 Takeda Pharmaceutical Company Limited Composé hétérocyclique et utilisation de celui-ci comme inhibiteur de phosphodiesterase 10a
WO2012124782A1 (fr) 2011-03-16 2012-09-20 武田薬品工業株式会社 Composé hétérocyclique condensé

Also Published As

Publication number Publication date
GEP20166475B (en) 2016-05-10
EP2723738A1 (fr) 2014-04-30
TW201313709A (zh) 2013-04-01
CN103608348A (zh) 2014-02-26
CR20140033A (es) 2014-03-12
UY34150A (es) 2013-01-31
AR087004A1 (es) 2014-02-05
CL2013003632A1 (es) 2014-06-06
ECSP14013165A (es) 2014-02-28
EP2723738B1 (fr) 2018-03-14
ZA201309611B (en) 2014-08-27
JP6025757B2 (ja) 2016-11-16
WO2012176934A1 (fr) 2012-12-27
CN103608348B (zh) 2016-03-30
MX342990B (es) 2016-10-20
EA201490092A1 (ru) 2014-05-30
KR20140040777A (ko) 2014-04-03
AU2012274292A1 (en) 2014-01-16
MX2013015354A (es) 2014-02-11
PE20141030A1 (es) 2014-08-29
EA026137B1 (ru) 2017-03-31
NZ618944A (en) 2015-08-28
TWI570122B (zh) 2017-02-11
UA112082C2 (uk) 2016-07-25
JP2014516918A (ja) 2014-07-17
US20140113932A1 (en) 2014-04-24
DOP2013000311A (es) 2014-02-28
US9512118B2 (en) 2016-12-06
CA2839825A1 (fr) 2012-12-27
MY163483A (en) 2017-09-15
AU2012274292B2 (en) 2016-10-27
CA2839825C (fr) 2019-04-09
CO6862150A2 (es) 2014-02-10
MA35274B1 (fr) 2014-07-03
BR112013032052A2 (pt) 2016-12-13

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