UY31953A - 3-cianopirrolidinil-fenil-oxazolidinonas como agentes antibacterianos - Google Patents

3-cianopirrolidinil-fenil-oxazolidinonas como agentes antibacterianos

Info

Publication number
UY31953A
UY31953A UY0001031953A UY31953A UY31953A UY 31953 A UY31953 A UY 31953A UY 0001031953 A UY0001031953 A UY 0001031953A UY 31953 A UY31953 A UY 31953A UY 31953 A UY31953 A UY 31953A
Authority
UY
Uruguay
Prior art keywords
oxazolidinonas
cianopirrolidinil
fenil
antibacterial agents
formula
Prior art date
Application number
UY0001031953A
Other languages
English (en)
Inventor
Guglietta Antonio
Cano Biosca Montserrat
Palomer Benet Albert
Original Assignee
Ferrer Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40010598&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY31953(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ferrer Int filed Critical Ferrer Int
Publication of UY31953A publication Critical patent/UY31953A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/08—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing alicyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La invención proporciona nuevos compuestos de oxazolidinona de fórmula (I) donde R1, R2 y R3 tienen diferentes significados. También se proporcionan procedimientos de preparación, composiciones farmacéuticas, y usos de los mismos para el tratamiento de infecciones bacterianas.
UY0001031953A 2008-07-01 2009-07-01 3-cianopirrolidinil-fenil-oxazolidinonas como agentes antibacterianos UY31953A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP08159446A EP2141161A1 (en) 2008-07-01 2008-07-01 3-cyanopyrrolidinyl-phenyl-oxazolidinones as antibacterial agents

Publications (1)

Publication Number Publication Date
UY31953A true UY31953A (es) 2010-01-29

Family

ID=40010598

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001031953A UY31953A (es) 2008-07-01 2009-07-01 3-cianopirrolidinil-fenil-oxazolidinonas como agentes antibacterianos

Country Status (23)

Country Link
US (1) US20110152333A1 (es)
EP (2) EP2141161A1 (es)
JP (1) JP2011526589A (es)
KR (1) KR20110036601A (es)
CN (1) CN102112471A (es)
AR (1) AR072389A1 (es)
AT (1) ATE541842T1 (es)
AU (1) AU2009265790A1 (es)
BR (1) BRPI0913842A2 (es)
CA (1) CA2729491A1 (es)
CL (2) CL2009001493A1 (es)
CY (1) CY1112684T1 (es)
DK (1) DK2321306T3 (es)
ES (1) ES2381155T3 (es)
MX (1) MX2011000141A (es)
PE (1) PE20110161A1 (es)
PL (1) PL2321306T3 (es)
PT (1) PT2321306E (es)
RU (1) RU2011103485A (es)
SI (1) SI2321306T1 (es)
TW (1) TW201006828A (es)
UY (1) UY31953A (es)
WO (1) WO2010000703A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101128029B1 (ko) 2010-03-08 2012-03-29 주식회사 레고켐 바이오사이언스 (ｒ)-3-(3-플루오로-4-(1-메틸-5,6-다이하이드로-1,2,4-트리아진-4(1ｈ)-일)페닐)-5-(치환된 메틸)옥사졸리딘-2-온 유도체의 제조방법
US9573910B2 (en) * 2013-11-08 2017-02-21 Lee Pharma Limited Oxazolidinone antibacterial compound

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5688792A (en) 1994-08-16 1997-11-18 Pharmacia & Upjohn Company Substituted oxazine and thiazine oxazolidinone antimicrobials
PT788498E (pt) * 1994-10-26 2002-02-28 Upjohn Co Compostos antimicrobianos de feniloxazolidinona
US7687627B2 (en) * 2003-09-08 2010-03-30 Wockhardt Limited Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy

Also Published As

Publication number Publication date
WO2010000703A1 (en) 2010-01-07
DK2321306T3 (da) 2012-04-10
EP2141161A1 (en) 2010-01-06
CN102112471A (zh) 2011-06-29
BRPI0913842A2 (pt) 2015-10-20
TW201006828A (en) 2010-02-16
JP2011526589A (ja) 2011-10-13
CL2009001493A1 (es) 2009-12-11
SI2321306T1 (sl) 2012-05-31
ATE541842T1 (de) 2012-02-15
RU2011103485A (ru) 2012-08-10
CL2010001589A1 (es) 2011-11-11
CY1112684T1 (el) 2016-02-10
PE20110161A1 (es) 2011-03-15
EP2321306B1 (en) 2012-01-18
US20110152333A1 (en) 2011-06-23
EP2321306A1 (en) 2011-05-18
MX2011000141A (es) 2011-04-05
PT2321306E (pt) 2012-04-13
KR20110036601A (ko) 2011-04-07
ES2381155T3 (es) 2012-05-23
AR072389A1 (es) 2010-08-25
PL2321306T3 (pl) 2012-06-29
CA2729491A1 (en) 2010-01-07
AU2009265790A1 (en) 2010-01-07

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