UY31698A - Preparacion solida de desintegracion oral - Google Patents

Preparacion solida de desintegracion oral

Info

Publication number
UY31698A
UY31698A UY0001031698A UY31698A UY31698A UY 31698 A UY31698 A UY 31698A UY 0001031698 A UY0001031698 A UY 0001031698A UY 31698 A UY31698 A UY 31698A UY 31698 A UY31698 A UY 31698A
Authority
UY
Uruguay
Prior art keywords
oral disintegration
solid preparation
solid oral
fine granules
disintegration preparation
Prior art date
Application number
UY0001031698A
Other languages
English (en)
Inventor
Kurasawa Takashi
Watanabe Yasuko
Omachi Yoshihiro
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40791576&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY31698(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of UY31698A publication Critical patent/UY31698A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A61K9/2081Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Zoology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención provee una preparación sólida de desintegración oral tales como un comprimido producido formando comprimidos los gránulos finos que muestran una liberación controlada de un principio activo para uso faramcéutico y un aditivo, y similares, y la preparación sólida de desintegración oral que contiene gránulos finos recubiertos con una capa de recubrimiento que contiene un polímero que produce una película de recubrimiento que tiene una elongación en la ruptura de alrededor de 100 - alrededor de 700 %.
UY0001031698A 2008-03-11 2009-03-10 Preparacion solida de desintegracion oral UY31698A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2008061673 2008-03-11
JP2008334920 2008-12-26

Publications (1)

Publication Number Publication Date
UY31698A true UY31698A (es) 2009-11-10

Family

ID=40791576

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001031698A UY31698A (es) 2008-03-11 2009-03-10 Preparacion solida de desintegracion oral

Country Status (26)

Country Link
US (2) US9241910B2 (es)
EP (1) EP2254556A2 (es)
JP (1) JP5604304B2 (es)
KR (1) KR20100129761A (es)
CN (2) CN102026627B (es)
AR (1) AR070863A1 (es)
AU (1) AU2009224254A1 (es)
BR (1) BRPI0909439A2 (es)
CA (1) CA2717947C (es)
CL (1) CL2009000557A1 (es)
CO (1) CO6321224A2 (es)
CR (1) CR11709A (es)
DO (1) DOP2010000273A (es)
EA (1) EA021792B1 (es)
EC (1) ECSP10010538A (es)
GE (1) GEP20135845B (es)
IL (1) IL207989A0 (es)
MA (1) MA32174B1 (es)
MX (1) MX2010009824A (es)
MY (1) MY173730A (es)
NZ (1) NZ588407A (es)
PE (2) PE20091620A1 (es)
TW (1) TWI441658B (es)
UY (1) UY31698A (es)
WO (1) WO2009113703A2 (es)
ZA (1) ZA201006679B (es)

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KR102555664B1 (ko) * 2017-02-21 2023-07-18 이에이 파마 가부시키가이샤 과립 제제
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JP2021512924A (ja) * 2018-02-08 2021-05-20 タイワンジェ ファーマシューティカルズ カンパニー リミテッドTaiwanj Pharmaceuticals Co., Ltd. オピオイド受容体拮抗薬の固体剤形の医薬製剤
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GB202001237D0 (en) * 2020-01-29 2020-03-11 Sisteks D O O Granular pharmaceutical product for oral administration from a pre-filled straw and method of manufacturing such pharmaceutical product
CA3168680A1 (en) 2020-01-31 2021-08-05 Nanocopoeia, Llc Amorphous nilotinib microparticles and uses thereof
CA3181361A1 (en) 2020-04-30 2021-11-04 Nanocopoeia, Llc Orally disintegrating tablet comprising amorphous solid dispersion of nilotinib
CN112121067A (zh) * 2020-11-16 2020-12-25 深圳科兴药业有限公司 一种婴儿型双歧杆菌微胶囊及其制备方法
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Also Published As

Publication number Publication date
US20150037423A1 (en) 2015-02-05
KR20100129761A (ko) 2010-12-09
CN102026627A (zh) 2011-04-20
JP5604304B2 (ja) 2014-10-08
AU2009224254A1 (en) 2009-09-17
PE20141034A1 (es) 2014-09-10
GEP20135845B (en) 2013-06-10
DOP2010000273A (es) 2010-09-30
MY173730A (en) 2020-02-18
WO2009113703A3 (en) 2010-06-17
NZ588407A (en) 2012-07-27
US9241910B2 (en) 2016-01-26
AU2009224254A2 (en) 2010-11-18
US20110091563A1 (en) 2011-04-21
CN104127368A (zh) 2014-11-05
CR11709A (es) 2010-11-04
MX2010009824A (es) 2010-09-28
ECSP10010538A (es) 2010-11-30
EP2254556A2 (en) 2010-12-01
CO6321224A2 (es) 2011-09-20
CN102026627B (zh) 2016-10-26
CA2717947C (en) 2020-07-07
AR070863A1 (es) 2010-05-12
MA32174B1 (fr) 2011-03-01
EA021792B1 (ru) 2015-09-30
IL207989A0 (en) 2010-12-30
TWI441658B (zh) 2014-06-21
TW200944249A (en) 2009-11-01
PE20091620A1 (es) 2009-11-12
WO2009113703A2 (en) 2009-09-17
CA2717947A1 (en) 2009-09-17
ZA201006679B (en) 2011-11-30
EA201071054A1 (ru) 2011-04-29
CL2009000557A1 (es) 2010-10-01
BRPI0909439A2 (pt) 2015-12-15
JP2011513204A (ja) 2011-04-28

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