UY30956A1 - Imidazo- y triazolopirimidinas sustituidas - Google Patents

Imidazo- y triazolopirimidinas sustituidas

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Publication number
UY30956A1
UY30956A1 UY30956A UY30956A UY30956A1 UY 30956 A1 UY30956 A1 UY 30956A1 UY 30956 A UY30956 A UY 30956A UY 30956 A UY30956 A UY 30956A UY 30956 A1 UY30956 A1 UY 30956A1
Authority
UY
Uruguay
Prior art keywords
imidazo
substituted
triazolopirimidines
preparation
triazolopyrimidines
Prior art date
Application number
UY30956A
Other languages
English (en)
Inventor
Sperzel Michael
Strayle Jochen
Zubov Dmitry
Rester Ulrich
Heitmeier Stefan
Gnoth Mark Jean
Svenstrup Niels
Rihrig Susanne
Wilmen Andreas
Siegel Stephan
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of UY30956A1 publication Critical patent/UY30956A1/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hematology (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Immunology (AREA)
  • Obesity (AREA)
  • Ophthalmology & Optometry (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)

Abstract

La invencion se refiere a imidazo-y triazolopirimidinas sustituidas, a procedimientos para su preparacion y a su uso para la preparacion de medicamentos para el tratamiento y/o profilaxis de enfermedades, en particular de trastornos hematologicos, preferiblemente de leucopenias y neutropenias.
UY30956A 2007-03-16 2008-03-11 Imidazo- y triazolopirimidinas sustituidas UY30956A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102007012645A DE102007012645A1 (de) 2007-03-16 2007-03-16 Substituierte Imidazo- und Triazolopyrimidine

Publications (1)

Publication Number Publication Date
UY30956A1 true UY30956A1 (es) 2008-10-31

Family

ID=39688187

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30956A UY30956A1 (es) 2007-03-16 2008-03-11 Imidazo- y triazolopirimidinas sustituidas

Country Status (13)

Country Link
US (2) US8273752B2 (es)
EP (1) EP2137188B1 (es)
JP (1) JP5400626B2 (es)
AR (1) AR065719A1 (es)
CA (1) CA2680697C (es)
CL (1) CL2008000703A1 (es)
DE (1) DE102007012645A1 (es)
ES (1) ES2387223T3 (es)
PA (1) PA8772101A1 (es)
PE (1) PE20081806A1 (es)
TW (1) TW200904819A (es)
UY (1) UY30956A1 (es)
WO (1) WO2008113469A2 (es)

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DE102007012645A1 (de) 2007-03-16 2008-09-18 Bayer Healthcare Ag Substituierte Imidazo- und Triazolopyrimidine
DE102008023801A1 (de) * 2008-05-15 2009-11-19 Bayer Schering Pharma Aktiengesellschaft Substituierte Imidazo- und Triazolopyrimidine, Imidazo- und Pyrazolopyrazine und Imidazotriazine
DE102008035552A1 (de) * 2008-07-30 2010-02-04 Bayer Schering Pharma Aktiengesellschaft Substituierte Pyridine und ihre Verwendung
CN102361872B (zh) * 2009-02-13 2014-12-03 拜耳知识产权有限责任公司 作为akt抑制剂的稠合嘧啶
JP5503930B2 (ja) * 2009-09-18 2014-05-28 住友化学株式会社 ３−アミノ−１−ｔｅｒｔ−ブトキシカルボニルピペリジンの精製方法およびそのクエン酸塩
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US8748582B2 (en) 2009-10-15 2014-06-10 Monash University Affinity ligands and methods for protein purification
CA2787714C (en) 2010-01-22 2019-04-09 Joaquin Pastor Fernandez Inhibitors of pi3 kinase
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
WO2011111705A1 (ja) 2010-03-12 2011-09-15 日本曹達株式会社 ｔ－ブトキシカルボニルアミン化合物の製造方法
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TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
AU2011338339A1 (en) 2010-12-08 2013-06-27 Vanderbilt University Bicyclic pyrazole compounds as allosteric modulators of mGluR5 receptors
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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JP2014528475A (ja) * 2011-10-12 2014-10-27 アレイ バイオファーマ、インコーポレイテッド ５，７置換イミダゾ［１，２−ｃ］ピリミジン
LT3105226T (lt) 2014-02-13 2019-11-11 Incyte Corp Ciklopropilaminai, kaip lsd1 inhibitoriai
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WO2015123437A1 (en) 2014-02-13 2015-08-20 Incyte Corporation Cyclopropylamines as lsd1 inhibitors
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