UY30956A1 - Imidazo- y triazolopirimidinas sustituidas - Google Patents
Imidazo- y triazolopirimidinas sustituidasInfo
- Publication number
- UY30956A1 UY30956A1 UY30956A UY30956A UY30956A1 UY 30956 A1 UY30956 A1 UY 30956A1 UY 30956 A UY30956 A UY 30956A UY 30956 A UY30956 A UY 30956A UY 30956 A1 UY30956 A1 UY 30956A1
- Authority
- UY
- Uruguay
- Prior art keywords
- imidazo
- substituted
- triazolopirimidines
- preparation
- triazolopyrimidines
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A—HUMAN NECESSITIES
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Hematology (AREA)
- Virology (AREA)
- Oncology (AREA)
- Cardiology (AREA)
- Communicable Diseases (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Endocrinology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Immunology (AREA)
- Obesity (AREA)
- Ophthalmology & Optometry (AREA)
- Molecular Biology (AREA)
- Pulmonology (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Dermatology (AREA)
- Emergency Medicine (AREA)
- Tropical Medicine & Parasitology (AREA)
Abstract
La invencion se refiere a imidazo-y triazolopirimidinas sustituidas, a procedimientos para su preparacion y a su uso para la preparacion de medicamentos para el tratamiento y/o profilaxis de enfermedades, en particular de trastornos hematologicos, preferiblemente de leucopenias y neutropenias.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102007012645A DE102007012645A1 (de) | 2007-03-16 | 2007-03-16 | Substituierte Imidazo- und Triazolopyrimidine |
Publications (1)
Publication Number | Publication Date |
---|---|
UY30956A1 true UY30956A1 (es) | 2008-10-31 |
Family
ID=39688187
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY30956A UY30956A1 (es) | 2007-03-16 | 2008-03-11 | Imidazo- y triazolopirimidinas sustituidas |
Country Status (13)
Country | Link |
---|---|
US (2) | US8273752B2 (es) |
EP (1) | EP2137188B1 (es) |
JP (1) | JP5400626B2 (es) |
AR (1) | AR065719A1 (es) |
CA (1) | CA2680697C (es) |
CL (1) | CL2008000703A1 (es) |
DE (1) | DE102007012645A1 (es) |
ES (1) | ES2387223T3 (es) |
PA (1) | PA8772101A1 (es) |
PE (1) | PE20081806A1 (es) |
TW (1) | TW200904819A (es) |
UY (1) | UY30956A1 (es) |
WO (1) | WO2008113469A2 (es) |
Families Citing this family (45)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102007012645A1 (de) | 2007-03-16 | 2008-09-18 | Bayer Healthcare Ag | Substituierte Imidazo- und Triazolopyrimidine |
DE102008023801A1 (de) * | 2008-05-15 | 2009-11-19 | Bayer Schering Pharma Aktiengesellschaft | Substituierte Imidazo- und Triazolopyrimidine, Imidazo- und Pyrazolopyrazine und Imidazotriazine |
DE102008035552A1 (de) * | 2008-07-30 | 2010-02-04 | Bayer Schering Pharma Aktiengesellschaft | Substituierte Pyridine und ihre Verwendung |
CN102361872B (zh) * | 2009-02-13 | 2014-12-03 | 拜耳知识产权有限责任公司 | 作为akt抑制剂的稠合嘧啶 |
JP5503930B2 (ja) * | 2009-09-18 | 2014-05-28 | 住友化学株式会社 | 3−アミノ−1−tert−ブトキシカルボニルピペリジンの精製方法およびそのクエン酸塩 |
DK2480546T3 (en) * | 2009-09-24 | 2015-02-02 | Hoffmann La Roche | Imidazopyridine or imidazopyrimidinderivater as phosphodiesterase inhibitors 10A |
US8748582B2 (en) | 2009-10-15 | 2014-06-10 | Monash University | Affinity ligands and methods for protein purification |
CA2787714C (en) | 2010-01-22 | 2019-04-09 | Joaquin Pastor Fernandez | Inhibitors of pi3 kinase |
WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
WO2011111705A1 (ja) | 2010-03-12 | 2011-09-15 | 日本曹達株式会社 | t-ブトキシカルボニルアミン化合物の製造方法 |
UA109131C2 (ru) * | 2010-04-14 | 2015-07-27 | Еррей Біофарма Інк. | 5,7-ЗАМЕЩЕННЫЕ ИМИДАЗО[1,2-c]ПИРИМИДИНЫ КАК ИНГИБИТОРЫ JAK-КИНАЗ |
US20130131057A1 (en) | 2010-05-13 | 2013-05-23 | Centro Nacional De Investigaciones Oncologicas (Cnio | New bicyclic compounds as pi3-k and mtor inhibitors |
WO2011157827A1 (de) | 2010-06-18 | 2011-12-22 | Sanofi | Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen |
US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
AU2011338339A1 (en) | 2010-12-08 | 2013-06-27 | Vanderbilt University | Bicyclic pyrazole compounds as allosteric modulators of mGluR5 receptors |
WO2013037390A1 (en) | 2011-09-12 | 2013-03-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
WO2013045413A1 (en) | 2011-09-27 | 2013-04-04 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
JP2014528475A (ja) * | 2011-10-12 | 2014-10-27 | アレイ バイオファーマ、インコーポレイテッド | 5,7置換イミダゾ[1,2−c]ピリミジン |
LT3105226T (lt) | 2014-02-13 | 2019-11-11 | Incyte Corp | Ciklopropilaminai, kaip lsd1 inhibitoriai |
EP3626713B1 (en) | 2014-02-13 | 2021-09-29 | Incyte Corporation | Cyclopropylamines for use as lsd1 inhibitors |
WO2015123437A1 (en) | 2014-02-13 | 2015-08-20 | Incyte Corporation | Cyclopropylamines as lsd1 inhibitors |
EP3105219B9 (en) | 2014-02-13 | 2018-10-03 | Incyte Corporation | Cyclopropylamines as lsd1 inhibitors |
MY185837A (en) | 2014-03-19 | 2021-06-12 | Boehringer Ingelheim Int | Heteroaryl syk inhibitors |
WO2016007736A1 (en) | 2014-07-10 | 2016-01-14 | Incyte Corporation | Imidazopyrazines as lsd1 inhibitors |
WO2016007722A1 (en) | 2014-07-10 | 2016-01-14 | Incyte Corporation | Triazolopyridines and triazolopyrazines as lsd1 inhibitors |
WO2016007731A1 (en) | 2014-07-10 | 2016-01-14 | Incyte Corporation | Imidazopyridines and imidazopyrazines as lsd1 inhibitors |
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TWI714567B (zh) | 2015-04-03 | 2021-01-01 | 美商英塞特公司 | 作為lsd1抑制劑之雜環化合物 |
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EP0641564A4 (en) * | 1992-05-21 | 1995-05-03 | Yoshitomi Pharmaceutical | OPTICALLY ACTIVE CONDENSED PYRAZOLE COMPOUND FOR THE TREATMENT OF THROMBOCYTOPENIA AND ERYTHROPENIA. |
JP2001302667A (ja) | 2000-04-28 | 2001-10-31 | Bayer Ag | イミダゾピリミジン誘導体およびトリアゾロピリミジン誘導体 |
US20030078232A1 (en) | 2001-08-08 | 2003-04-24 | Elfatih Elzein | Adenosine receptor A3 agonists |
CA2469316A1 (en) * | 2001-12-07 | 2003-06-19 | Vertex Pharmaceuticals, Inc. | Pyrimidine-based compounds useful as gsk-3 inhibitors |
EP1537116B1 (en) * | 2002-09-04 | 2010-06-02 | Schering Corporation | Pyrazolopyrimidines suitable for the treatment of cancer diseases |
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EP1812439B2 (en) | 2004-10-15 | 2017-12-06 | Takeda Pharmaceutical Company Limited | Kinase inhibitors |
DE102007012645A1 (de) | 2007-03-16 | 2008-09-18 | Bayer Healthcare Ag | Substituierte Imidazo- und Triazolopyrimidine |
DE102008023801A1 (de) * | 2008-05-15 | 2009-11-19 | Bayer Schering Pharma Aktiengesellschaft | Substituierte Imidazo- und Triazolopyrimidine, Imidazo- und Pyrazolopyrazine und Imidazotriazine |
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2007
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2008
- 2008-03-04 US US12/529,711 patent/US8273752B2/en not_active Expired - Fee Related
- 2008-03-04 CA CA2680697A patent/CA2680697C/en not_active Expired - Fee Related
- 2008-03-04 WO PCT/EP2008/001682 patent/WO2008113469A2/de active Application Filing
- 2008-03-04 ES ES08716201T patent/ES2387223T3/es active Active
- 2008-03-04 EP EP08716201A patent/EP2137188B1/de not_active Not-in-force
- 2008-03-04 JP JP2009553944A patent/JP5400626B2/ja not_active Expired - Fee Related
- 2008-03-10 PE PE2008000448A patent/PE20081806A1/es not_active Application Discontinuation
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- 2008-03-13 AR ARP080101031A patent/AR065719A1/es unknown
- 2008-03-14 TW TW097108955A patent/TW200904819A/zh unknown
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JP5400626B2 (ja) | 2014-01-29 |
EP2137188A2 (de) | 2009-12-30 |
EP2137188B1 (de) | 2012-06-06 |
CA2680697C (en) | 2016-09-20 |
WO2008113469A8 (de) | 2009-09-24 |
CL2008000703A1 (es) | 2008-09-26 |
US9051323B2 (en) | 2015-06-09 |
CA2680697A1 (en) | 2008-09-25 |
ES2387223T3 (es) | 2012-09-18 |
WO2008113469A3 (de) | 2008-11-13 |
US20100113441A1 (en) | 2010-05-06 |
US8273752B2 (en) | 2012-09-25 |
DE102007012645A1 (de) | 2008-09-18 |
WO2008113469A2 (de) | 2008-09-25 |
PA8772101A1 (es) | 2009-02-09 |
TW200904819A (en) | 2009-02-01 |
JP2010521506A (ja) | 2010-06-24 |
AR065719A1 (es) | 2009-06-24 |
PE20081806A1 (es) | 2009-02-07 |
US20130040946A1 (en) | 2013-02-14 |
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