UY30906A1 - Productos farmaceuticos comprendiendo primer ingrediente activo n-[2-(dietilamino)-n-(2-{[2-(4-hidroxi-2-oxo-2,3-dihidro-1,3-benziotazol-7-il)etil)-3-[2-(1-nafti)etoxi]propanamida o una sal y un segundo seleccionado de un grupo especifico - Google Patents

Productos farmaceuticos comprendiendo primer ingrediente activo n-[2-(dietilamino)-n-(2-{[2-(4-hidroxi-2-oxo-2,3-dihidro-1,3-benziotazol-7-il)etil)-3-[2-(1-nafti)etoxi]propanamida o una sal y un segundo seleccionado de un grupo especifico

Info

Publication number
UY30906A1
UY30906A1 UY30906A UY30906A UY30906A1 UY 30906 A1 UY30906 A1 UY 30906A1 UY 30906 A UY30906 A UY 30906A UY 30906 A UY30906 A UY 30906A UY 30906 A1 UY30906 A1 UY 30906A1
Authority
UY
Uruguay
Prior art keywords
bromide
propanamide
oxo
salt
active ingredient
Prior art date
Application number
UY30906A
Other languages
English (en)
Inventor
Alan Young
Katherine Elisabeth Wiley
David John Nicholls
Stephen Connolly
Elaine Bridget Cadogan
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY30906A1 publication Critical patent/UY30906A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/428Thiazoles condensed with carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Producto farmacéutico comprendiendo primer ingrediente activo N-[2-(Dietilamino)etil]-N-(2.{[2-4-hidroxi-2-oxo-2,3-dihidro-1,3-benzotiazol-7-il)etil]amino}etil)-3-[2-(1-naftil)etoxi]propanamida o una sal y un segundo seleccionado del siguiente grupo. a) agonista de : receptor de glucocorticoides no esteroídico; CCR1; PPARy; b) antioxidante; c) antagonistas de : quimioquinas (no CCR1); CRTh2; receptor de leucotrieno;tromboxano; muscarínico que es bromuro de Aclidinio, Glicopirrolato, bromuro de Oxitropio, Pirezepina, telenzepina, bromuro de tiotropio, bromuro de 3(R)-(2-hidorxi-2,2-ditien-2-ilacetoxi)-1-(3-fenoxipropil)-1-azoniabicilo[2.2.2]octano, bromuro de 3(R)-1-fenetil-3-(9H-xanten-9-caboniloxi)-1-azoniabiciclo[2.2.2]octano o bromuro de azoniabiciclo[2.2.2]actano;un inhibidor de p38; d) corticoesteroide; e) inductor de la Histona-Desacetilasa; f) inhibidores de IKK2; COX; lipoxigenasa; MPO; proteasa; PDE; g) estatina; h) vasodilatador; i) un bloqueador ENAC; y utilizacion en tratamiento de enfermedad respiratoria.
UY30906A 2007-02-08 2008-02-08 Productos farmaceuticos comprendiendo primer ingrediente activo n-[2-(dietilamino)-n-(2-{[2-(4-hidroxi-2-oxo-2,3-dihidro-1,3-benziotazol-7-il)etil)-3-[2-(1-nafti)etoxi]propanamida o una sal y un segundo seleccionado de un grupo especifico UY30906A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0702456.5A GB0702456D0 (en) 2007-02-08 2007-02-08 New combination

Publications (1)

Publication Number Publication Date
UY30906A1 true UY30906A1 (es) 2008-09-30

Family

ID=37898976

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30906A UY30906A1 (es) 2007-02-08 2008-02-08 Productos farmaceuticos comprendiendo primer ingrediente activo n-[2-(dietilamino)-n-(2-{[2-(4-hidroxi-2-oxo-2,3-dihidro-1,3-benziotazol-7-il)etil)-3-[2-(1-nafti)etoxi]propanamida o una sal y un segundo seleccionado de un grupo especifico

Country Status (29)

Country Link
US (2) US20100029732A1 (es)
EP (2) EP2364704A1 (es)
JP (1) JP2010518056A (es)
KR (1) KR20090114391A (es)
CN (1) CN101652137A (es)
AR (1) AR065277A1 (es)
AT (1) ATE520401T1 (es)
AU (1) AU2008212713A1 (es)
BR (1) BRPI0806964A2 (es)
CA (1) CA2675465A1 (es)
CL (1) CL2008000379A1 (es)
CO (1) CO6210723A2 (es)
CY (1) CY1111932T1 (es)
DK (1) DK2117542T3 (es)
EC (1) ECSP099567A (es)
ES (1) ES2368967T3 (es)
GB (1) GB0702456D0 (es)
HR (1) HRP20110695T1 (es)
IL (1) IL199840A0 (es)
MX (1) MX2009007865A (es)
PE (1) PE20081759A1 (es)
PL (1) PL2117542T3 (es)
PT (1) PT2117542E (es)
RS (1) RS51956B (es)
RU (1) RU2009133255A (es)
SI (1) SI2117542T1 (es)
TW (1) TW200843750A (es)
UY (1) UY30906A1 (es)
WO (1) WO2008096111A1 (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200738658A (en) * 2005-08-09 2007-10-16 Astrazeneca Ab Novel compounds
TW200738659A (en) * 2005-08-29 2007-10-16 Astrazeneca Ab Novel compounds
TW200745067A (en) 2006-03-14 2007-12-16 Astrazeneca Ab Novel compounds
TW200825084A (en) 2006-11-14 2008-06-16 Astrazeneca Ab New compounds 521
TW200833670A (en) * 2006-12-20 2008-08-16 Astrazeneca Ab Novel compounds 569
GB0702458D0 (en) 2007-02-08 2007-03-21 Astrazeneca Ab Salts 668
CN102089304A (zh) 2008-05-13 2011-06-08 阿斯利康(瑞典)有限公司 作为m3毒蕈碱性受体拮抗剂的奎宁环衍生物
EP2315589A4 (en) * 2008-05-13 2013-09-11 Astrazeneca Ab PHARMACEUTICAL PRODUCT COMPRISING A MUSCARINIC RECEPTOR ANTAGONIST AND A beta2-ADRENOCEPTOR AGONIST
UY31905A (es) 2008-06-18 2010-01-29 Astrazeneca Ab Derivados de benzoxazinona, procesos de preparación, composiciones farmacéuticas conteniéndolos y aplicaciones.
KR20110022611A (ko) * 2008-06-20 2011-03-07 아스트라제네카 아베 베타2-아드레날린수용체 활성의 조절을 위한, 4-히드록시-2-옥소-2,3-디히드로-1,3-벤조티아졸-7-일 화합물을 포함하는 제약 조성물
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
US9827212B2 (en) 2009-03-18 2017-11-28 The Trustees Of The University Of Pennsylvania Compositions and methods for treating asthma and other lung diseases
JP2012533621A (ja) 2009-07-22 2012-12-27 ピュアテック ベンチャーズ ムスカリン性受容体活性化によって改善される疾患の治療のための方法および組成物
US10265311B2 (en) 2009-07-22 2019-04-23 PureTech Health LLC Methods and compositions for treatment of disorders ameliorated by muscarinic receptor activation
WO2011061527A1 (en) 2009-11-17 2011-05-26 Astrazeneca Ab Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination
MX2017003080A (es) 2014-09-09 2017-11-15 Vectura Ltd Formulacion que comprende glicopirrolato, metodo y aparato.
ES2902139T3 (es) * 2015-05-04 2022-03-25 Astrazeneca Ab Derivados de pirazol útiles como inhibidores de la proteína activadora de 5-lipoxigenasa (FLAP)
CN115581696A (zh) 2018-09-28 2023-01-10 卡鲁娜治疗学有限公司 用于治疗由毒蕈碱受体激活所缓解的障碍的组合物和方法

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ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
CO5300399A1 (es) 2000-02-25 2003-07-31 Astrazeneca Ab Heterocicliocs que contienen nitrogeno, proceso para su preparacion y composiciones farmaceuticas que los contienen
AR028948A1 (es) 2000-06-20 2003-05-28 Astrazeneca Ab Compuestos novedosos
SE0100902D0 (sv) 2001-03-15 2001-03-15 Astrazeneca Ab Compounds
SE0104251D0 (sv) 2001-12-14 2001-12-14 Astrazeneca Ab Novel compounds
SE0301569D0 (sv) 2003-05-27 2003-05-27 Astrazeneca Ab Novel compounds
SA04250253B1 (ar) 2003-08-21 2009-11-10 استرازينيكا ايه بي احماض فينوكسي اسيتيك مستبدلة باعتبارها مركبات صيدلانية لعلاج الامراض التنفسية مثل الربو ومرض الانسداد الرئوي المزمن
SE0302486D0 (sv) 2003-09-18 2003-09-18 Astrazeneca Ab Novel compounds
GB0324790D0 (en) 2003-10-24 2003-11-26 Astrazeneca Ab Amide derivatives
GB0402797D0 (en) * 2004-02-09 2004-03-10 Novartis Ag Organic compounds
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Also Published As

Publication number Publication date
PE20081759A1 (es) 2009-01-31
BRPI0806964A2 (pt) 2014-04-08
RU2009133255A (ru) 2011-03-20
DK2117542T3 (da) 2011-10-31
AU2008212713A1 (en) 2008-08-14
GB0702456D0 (en) 2007-03-21
KR20090114391A (ko) 2009-11-03
CN101652137A (zh) 2010-02-17
JP2010518056A (ja) 2010-05-27
TW200843750A (en) 2008-11-16
RS51956B (en) 2012-02-29
US20100029732A1 (en) 2010-02-04
PL2117542T3 (pl) 2011-12-30
CO6210723A2 (es) 2010-10-20
ATE520401T1 (de) 2011-09-15
EP2117542A1 (en) 2009-11-18
CY1111932T1 (el) 2015-11-04
WO2008096111A1 (en) 2008-08-14
PT2117542E (pt) 2011-10-06
CA2675465A1 (en) 2008-08-14
HRP20110695T1 (hr) 2011-11-30
ECSP099567A (es) 2009-09-29
AR065277A1 (es) 2009-05-27
EP2364704A1 (en) 2011-09-14
US20080242649A1 (en) 2008-10-02
SI2117542T1 (sl) 2011-11-30
IL199840A0 (en) 2010-04-15
EP2117542B1 (en) 2011-08-17
ES2368967T3 (es) 2011-11-24
CL2008000379A1 (es) 2008-10-24
MX2009007865A (es) 2009-07-31

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