HRP20110695T1 - Kombinacije beta-2-adrenoceptorskog agonističkog benzotiazolona - Google Patents

Kombinacije beta-2-adrenoceptorskog agonističkog benzotiazolona Download PDF

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Publication number
HRP20110695T1
HRP20110695T1 HR20110695T HRP20110695T HRP20110695T1 HR P20110695 T1 HRP20110695 T1 HR P20110695T1 HR 20110695 T HR20110695 T HR 20110695T HR P20110695 T HRP20110695 T HR P20110695T HR P20110695 T1 HRP20110695 T1 HR P20110695T1
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Croatia
Prior art keywords
ethyl
active ingredient
preparation
bromide
pharmaceutical product
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HR20110695T
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English (en)
Inventor
Bridget Cadogan Elaine
Connolly Stephen
John Nicholls David
Elisabeth Wiley Katherine
Young Alan
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Astrazeneca Ab
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Publication of HRP20110695T1 publication Critical patent/HRP20110695T1/hr

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/428Thiazoles condensed with carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Farmaceutski proizvod, naznačen time, da sadrži u kombinaciji, prvi aktivni sastojak koji je N-[2-(Dietilamino)etil]-N-(2-{[2-(4-hidroksi-2-okso-2,3-dihidro-1,3-benzotiazol-7-il)etil]amino}etil)-3-[2-(1-naftil)

Claims (8)

1. Farmaceutski proizvod, naznačen time, da sadrži u kombinaciji, prvi aktivni sastojak koji je N-[2-(Dietilamino)etil]-N-(2-{[2-(4-hidroksi-2-okso-2,3-dihidro-1,3-benzotiazol-7-il)etil]amino}etil)-3-[2-(1-naftil)etoksi]propanamid dihidrobromid, te drugi aktivni sastojak koji je muskarinski antagonist koji je aklidinij bromid, glikopirolat, oksitropij bromid, pirenzepin, telenzepin ili tiotropij bromid.
2. Komplet naznačen time, da sadrži: pripravak prvog aktivnog sastojaka koji je N-[2-(Dietilamino)etil]-N-(2-{[2-(4-hidroksi-2-okso-2,3-dihidro-1,3-benzotiazol-7-il)etil]amino}etil)-3-[2-(1-naftil)etoksi]propanamid dihidrobromid, pripravak drugog aktivnog sastojaka koji je muskarinski antagonist kao aklidinij bromid, glikopirolat, oksitropij bromid, pirenzepin, telenzepin ili tiotropij bromid, te proizvoljno, upute za simultano, sekvencijalno ili odvojeno davanje navedenih pripravaka pacijentu kojem oni trebaju.
3. Farmaceutski pripravak, naznačen time, da sadrži, kao mješavinu: prvi aktivni sastojak koji je N-[2-(Dietilamino)etil]-N-(2-{[2-(4-hidroksi-2-okso-2,3-dihidro-1,3-benzotiazol-7-il)etil]amino}etil)-3-[2-(1-naftil)etoksi]propanamid dihidrobromid; drugi aktivni sastojak koji je muskarinski antagonist kao aklidinij bromid, glikopirolat, oksitropij bromid, pirenzepin, telenzepin ili tiotropij bromid; te farmaceutski prihvatljivu pomoćnu tvar, razrjeđivač ili nosač.
4. Farmaceutski proizvod, komplet ili pripravak, prema bilo kojem od prethodnih zahtjeva, naznačen time, da drugi aktivni sastojak je tiotropij bromid.
5. Farmaceutski proizvod, komplet ili pripravak, prema bilo kojem od zahtjeva od 1-4, naznačen time, da se koristi kod liječenja.
6. Uporaba farmaceutskog proizvoda, kompleta ili pripravka, prema bilo kojem od zahtjeva od 1-4, naznačena time, da se upotrebljava za proizvodnju lijeka za liječenje respiratorne bolesti.
7. Farmaceutski proizvod, komplet ili pripravak, prema bilo kojem od zahtjeva od 1-4, naznačena time, da se koristi kod liječenja respiratorne bolesti.
8. Uporaba prema zahtjevu 6 ili 7, naznačena time, da je respiratorna bolest kronična opstruktivna plućna bolest ili astma.
HR20110695T 2007-02-08 2011-09-28 Kombinacije beta-2-adrenoceptorskog agonističkog benzotiazolona HRP20110695T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0702456.5A GB0702456D0 (en) 2007-02-08 2007-02-08 New combination
PCT/GB2008/000386 WO2008096111A1 (en) 2007-02-08 2008-02-06 Combinations of beta- 2 -adrenoceptor agonistic benzothiazolone

Publications (1)

Publication Number Publication Date
HRP20110695T1 true HRP20110695T1 (hr) 2011-11-30

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ID=37898976

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20110695T HRP20110695T1 (hr) 2007-02-08 2011-09-28 Kombinacije beta-2-adrenoceptorskog agonističkog benzotiazolona

Country Status (29)

Country Link
US (2) US20100029732A1 (hr)
EP (2) EP2117542B1 (hr)
JP (1) JP2010518056A (hr)
KR (1) KR20090114391A (hr)
CN (1) CN101652137A (hr)
AR (1) AR065277A1 (hr)
AT (1) ATE520401T1 (hr)
AU (1) AU2008212713A1 (hr)
BR (1) BRPI0806964A2 (hr)
CA (1) CA2675465A1 (hr)
CL (1) CL2008000379A1 (hr)
CO (1) CO6210723A2 (hr)
CY (1) CY1111932T1 (hr)
DK (1) DK2117542T3 (hr)
EC (1) ECSP099567A (hr)
ES (1) ES2368967T3 (hr)
GB (1) GB0702456D0 (hr)
HR (1) HRP20110695T1 (hr)
IL (1) IL199840A0 (hr)
MX (1) MX2009007865A (hr)
PE (1) PE20081759A1 (hr)
PL (1) PL2117542T3 (hr)
PT (1) PT2117542E (hr)
RS (1) RS51956B (hr)
RU (1) RU2009133255A (hr)
SI (1) SI2117542T1 (hr)
TW (1) TW200843750A (hr)
UY (1) UY30906A1 (hr)
WO (1) WO2008096111A1 (hr)

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TW200745067A (en) 2006-03-14 2007-12-16 Astrazeneca Ab Novel compounds
TW200825084A (en) 2006-11-14 2008-06-16 Astrazeneca Ab New compounds 521
TW200833670A (en) 2006-12-20 2008-08-16 Astrazeneca Ab Novel compounds 569
GB0702458D0 (en) 2007-02-08 2007-03-21 Astrazeneca Ab Salts 668
JP4837800B2 (ja) 2008-05-13 2011-12-14 アストラゼネカ・アクチエボラーグ ムスカリンm3受容体アンタゴニストとしてのキヌクリジン誘導体
CA2723909A1 (en) * 2008-05-13 2009-11-19 Richard James Bull Pharmaceutical product comprising a muscarinic receptor antagonist and a beta2-adrenoceptor agonist
KR20110017456A (ko) 2008-06-18 2011-02-21 아스트라제네카 아베 호흡기 장애의 치료를 위한 베타2-아드레날린성 수용체 효능제로서 작용하는 벤족사지논 유도체
CA2727908A1 (en) * 2008-06-20 2009-12-23 Astrazeneca Ab Pharmaceutical composition comprising a 4-hydroxy-2-oxo-2, 3- dihydro-1, 3-benzothiazol-7-yl compound for modulation of beta2-adrenoreceptor activity
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
US9827212B2 (en) 2009-03-18 2017-11-28 The Trustees Of The University Of Pennsylvania Compositions and methods for treating asthma and other lung diseases
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WO2011011060A1 (en) 2009-07-22 2011-01-27 Puretech Ventures Methods and compositions for treatment of disorders ameliorated by muscarinic receptor activation
WO2011061527A1 (en) 2009-11-17 2011-05-26 Astrazeneca Ab Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination
WO2016038116A1 (en) 2014-09-09 2016-03-17 Vectura Limited Formulation comprising glycopyrrolate, method and apparatus
EA032221B1 (ru) * 2015-05-04 2019-04-30 Астразенека Аб Производные пиразола, пригодные в качестве ингибиторов белка, активирующего 5-липоксигеназу (flap)
KR102408292B1 (ko) 2018-09-28 2022-06-10 카루나 세러퓨틱스 인코포레이티드 무스카린성 수용체 활성화에 의해 개선된 장애의 치료를 위한 조성물 및 방법

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Also Published As

Publication number Publication date
ECSP099567A (es) 2009-09-29
US20100029732A1 (en) 2010-02-04
AU2008212713A1 (en) 2008-08-14
PE20081759A1 (es) 2009-01-31
WO2008096111A1 (en) 2008-08-14
MX2009007865A (es) 2009-07-31
RS51956B (en) 2012-02-29
BRPI0806964A2 (pt) 2014-04-08
ATE520401T1 (de) 2011-09-15
RU2009133255A (ru) 2011-03-20
CL2008000379A1 (es) 2008-10-24
US20080242649A1 (en) 2008-10-02
AR065277A1 (es) 2009-05-27
EP2117542B1 (en) 2011-08-17
SI2117542T1 (sl) 2011-11-30
TW200843750A (en) 2008-11-16
PT2117542E (pt) 2011-10-06
JP2010518056A (ja) 2010-05-27
UY30906A1 (es) 2008-09-30
GB0702456D0 (en) 2007-03-21
ES2368967T3 (es) 2011-11-24
CO6210723A2 (es) 2010-10-20
KR20090114391A (ko) 2009-11-03
DK2117542T3 (da) 2011-10-31
CY1111932T1 (el) 2015-11-04
EP2364704A1 (en) 2011-09-14
PL2117542T3 (pl) 2011-12-30
EP2117542A1 (en) 2009-11-18
IL199840A0 (en) 2010-04-15
CA2675465A1 (en) 2008-08-14
CN101652137A (zh) 2010-02-17

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