UA90038C2 - SULFOXIMINE DERIVATIVES AS p38 MAP KINASE INHIBITORS - Google Patents
SULFOXIMINE DERIVATIVES AS p38 MAP KINASE INHIBITORSInfo
- Publication number
- UA90038C2 UA90038C2 UAA200808221A UAA200808221A UA90038C2 UA 90038 C2 UA90038 C2 UA 90038C2 UA A200808221 A UAA200808221 A UA A200808221A UA A200808221 A UAA200808221 A UA A200808221A UA 90038 C2 UA90038 C2 UA 90038C2
- Authority
- UA
- Ukraine
- Prior art keywords
- kinase inhibitors
- map kinase
- sulfoximine derivatives
- regioisomers
- synthesis
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Изобретение также касается способа получения соединений общей формулы (И), их региоизомеров, их таутомерных форм, их фармацевтически приемлемых солей, фармацевтических композиций, которые их содержат, и новых промежуточных соединений, которые используются при их синтезе., (I)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1551MU2005 | 2005-12-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
UA90038C2 true UA90038C2 (en) | 2010-03-25 |
Family
ID=38173564
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA200808221A UA90038C2 (en) | 2005-12-13 | 2006-12-11 | SULFOXIMINE DERIVATIVES AS p38 MAP KINASE INHIBITORS |
Country Status (12)
Country | Link |
---|---|
US (1) | US20100240709A1 (ru) |
EP (1) | EP1971603B1 (ru) |
JP (1) | JP4955698B2 (ru) |
KR (1) | KR101091796B1 (ru) |
AT (1) | ATE549331T1 (ru) |
BR (1) | BRPI0620694A2 (ru) |
CA (1) | CA2633083C (ru) |
EA (1) | EA015497B1 (ru) |
IL (1) | IL191929A0 (ru) |
UA (1) | UA90038C2 (ru) |
WO (1) | WO2007077574A2 (ru) |
ZA (1) | ZA200804858B (ru) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2198710A1 (de) | 2008-12-19 | 2010-06-23 | Bayer CropScience AG | Verwendung von 5-Pyridin-4yl-(1,3)Thiazole zur Bekämpfung phytopathogener Pilze |
EP2917185B1 (en) * | 2012-11-09 | 2017-05-10 | Evotec International GmbH | Sulfoximine substituted quinazolines for pharmaceutical compositions |
KR101742226B1 (ko) | 2015-12-24 | 2017-05-31 | 강원대학교산학협력단 | 신규한 n-이미다졸릴 설폭시민 유도체 및 이의 제조방법 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001074811A2 (en) * | 2000-03-30 | 2001-10-11 | Takeda Chemical Industries, Ltd. | Substituted 1,3-thiazole compounds, their production and use |
-
2006
- 2006-12-11 EA EA200870045A patent/EA015497B1/ru not_active IP Right Cessation
- 2006-12-11 JP JP2008545254A patent/JP4955698B2/ja not_active Expired - Fee Related
- 2006-12-11 US US12/086,282 patent/US20100240709A1/en not_active Abandoned
- 2006-12-11 WO PCT/IN2006/000490 patent/WO2007077574A2/en active Application Filing
- 2006-12-11 EP EP06849043A patent/EP1971603B1/en active Active
- 2006-12-11 UA UAA200808221A patent/UA90038C2/ru unknown
- 2006-12-11 CA CA2633083A patent/CA2633083C/en not_active Expired - Fee Related
- 2006-12-11 AT AT06849043T patent/ATE549331T1/de active
- 2006-12-11 KR KR1020087016767A patent/KR101091796B1/ko not_active IP Right Cessation
- 2006-12-11 BR BRPI0620694-8A patent/BRPI0620694A2/pt not_active IP Right Cessation
-
2008
- 2008-06-03 IL IL191929A patent/IL191929A0/en unknown
- 2008-06-04 ZA ZA200804858A patent/ZA200804858B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
BRPI0620694A2 (pt) | 2012-03-13 |
KR101091796B1 (ko) | 2011-12-08 |
US20100240709A1 (en) | 2010-09-23 |
JP4955698B2 (ja) | 2012-06-20 |
KR20080077280A (ko) | 2008-08-21 |
CA2633083A1 (en) | 2007-07-12 |
EP1971603A2 (en) | 2008-09-24 |
IL191929A0 (en) | 2009-08-03 |
ATE549331T1 (de) | 2012-03-15 |
EA015497B1 (ru) | 2011-08-30 |
WO2007077574A3 (en) | 2007-08-23 |
JP2009519322A (ja) | 2009-05-14 |
ZA200804858B (en) | 2010-10-27 |
EP1971603B1 (en) | 2012-03-14 |
CA2633083C (en) | 2011-02-15 |
EA200870045A1 (ru) | 2009-02-27 |
WO2007077574A8 (en) | 2008-07-24 |
WO2007077574A2 (en) | 2007-07-12 |
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