UA75980C2 - Substituted 4-pheny1-4-[1h-imidazol-2-yl] piperidine derivative for reducing ischaemic damages - Google Patents
Substituted 4-pheny1-4-[1h-imidazol-2-yl] piperidine derivative for reducing ischaemic damages Download PDFInfo
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- UA75980C2 UA75980C2 UA20040503666A UA20040503666A UA75980C2 UA 75980 C2 UA75980 C2 UA 75980C2 UA 20040503666 A UA20040503666 A UA 20040503666A UA 20040503666 A UA20040503666 A UA 20040503666A UA 75980 C2 UA75980 C2 UA 75980C2
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP01203927 | 2001-10-15 | ||
| PCT/EP2002/011371 WO2003039440A2 (en) | 2001-10-15 | 2002-10-10 | Substituted 4-phenyl-4-(1h-imidazol-2-yl)-piperidine derivatives for reducing ischaemic damage |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA75980C2 true UA75980C2 (en) | 2006-06-15 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA20040503666A UA75980C2 (en) | 2001-10-15 | 2002-10-10 | Substituted 4-pheny1-4-[1h-imidazol-2-yl] piperidine derivative for reducing ischaemic damages |
Country Status (27)
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|---|---|
| US (1) | US7390822B2 (es) |
| EP (1) | EP1438049B1 (es) |
| JP (1) | JP4418676B2 (es) |
| KR (1) | KR100967599B1 (es) |
| CN (1) | CN1283252C (es) |
| AR (1) | AR036800A1 (es) |
| AT (1) | ATE345799T1 (es) |
| AU (1) | AU2002363369B2 (es) |
| BR (1) | BR0213325A (es) |
| CA (1) | CA2462374C (es) |
| CY (1) | CY1106335T1 (es) |
| DE (1) | DE60216310T2 (es) |
| EA (1) | EA007657B1 (es) |
| ES (1) | ES2276980T3 (es) |
| HK (1) | HK1072562A1 (es) |
| HR (1) | HRP20040325A2 (es) |
| HU (1) | HUP0402332A3 (es) |
| IL (1) | IL161347A0 (es) |
| MX (1) | MXPA04003480A (es) |
| MY (1) | MY139586A (es) |
| NO (1) | NO20041681L (es) |
| NZ (1) | NZ531733A (es) |
| PL (1) | PL370371A1 (es) |
| PT (1) | PT1438049E (es) |
| UA (1) | UA75980C2 (es) |
| WO (1) | WO2003039440A2 (es) |
| ZA (1) | ZA200402816B (es) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
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| TW200403058A (en) * | 2002-04-19 | 2004-03-01 | Bristol Myers Squibb Co | Heterocyclo inhibitors of potassium channel function |
| AR044010A1 (es) * | 2003-04-11 | 2005-08-24 | Janssen Pharmaceutica Nv | Uso de derivados de 4-fenil-4- [1h-imidazol-2-il]- piperidina sustituidos como agonistas delta opioideos no peptidos selectivos, con actividad antidepresiva y ansiolitica |
| WO2005005478A2 (en) * | 2003-07-02 | 2005-01-20 | Bayer Healthcare Ag | Diagnostics and therapeutics for diseases associated with g protein-coupled opioid receptor; delta 1 (oprd1) |
| WO2005015242A1 (en) * | 2003-08-06 | 2005-02-17 | Bayer Healthcare Ag | Diagnostics and therapeutics for diseases associated with g protein-coupled opioid receptor kappa 1 (opkr1) |
| TW200633990A (en) * | 2004-11-18 | 2006-10-01 | Takeda Pharmaceuticals Co | Amide compound |
| CA2706991A1 (en) * | 2007-11-30 | 2009-06-04 | Bayer Schering Pharma Aktiengesellschaft | Heteroaryl-substituted piperidines |
| DE102009014484A1 (de) | 2009-03-23 | 2010-09-30 | Bayer Schering Pharma Aktiengesellschaft | Substituierte Piperidine |
| DE102009022896A1 (de) | 2009-05-27 | 2010-12-02 | Bayer Schering Pharma Aktiengesellschaft | Substituierte Piperidine |
| DE102009022894A1 (de) | 2009-05-27 | 2010-12-02 | Bayer Schering Pharma Aktiengesellschaft | Substituierte Piperidine |
| DE102009056387B9 (de) * | 2009-10-30 | 2020-05-07 | Osram Opto Semiconductors Gmbh | Kantenemittierender Halbleiterlaser mit einem Phasenstrukturbereich zur Selektion lateraler Lasermoden |
| EP3697410A4 (en) | 2017-10-19 | 2021-08-11 | Amgen Inc. | BENZIMIDAZOLE DERIVATIVES AND THEIR USES |
| CN113209294B (zh) * | 2020-02-05 | 2023-06-13 | 复旦大学 | Dor激动剂在制备对抗肾脏纤维化药物中的应用 |
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| PL185124B1 (pl) | 1995-03-06 | 2003-02-28 | Interneuron Pharmaceuticals | Zastosowanie cytykoliny oraz jej kompozycja do wytwarzania leku przeznaczonego do ochrony tkanki mózgowej |
| ES2251740T3 (es) | 1996-08-23 | 2006-05-01 | Ludwig Institute For Cancer Research | Factor de crecimiento de celulas de endotelio vascular d recombinante (vegf-d). |
| CA2287538A1 (en) | 1997-04-25 | 1998-11-05 | Collateral Therapeutics | Truncated vegf-related proteins |
| US6103722A (en) * | 1997-07-23 | 2000-08-15 | The Medical College Of Wisconsin Research Foundation Inc. | Ischemic preconditioning |
| GB2332373A (en) * | 1997-12-19 | 1999-06-23 | Merck & Co Inc | Treatment of coronary and/or peripheral ischemia using an antithrombotic agent and an angiogenesis promoter |
| JP4601175B2 (ja) | 1998-12-19 | 2010-12-22 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | 抗ヒスタミン性スピロ化合物 |
| EP1038872A1 (en) * | 1999-02-22 | 2000-09-27 | Pfizer Products Inc. | 4-Phenyl-4-heteroarylpiperdine derivatives as opioid receptor ligands |
| US6297256B1 (en) * | 1999-06-15 | 2001-10-02 | Neurogen Corporation | Aryl and heteroaryl substituted pyridino derivatives GABA brain receptor ligands |
| UA76224C2 (en) * | 2001-10-15 | 2006-07-17 | Janssen Pharmaceutica Nv | Substituted 4-phenyl 4-[1h-imidazol-2-yl]-piperidine derivatives and use thereof as selective non-peptide delta-opioid agonists |
| FR2831166B1 (fr) | 2001-10-18 | 2004-02-27 | Sanofi Synthelabo | Aralkyl-tetrahydro-pyridines, leur preparation et compositions pharmaceutiques les contenant |
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2002
- 2002-10-10 PL PL02370371A patent/PL370371A1/xx not_active Application Discontinuation
- 2002-10-10 EA EA200400547A patent/EA007657B1/ru not_active IP Right Cessation
- 2002-10-10 AT AT02799040T patent/ATE345799T1/de active
- 2002-10-10 IL IL16134702A patent/IL161347A0/xx not_active IP Right Cessation
- 2002-10-10 BR BR0213325-3A patent/BR0213325A/pt not_active Application Discontinuation
- 2002-10-10 MX MXPA04003480A patent/MXPA04003480A/es active IP Right Grant
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- 2002-10-10 CA CA2462374A patent/CA2462374C/en not_active Expired - Lifetime
- 2002-10-10 UA UA20040503666A patent/UA75980C2/uk unknown
- 2002-10-10 US US10/492,778 patent/US7390822B2/en not_active Expired - Fee Related
- 2002-10-10 HU HU0402332A patent/HUP0402332A3/hu unknown
- 2002-10-10 ES ES02799040T patent/ES2276980T3/es not_active Expired - Lifetime
- 2002-10-10 KR KR1020047002380A patent/KR100967599B1/ko not_active IP Right Cessation
- 2002-10-10 WO PCT/EP2002/011371 patent/WO2003039440A2/en active IP Right Grant
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- 2002-10-10 CN CNB028202961A patent/CN1283252C/zh not_active Expired - Fee Related
- 2002-10-10 AU AU2002363369A patent/AU2002363369B2/en not_active Ceased
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- 2002-10-11 AR ARP020103836A patent/AR036800A1/es unknown
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2004
- 2004-04-06 HR HR20040325A patent/HRP20040325A2/hr not_active Application Discontinuation
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2005
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2007
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