UA121473C2 - Поліморфна форма [5-фтор-3-({2-[(4-фторбензол)сульфоніл]піридин-3-іл}метил)-2-метиліндол-1-іл]-оцтової кислоти - Google Patents
Поліморфна форма [5-фтор-3-({2-[(4-фторбензол)сульфоніл]піридин-3-іл}метил)-2-метиліндол-1-іл]-оцтової кислоти Download PDFInfo
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- UA121473C2 UA121473C2 UAA201611544A UAA201611544A UA121473C2 UA 121473 C2 UA121473 C2 UA 121473C2 UA A201611544 A UAA201611544 A UA A201611544A UA A201611544 A UAA201611544 A UA A201611544A UA 121473 C2 UA121473 C2 UA 121473C2
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
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- Dermatology (AREA)
- Ophthalmology & Optometry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| GBGB1407807.5A GB201407807D0 (en) | 2014-05-02 | 2014-05-02 | Polymorphic form |
| PCT/GB2015/051289 WO2015166274A1 (en) | 2014-05-02 | 2015-05-01 | Polymorphic form of [5-fluoro-3-({2-[(4-fluorobenzene) sulfonyl]pyridin-3-yl}methyl)-2-methylindol-1-yl]-acetic acid |
Publications (1)
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| UA121473C2 true UA121473C2 (uk) | 2020-06-10 |
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| UAA201611544A UA121473C2 (uk) | 2014-05-02 | 2015-05-01 | Поліморфна форма [5-фтор-3-({2-[(4-фторбензол)сульфоніл]піридин-3-іл}метил)-2-метиліндол-1-іл]-оцтової кислоти |
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| GB201322273D0 (en) | 2013-12-17 | 2014-01-29 | Atopix Therapeutics Ltd | Process |
| GB201407820D0 (en) | 2014-05-02 | 2014-06-18 | Atopix Therapeutics Ltd | Polymorphic form |
| EP3555061B1 (en) | 2016-12-13 | 2023-06-07 | Watson Laboratories Inc. | Solid state forms of apalutamide |
| CN108658858B (zh) * | 2017-06-27 | 2022-02-25 | 上海中西三维药业有限公司 | 一种羟氯喹的制备和精制方法及其硫酸盐的制备方法 |
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| BE790679A (fr) | 1971-11-03 | 1973-04-27 | Ici Ltd | Derives de l'indole |
| DK151884C (da) | 1979-03-07 | 1988-06-13 | Pfizer | Analogifremgangsmaade til fremstilling af 3-(1-imidazolylalkyl)indolderivater eller farmaceutisk acceptable syreadditionssalte deraf |
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| GB8607294D0 (en) | 1985-04-17 | 1986-04-30 | Ici America Inc | Heterocyclic amide derivatives |
| DE3514696A1 (de) | 1985-04-24 | 1986-11-06 | Bayer Ag, 5090 Leverkusen | N-indolylethyl-sulfonsaeureamide, verfahren zu ihrer herstellung und ihre verwendung |
| US5214059A (en) | 1989-07-03 | 1993-05-25 | Hoechst-Roussel Pharmaceuticals Incorporated | 2-(aminoaryl) indoles and indolines as topical antiinflammatory agents for the treatment of skin disorders |
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| SE0202241D0 (sv) | 2002-07-17 | 2002-07-17 | Astrazeneca Ab | Novel Compounds |
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| GB0614068D0 (en) | 2006-07-14 | 2006-08-23 | Glaxo Group Ltd | Compounds |
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| JP2011509991A (ja) | 2008-01-22 | 2011-03-31 | オキサジェン リミテッド | Ｃｒｔｈ２アンタゴニスト活性を有する化合物 |
| JP2011509990A (ja) | 2008-01-22 | 2011-03-31 | オキサジェン リミテッド | Ｃｒｔｈ２アンタゴニスト活性を有する化合物 |
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| GB201121557D0 (en) | 2011-12-15 | 2012-01-25 | Oxagen Ltd | Process |
| EP2790696A1 (en) | 2011-12-16 | 2014-10-22 | Atopix Therapeutics Limited | Combination of crth2 antagonist and a proton pump inhibitor for the treatment of eosinophilic esophagitis |
| GB201322273D0 (en) | 2013-12-17 | 2014-01-29 | Atopix Therapeutics Ltd | Process |
| GB201407820D0 (en) | 2014-05-02 | 2014-06-18 | Atopix Therapeutics Ltd | Polymorphic form |
| GB201407813D0 (en) | 2014-05-02 | 2014-06-18 | Atopix Therapeutics Ltd | Polymorphic form |
-
2014
- 2014-05-02 GB GBGB1407807.5A patent/GB201407807D0/en not_active Ceased
-
2015
- 2015-05-01 UA UAA201611544A patent/UA121473C2/uk unknown
- 2015-05-01 US US15/308,288 patent/US10011584B2/en active Active
- 2015-05-01 RU RU2016141463A patent/RU2751319C2/ru active
- 2015-05-01 JP JP2016565467A patent/JP2017514842A/ja active Pending
- 2015-05-01 WO PCT/GB2015/051289 patent/WO2015166274A1/en not_active Ceased
- 2015-05-01 EP EP15721029.5A patent/EP3137452B1/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| RU2751319C2 (ru) | 2021-07-13 |
| US20170057944A1 (en) | 2017-03-02 |
| RU2016141463A (ru) | 2018-06-05 |
| US10011584B2 (en) | 2018-07-03 |
| GB201407807D0 (en) | 2014-06-18 |
| EP3137452B1 (en) | 2019-12-25 |
| EP3137452A1 (en) | 2017-03-08 |
| RU2016141463A3 (enExample) | 2018-11-06 |
| WO2015166274A1 (en) | 2015-11-05 |
| JP2017514842A (ja) | 2017-06-08 |
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