UA117673C2 - Поліміксини, композиція, спосіб одержання і спосіб застосування (варіанти) - Google Patents

Поліміксини, композиція, спосіб одержання і спосіб застосування (варіанти)

Info

Publication number
UA117673C2
UA117673C2 UAA201507907A UAA201507907A UA117673C2 UA 117673 C2 UA117673 C2 UA 117673C2 UA A201507907 A UAA201507907 A UA A201507907A UA A201507907 A UAA201507907 A UA A201507907A UA 117673 C2 UA117673 C2 UA 117673C2
Authority
UA
Ukraine
Prior art keywords
methods
polymyxins
compositions
making
сн2сн3
Prior art date
Application number
UAA201507907A
Other languages
English (en)
Ukrainian (uk)
Inventor
Сьольві Гуннес
Відар Бьйонстад
Торбен Кох
Клес Меландер
Мартін Монссон
Original Assignee
Кселлія Фармасьютікалз Апс
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Кселлія Фармасьютікалз Апс filed Critical Кселлія Фармасьютікалз Апс
Publication of UA117673C2 publication Critical patent/UA117673C2/uk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/60Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation occurring through the 4-amino group of 2,4-diamino-butanoic acid
    • C07K7/62Polymyxins; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
UAA201507907A 2013-01-11 2014-01-09 Поліміксини, композиція, спосіб одержання і спосіб застосування (варіанти) UA117673C2 (uk)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361751341P 2013-01-11 2013-01-11
US201361904793P 2013-11-15 2013-11-15
PCT/EP2014/050320 WO2014108469A1 (en) 2013-01-11 2014-01-09 Polymyxins, compositions, methods of making and methods of use

Publications (1)

Publication Number Publication Date
UA117673C2 true UA117673C2 (uk) 2018-09-10

Family

ID=50101865

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201507907A UA117673C2 (uk) 2013-01-11 2014-01-09 Поліміксини, композиція, спосіб одержання і спосіб застосування (варіанти)

Country Status (20)

Country Link
US (1) US10640536B2 (OSRAM)
EP (1) EP2943503B1 (OSRAM)
JP (1) JP6316846B2 (OSRAM)
KR (1) KR20150107793A (OSRAM)
CN (1) CN104918951B (OSRAM)
AU (1) AU2014204873B2 (OSRAM)
BR (1) BR112015016548A2 (OSRAM)
CA (1) CA2895910C (OSRAM)
EA (1) EA027067B1 (OSRAM)
ES (1) ES2641017T3 (OSRAM)
HU (1) HUE034562T2 (OSRAM)
IL (1) IL239840A (OSRAM)
MX (1) MX360905B (OSRAM)
PT (1) PT2943503T (OSRAM)
RU (1) RU2015132569A (OSRAM)
SI (1) SI2943503T1 (OSRAM)
TW (1) TWI613219B (OSRAM)
UA (1) UA117673C2 (OSRAM)
WO (1) WO2014108469A1 (OSRAM)
ZA (1) ZA201504565B (OSRAM)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10640536B2 (en) 2013-01-11 2020-05-05 Xellia Pharmaceuticals Aps Polymyxins, compositions, methods of making and methods of use
TW201522364A (zh) * 2013-06-07 2015-06-16 Xellia Pharmaceuticals Aps 黏菌素甲磺酸鈉(cms)之定性方法
CA2949328C (en) * 2014-07-09 2023-01-31 Xellia Pharmaceuticals Aps Low substituted polymyxins and compositions thereof
SG11201702717XA (en) 2014-10-03 2017-04-27 Xellia Pharmaceuticals Aps Compositions
CN106999542B (zh) 2014-10-03 2021-02-02 埃克斯利亚制药有限公司 吸入装置
CN107257803B (zh) 2014-12-16 2021-02-05 上海盟科药业股份有限公司 用于治疗细菌感染的多粘菌素类抗菌剂
FI126143B (en) * 2015-01-15 2016-07-15 Northern Antibiotics Oy Polymyxine derivative and its uses
JP7367950B2 (ja) * 2015-09-29 2023-10-24 モナッシュ ユニバーシティ 抗菌性ポリミキシン誘導体化合物
CN109996806B (zh) * 2016-12-09 2021-11-02 正大天晴药业集团股份有限公司 高效价的多黏菌素e2甲磺酸钠
CN115298198A (zh) 2020-01-21 2022-11-04 上海盟科药业股份有限公司 用于肾相关癌症靶向治疗的新型化合物和组合物

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1062895A (en) 1962-12-13 1967-03-22 Wellcome Found Sulphomethyl derivatives of polymxin
FR1586834A (OSRAM) 1968-02-12 1970-03-06
DE1906699A1 (de) 1968-02-12 1970-02-05 Pfizer Neue Polymyxinderivate und Verfahren zu deren Herstellung
EP0362370A1 (en) * 1988-04-07 1990-04-11 Edward Shanbrom Non-thrombogenic intravascular time release catheter
JP2001505557A (ja) 1996-11-15 2001-04-24 パソジェネシス コーポレイション 肺感染を処置するための、純粋な生物学的活性コリスチン、その成分、およびコリスチン処方物
US5767068A (en) 1997-02-13 1998-06-16 Pathogenesis Corporation Pure biologically active colistin, its components and a colistin formulation for treatment of pulmonary infections
DK1320355T3 (da) 2001-05-18 2006-07-31 Chiron Corp System til administration af en tobramycinformulering
US20040022740A1 (en) 2001-07-10 2004-02-05 Baker William R. Macrolide formulations for inhalation and methods of treatment of endobronchial infections
WO2007049294A1 (en) * 2005-10-28 2007-05-03 Arch Pharmalabs Limited An improved process for preparation of gemcitabine hydrochloride.
WO2008025560A1 (en) 2006-09-01 2008-03-06 Pari Pharma Gmbh Methods for taste masking of nebulised compositions for nasal and pulmonary inhalation therapy
US20080066739A1 (en) 2006-09-20 2008-03-20 Lemahieu Edward Methods and systems of delivering medication via inhalation
WO2012168820A1 (en) 2011-06-08 2012-12-13 Pfizer Inc. Polymyxin derivatives useful as antibacterial agents
US10640536B2 (en) 2013-01-11 2020-05-05 Xellia Pharmaceuticals Aps Polymyxins, compositions, methods of making and methods of use
TW201522364A (zh) 2013-06-07 2015-06-16 Xellia Pharmaceuticals Aps 黏菌素甲磺酸鈉(cms)之定性方法
CA2949328C (en) 2014-07-09 2023-01-31 Xellia Pharmaceuticals Aps Low substituted polymyxins and compositions thereof
SG11201702717XA (en) 2014-10-03 2017-04-27 Xellia Pharmaceuticals Aps Compositions

Also Published As

Publication number Publication date
IL239840A (en) 2017-09-28
US20160002296A1 (en) 2016-01-07
PT2943503T (pt) 2017-09-28
JP6316846B2 (ja) 2018-04-25
EA027067B1 (ru) 2017-06-30
BR112015016548A2 (pt) 2017-07-11
SI2943503T1 (sl) 2017-11-30
EP2943503B1 (en) 2017-08-23
MX360905B (es) 2018-11-21
TWI613219B (zh) 2018-02-01
EP2943503A1 (en) 2015-11-18
CN104918951A (zh) 2015-09-16
US10640536B2 (en) 2020-05-05
MX2015008878A (es) 2015-10-30
CA2895910C (en) 2021-12-21
ZA201504565B (en) 2016-11-30
WO2014108469A1 (en) 2014-07-17
IL239840A0 (en) 2015-08-31
AU2014204873A1 (en) 2015-07-09
ES2641017T3 (es) 2017-11-07
KR20150107793A (ko) 2015-09-23
RU2015132569A (ru) 2017-02-14
AU2014204873B2 (en) 2017-07-06
CA2895910A1 (en) 2014-07-17
TW201429995A (zh) 2014-08-01
EA201591280A1 (ru) 2015-12-30
HUE034562T2 (en) 2018-03-28
JP2016505007A (ja) 2016-02-18
CN104918951B (zh) 2018-03-30

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