TWI767937B - 外核苷酸酶抑制劑及其使用方法 - Google Patents
外核苷酸酶抑制劑及其使用方法 Download PDFInfo
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- TWI767937B TWI767937B TW106130807A TW106130807A TWI767937B TW I767937 B TWI767937 B TW I767937B TW 106130807 A TW106130807 A TW 106130807A TW 106130807 A TW106130807 A TW 106130807A TW I767937 B TWI767937 B TW I767937B
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| KR102638592B1 (ko) * | 2016-12-22 | 2024-02-19 | 안텐진 테라퓨틱스 리미티드 | 엑토뉴클레오티다제 억제제 및 이의 용도 |
| WO2018208980A1 (en) | 2017-05-10 | 2018-11-15 | Oric Pharmaceuticals, Inc. | Cd73 inhibitors |
| EP3622092A4 (en) * | 2017-05-11 | 2021-06-23 | The Broad Institute, Inc. | METHODS AND COMPOSITIONS OF USE OF CD8 + TUMOR-INFILTRATING LYMPHOCYTE SUBTYPES AND GENE SIGNATURES THEREOF |
| US11377469B2 (en) | 2017-11-03 | 2022-07-05 | Oric Pharmaceuticals, Inc. | CD73 inhibitors |
| IL304348B2 (en) | 2018-04-30 | 2024-08-01 | Oric Pharmaceuticals Inc | CD73 inhibitors |
| WO2019232319A1 (en) | 2018-05-31 | 2019-12-05 | Peloton Therapeutics, Inc. | Compositions and methods for inhibiting cd73 |
| SG11202012001YA (en) * | 2018-06-21 | 2021-01-28 | Calithera Biosciences Inc | Ectonucleotidase inhibitors and methods of use thereof |
| CN112638389A (zh) * | 2018-08-28 | 2021-04-09 | 江苏恒瑞医药股份有限公司 | Cd73抑制剂及其治疗用途 |
| MX2021002878A (es) | 2018-09-11 | 2021-08-16 | Risen Suzhou Pharma Tech Co Ltd | Inhibidores de cd73 y usos farmaceuticos de los mismos. |
| US11530234B2 (en) | 2018-09-11 | 2022-12-20 | Risen (Suzhou) Pharma Tech Co., Ltd. | CD73 inhibitors and pharmaceutical uses thereof |
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| WO2020190073A1 (ko) * | 2019-03-20 | 2020-09-24 | 한국화학연구원 | 신규한 아졸로피리미딘 헤테로고리 화합물을 유효 성분으로 함유하는 약제학적 조성물 |
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| PL4051688T3 (pl) * | 2019-10-30 | 2025-09-22 | Oric Pharmaceuticals, Inc. | Inhibitory cd73 |
| AU2021341258A1 (en) * | 2020-09-08 | 2023-04-13 | Betta Pharmaceuticals Co., Ltd. | CD73 inhibitor and application thereof in medicine |
| CN114099698B (zh) * | 2021-11-26 | 2024-02-09 | 山东大学齐鲁医院 | 一种pH敏感脂质体及其制备方法与应用 |
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| CN115611954A (zh) * | 2022-12-19 | 2023-01-17 | 天津奥瑞芙生物医药有限公司 | 一种5′-o-(4,4′-二甲氧基三苯甲基)-核苷的制备方法 |
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| WO2025162964A1 (en) | 2024-01-30 | 2025-08-07 | Institut National de la Santé et de la Recherche Médicale | Methods for the treatment of endometriosis |
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| KR102638592B1 (ko) | 2016-12-22 | 2024-02-19 | 안텐진 테라퓨틱스 리미티드 | 엑토뉴클레오티다제 억제제 및 이의 용도 |
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| WO2004096233A2 (en) * | 2003-04-25 | 2004-11-11 | Gilead Sciences, Inc. | Nucleoside phosphonate conjugates |
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| CN110234656A (zh) | 2019-09-13 |
| WO2018049145A1 (en) | 2018-03-15 |
| US10472364B2 (en) | 2019-11-12 |
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| JP7125144B2 (ja) | 2022-08-24 |
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| US20180072742A1 (en) | 2018-03-15 |
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| US20200087310A1 (en) | 2020-03-19 |
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| EP3510040A1 (en) | 2019-07-17 |
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