TWI659019B - 吡唑醯胺衍生物 - Google Patents

吡唑醯胺衍生物 Download PDF

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Publication number
TWI659019B
TWI659019B TW104106256A TW104106256A TWI659019B TW I659019 B TWI659019 B TW I659019B TW 104106256 A TW104106256 A TW 104106256A TW 104106256 A TW104106256 A TW 104106256A TW I659019 B TWI659019 B TW I659019B
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Taiwan
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alkyl
substituted
groups
group
mmol
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TW104106256A
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Chinese (zh)
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TW201623236A (zh
Inventor
希拉瑞 貝克
修恩 布克
哈沃德 布萊格曼
維克多 希
納格斯瑞 恰卡
堤蒙西 康辛
歐雷格 艾普斯坦
布萊恩 福斯
史蒂芬妮 吉恩斯梅爾
郝小林
日比谷健太
平田潤
花子皓
傑森 胡曼
角田真二
派翠西亞 羅培茲
中島良太
岡田和久
史蒂芬 歐森
大野裕之
路易士 潘寧頓
佐佐木浩介
嶋田啓子
永淑 申
雷恩 懷特
雷恩 渥茲
易姝燕
曉媚 鄭
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日商帝人製藥股份有限公司
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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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  • Chemical & Material Sciences (AREA)
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  • Diabetes (AREA)
  • Transplantation (AREA)
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  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
TW104106256A 2014-02-28 2015-02-26 吡唑醯胺衍生物 TWI659019B (zh)

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