TWI617563B - 用於由４－氯－２，５－二甲氧基嘧啶製備２－胺基－５，８－二甲氧基［１，２，４］三唑并［１，５－ｃ］嘧啶的方法 - Google Patents

用於由４－氯－２，５－二甲氧基嘧啶製備２－胺基－５，８－二甲氧基［１，２，４］三唑并［１，５－ｃ］嘧啶的方法 Download PDF

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Publication number
TWI617563B
TWI617563B TW102133212A TW102133212A TWI617563B TW I617563 B TWI617563 B TW I617563B TW 102133212 A TW102133212 A TW 102133212A TW 102133212 A TW102133212 A TW 102133212A TW I617563 B TWI617563 B TW I617563B
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TW
Taiwan
Prior art keywords
dialkoxy
pyrimidine
amino
triazolo
salt
Prior art date
Application number
TW102133212A
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English (en)
Chinese (zh)
Other versions
TW201414739A (zh
Inventor
道格拉斯Ｃ 布蘭德
葛雷 羅斯
克雷格 博特
克里斯多弗Ｔ 漢米爾頓
約瑟夫 紐曼
Original Assignee
陶氏農業科學公司
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Filing date
Publication date
Application filed by 陶氏農業科學公司 filed Critical 陶氏農業科學公司
Publication of TW201414739A publication Critical patent/TW201414739A/zh
Application granted granted Critical
Publication of TWI617563B publication Critical patent/TWI617563B/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08F—MACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F10/00—Homopolymers and copolymers of unsaturated aliphatic hydrocarbons having only one carbon-to-carbon double bond
    • C08F10/04—Monomers containing three or four carbon atoms
    • C08F10/06—Propene
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08F—MACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F4/00—Polymerisation catalysts
    • C08F4/42—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors
    • C08F4/44—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors selected from light metals, zinc, cadmium, mercury, copper, silver, gold, boron, gallium, indium, thallium, rare earths or actinides
    • C08F4/60—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors selected from light metals, zinc, cadmium, mercury, copper, silver, gold, boron, gallium, indium, thallium, rare earths or actinides together with refractory metals, iron group metals, platinum group metals, manganese, rhenium technetium or compounds thereof
    • C08F4/62—Refractory metals or compounds thereof
    • C08F4/64—Titanium, zirconium, hafnium or compounds thereof
    • C08F4/65—Pretreating the metal or compound covered by group C08F4/64 before the final contacting with the metal or compound covered by group C08F4/44
    • C08F4/651—Pretreating with non-metals or metal-free compounds
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08F—MACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F4/00—Polymerisation catalysts
    • C08F4/42—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors
    • C08F4/44—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors selected from light metals, zinc, cadmium, mercury, copper, silver, gold, boron, gallium, indium, thallium, rare earths or actinides
    • C08F4/60—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors selected from light metals, zinc, cadmium, mercury, copper, silver, gold, boron, gallium, indium, thallium, rare earths or actinides together with refractory metals, iron group metals, platinum group metals, manganese, rhenium technetium or compounds thereof
    • C08F4/62—Refractory metals or compounds thereof
    • C08F4/64—Titanium, zirconium, hafnium or compounds thereof
    • C08F4/65—Pretreating the metal or compound covered by group C08F4/64 before the final contacting with the metal or compound covered by group C08F4/44
    • C08F4/652—Pretreating with metals or metal-containing compounds
    • C08F4/657—Pretreating with metals or metal-containing compounds with metals or metal-containing compounds, not provided for in groups C08F4/653 - C08F4/656

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
TW102133212A 2012-09-14 2013-09-13 用於由４－氯－２，５－二甲氧基嘧啶製備２－胺基－５，８－二甲氧基［１，２，４］三唑并［１，５－ｃ］嘧啶的方法 TWI617563B (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261701250P 2012-09-14 2012-09-14
US61/701,250 2012-09-14

Publications (2)

Publication Number Publication Date
TW201414739A TW201414739A (zh) 2014-04-16
TWI617563B true TWI617563B (zh) 2018-03-11

Family

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Family Applications (1)

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TW102133212A TWI617563B (zh) 2012-09-14 2013-09-13 用於由４－氯－２，５－二甲氧基嘧啶製備２－胺基－５，８－二甲氧基［１，２，４］三唑并［１，５－ｃ］嘧啶的方法

Country Status (20)

Country Link
US (1) US9000160B2 (enExample)
EP (1) EP2895486B1 (enExample)
JP (1) JP6293758B2 (enExample)
KR (1) KR20150056590A (enExample)
CN (1) CN104768953A (enExample)
AR (1) AR092563A1 (enExample)
AU (1) AU2013315734B2 (enExample)
BR (1) BR102013023482A8 (enExample)
CA (1) CA2884106A1 (enExample)
HK (1) HK1212334A1 (enExample)
IL (1) IL237677B (enExample)
IN (1) IN2015DN01972A (enExample)
MX (1) MX2015003314A (enExample)
NZ (1) NZ705676A (enExample)
PL (1) PL2895486T3 (enExample)
PY (2) PY1342185A (enExample)
RU (1) RU2635352C2 (enExample)
TW (1) TWI617563B (enExample)
UY (1) UY35034A (enExample)
WO (1) WO2014043087A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112730689B (zh) * 2020-12-29 2023-04-07 营口昌成新材料科技有限公司 2-氨基-5,8-二甲氧基[1,2,4]三唑并[1,5-c]嘧啶液相色谱分析方法
CN115417875B (zh) * 2022-09-19 2024-05-31 山东华升新材料有限公司 一种5,8-二甲氧基-[1,2,4]三唑并[1,5-c]嘧啶-2-胺的合成方法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011149861A1 (en) * 2010-05-25 2011-12-01 Dow Agrosciences Llc Process for the preparation of 5-substituted-8-alkoxy[1,2,4]triazolo[1,5-c]pyrimidin-2-amines

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE122009000052I2 (de) 1996-09-24 2009-12-31 Dow Agrosciences Llc N-((1,2,4)triazoloazinyl)benzolsulfonamid- und pyridinsulfonamidverbindungen und deren verwendung als herbizide
ATE261971T1 (de) 2000-06-16 2004-04-15 Dow Agrosciences Llc Verfahren zur herstellung von 2-amino-5,8- dimethoxy(1,2,4)triazolo(1,5-c)pyrimidine

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011149861A1 (en) * 2010-05-25 2011-12-01 Dow Agrosciences Llc Process for the preparation of 5-substituted-8-alkoxy[1,2,4]triazolo[1,5-c]pyrimidin-2-amines

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
Bell et al., "Application of the tisler triazolopyrimidine cyclization to the synthesis of a crop protection agent and an intermediate", Organic Process Research & Development, 2006, 10(6), pp 1167-1171. *

Also Published As

Publication number Publication date
PL2895486T3 (pl) 2018-08-31
AU2013315734A1 (en) 2015-03-26
IL237677B (en) 2018-07-31
BR102013023482A2 (pt) 2015-08-11
PY1342186A (es) 2016-09-01
TW201414739A (zh) 2014-04-16
US9000160B2 (en) 2015-04-07
BR102013023482A8 (pt) 2016-07-12
EP2895486A1 (en) 2015-07-22
CA2884106A1 (en) 2014-03-20
RU2015113560A (ru) 2016-11-10
IN2015DN01972A (enExample) 2015-08-14
JP6293758B2 (ja) 2018-03-14
AU2013315734B2 (en) 2016-03-17
HK1212334A1 (en) 2016-06-10
EP2895486B1 (en) 2018-03-07
US20140081023A1 (en) 2014-03-20
EP2895486A4 (en) 2016-01-27
AR092563A1 (es) 2015-04-22
RU2635352C2 (ru) 2017-11-13
NZ705676A (en) 2016-10-28
KR20150056590A (ko) 2015-05-26
IL237677A0 (en) 2015-04-30
CN104768953A (zh) 2015-07-08
MX2015003314A (es) 2016-01-20
WO2014043087A1 (en) 2014-03-20
UY35034A (es) 2014-04-30
PY1342185A (es) 2016-12-01
JP2015531783A (ja) 2015-11-05

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