JP6293758B2 - ４−クロロ−２，５−ジメトキシピリミジンから２−アミノ−５，８−ジメトキシ［１，２，４］トリアゾロ［１，５−ｃ］ピリミジンを調製するための方法 - Google Patents
４−クロロ−２，５−ジメトキシピリミジンから２−アミノ−５，８−ジメトキシ［１，２，４］トリアゾロ［１，５−ｃ］ピリミジンを調製するための方法 Download PDFInfo
- Publication number
- JP6293758B2 JP6293758B2 JP2015531996A JP2015531996A JP6293758B2 JP 6293758 B2 JP6293758 B2 JP 6293758B2 JP 2015531996 A JP2015531996 A JP 2015531996A JP 2015531996 A JP2015531996 A JP 2015531996A JP 6293758 B2 JP6293758 B2 JP 6293758B2
- Authority
- JP
- Japan
- Prior art keywords
- dialkoxy
- salt
- triazolo
- amino
- pyrimidine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08F—MACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
- C08F10/00—Homopolymers and copolymers of unsaturated aliphatic hydrocarbons having only one carbon-to-carbon double bond
- C08F10/04—Monomers containing three or four carbon atoms
- C08F10/06—Propene
-
- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08F—MACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
- C08F4/00—Polymerisation catalysts
- C08F4/42—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors
- C08F4/44—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors selected from light metals, zinc, cadmium, mercury, copper, silver, gold, boron, gallium, indium, thallium, rare earths or actinides
- C08F4/60—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors selected from light metals, zinc, cadmium, mercury, copper, silver, gold, boron, gallium, indium, thallium, rare earths or actinides together with refractory metals, iron group metals, platinum group metals, manganese, rhenium technetium or compounds thereof
- C08F4/62—Refractory metals or compounds thereof
- C08F4/64—Titanium, zirconium, hafnium or compounds thereof
- C08F4/65—Pretreating the metal or compound covered by group C08F4/64 before the final contacting with the metal or compound covered by group C08F4/44
- C08F4/651—Pretreating with non-metals or metal-free compounds
-
- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08F—MACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
- C08F4/00—Polymerisation catalysts
- C08F4/42—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors
- C08F4/44—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors selected from light metals, zinc, cadmium, mercury, copper, silver, gold, boron, gallium, indium, thallium, rare earths or actinides
- C08F4/60—Metals; Metal hydrides; Metallo-organic compounds; Use thereof as catalyst precursors selected from light metals, zinc, cadmium, mercury, copper, silver, gold, boron, gallium, indium, thallium, rare earths or actinides together with refractory metals, iron group metals, platinum group metals, manganese, rhenium technetium or compounds thereof
- C08F4/62—Refractory metals or compounds thereof
- C08F4/64—Titanium, zirconium, hafnium or compounds thereof
- C08F4/65—Pretreating the metal or compound covered by group C08F4/64 before the final contacting with the metal or compound covered by group C08F4/44
- C08F4/652—Pretreating with metals or metal-containing compounds
- C08F4/657—Pretreating with metals or metal-containing compounds with metals or metal-containing compounds, not provided for in groups C08F4/653 - C08F4/656
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261701250P | 2012-09-14 | 2012-09-14 | |
| US61/701,250 | 2012-09-14 | ||
| PCT/US2013/058941 WO2014043087A1 (en) | 2012-09-14 | 2013-09-10 | Process for the preparation of 2-amino-5,8-dimethoxy[1,2,4]triazolo[1,5-c]pyrimidine from 4-chloro-2,5-dimethoxypyrimidine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2015531783A JP2015531783A (ja) | 2015-11-05 |
| JP6293758B2 true JP6293758B2 (ja) | 2018-03-14 |
Family
ID=50275133
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015531996A Active JP6293758B2 (ja) | 2012-09-14 | 2013-09-10 | ４−クロロ−２，５−ジメトキシピリミジンから２−アミノ−５，８−ジメトキシ［１，２，４］トリアゾロ［１，５−ｃ］ピリミジンを調製するための方法 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US9000160B2 (enExample) |
| EP (1) | EP2895486B1 (enExample) |
| JP (1) | JP6293758B2 (enExample) |
| KR (1) | KR20150056590A (enExample) |
| CN (1) | CN104768953A (enExample) |
| AR (1) | AR092563A1 (enExample) |
| AU (1) | AU2013315734B2 (enExample) |
| BR (1) | BR102013023482A8 (enExample) |
| CA (1) | CA2884106A1 (enExample) |
| HK (1) | HK1212334A1 (enExample) |
| IL (1) | IL237677B (enExample) |
| IN (1) | IN2015DN01972A (enExample) |
| MX (1) | MX2015003314A (enExample) |
| NZ (1) | NZ705676A (enExample) |
| PL (1) | PL2895486T3 (enExample) |
| PY (2) | PY1342185A (enExample) |
| RU (1) | RU2635352C2 (enExample) |
| TW (1) | TWI617563B (enExample) |
| UY (1) | UY35034A (enExample) |
| WO (1) | WO2014043087A1 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112730689B (zh) * | 2020-12-29 | 2023-04-07 | 营口昌成新材料科技有限公司 | 2-氨基-5,8-二甲氧基[1,2,4]三唑并[1,5-c]嘧啶液相色谱分析方法 |
| CN115417875B (zh) * | 2022-09-19 | 2024-05-31 | 山东华升新材料有限公司 | 一种5,8-二甲氧基-[1,2,4]三唑并[1,5-c]嘧啶-2-胺的合成方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE122009000052I2 (de) | 1996-09-24 | 2009-12-31 | Dow Agrosciences Llc | N-((1,2,4)triazoloazinyl)benzolsulfonamid- und pyridinsulfonamidverbindungen und deren verwendung als herbizide |
| ATE261971T1 (de) | 2000-06-16 | 2004-04-15 | Dow Agrosciences Llc | Verfahren zur herstellung von 2-amino-5,8- dimethoxy(1,2,4)triazolo(1,5-c)pyrimidine |
| ES2528145T3 (es) * | 2010-05-25 | 2015-02-04 | Dow Agrosciences Llc | Procedimiento para la preparación de 8-alcoxi[1,2,4]triazolo[1,5-c]pirimidin-2-aminas 5-sustituidas |
-
2013
- 2013-09-10 IN IN1972DEN2015 patent/IN2015DN01972A/en unknown
- 2013-09-10 US US14/022,766 patent/US9000160B2/en active Active
- 2013-09-10 AU AU2013315734A patent/AU2013315734B2/en not_active Ceased
- 2013-09-10 KR KR1020157009142A patent/KR20150056590A/ko not_active Withdrawn
- 2013-09-10 CN CN201380058711.8A patent/CN104768953A/zh active Pending
- 2013-09-10 HK HK16100133.0A patent/HK1212334A1/xx unknown
- 2013-09-10 NZ NZ705676A patent/NZ705676A/en not_active IP Right Cessation
- 2013-09-10 JP JP2015531996A patent/JP6293758B2/ja active Active
- 2013-09-10 CA CA2884106A patent/CA2884106A1/en not_active Abandoned
- 2013-09-10 EP EP13837178.6A patent/EP2895486B1/en active Active
- 2013-09-10 MX MX2015003314A patent/MX2015003314A/es unknown
- 2013-09-10 RU RU2015113560A patent/RU2635352C2/ru not_active IP Right Cessation
- 2013-09-10 PL PL13837178T patent/PL2895486T3/pl unknown
- 2013-09-10 WO PCT/US2013/058941 patent/WO2014043087A1/en not_active Ceased
- 2013-09-12 BR BR102013023482A patent/BR102013023482A8/pt not_active Application Discontinuation
- 2013-09-13 PY PY201301342185A patent/PY1342185A/es unknown
- 2013-09-13 PY PY201301342186A patent/PY1342186A/es unknown
- 2013-09-13 TW TW102133212A patent/TWI617563B/zh not_active IP Right Cessation
- 2013-09-13 UY UY0001035034A patent/UY35034A/es not_active Application Discontinuation
- 2013-09-13 AR ARP130103289A patent/AR092563A1/es unknown
-
2015
- 2015-03-11 IL IL237677A patent/IL237677B/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| PL2895486T3 (pl) | 2018-08-31 |
| AU2013315734A1 (en) | 2015-03-26 |
| IL237677B (en) | 2018-07-31 |
| BR102013023482A2 (pt) | 2015-08-11 |
| PY1342186A (es) | 2016-09-01 |
| TW201414739A (zh) | 2014-04-16 |
| US9000160B2 (en) | 2015-04-07 |
| BR102013023482A8 (pt) | 2016-07-12 |
| EP2895486A1 (en) | 2015-07-22 |
| CA2884106A1 (en) | 2014-03-20 |
| RU2015113560A (ru) | 2016-11-10 |
| IN2015DN01972A (enExample) | 2015-08-14 |
| TWI617563B (zh) | 2018-03-11 |
| AU2013315734B2 (en) | 2016-03-17 |
| HK1212334A1 (en) | 2016-06-10 |
| EP2895486B1 (en) | 2018-03-07 |
| US20140081023A1 (en) | 2014-03-20 |
| EP2895486A4 (en) | 2016-01-27 |
| AR092563A1 (es) | 2015-04-22 |
| RU2635352C2 (ru) | 2017-11-13 |
| NZ705676A (en) | 2016-10-28 |
| KR20150056590A (ko) | 2015-05-26 |
| IL237677A0 (en) | 2015-04-30 |
| CN104768953A (zh) | 2015-07-08 |
| MX2015003314A (es) | 2016-01-20 |
| WO2014043087A1 (en) | 2014-03-20 |
| UY35034A (es) | 2014-04-30 |
| PY1342185A (es) | 2016-12-01 |
| JP2015531783A (ja) | 2015-11-05 |
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