TWI428325B - 製備吡唑羧醯胺之方法 - Google Patents

製備吡唑羧醯胺之方法 Download PDF

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Publication number
TWI428325B
TWI428325B TW100113507A TW100113507A TWI428325B TW I428325 B TWI428325 B TW I428325B TW 100113507 A TW100113507 A TW 100113507A TW 100113507 A TW100113507 A TW 100113507A TW I428325 B TWI428325 B TW I428325B
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TW
Taiwan
Prior art keywords
formula
compound
chloro
palladium
reacting
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TW100113507A
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English (en)
Chinese (zh)
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TW201204704A (en
Inventor
瑞菲爾 督門尤尼爾
浮羅倫 史雷斯
湯瑪斯 凡特吉
麥可 羅摩
史帝芬 崔
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先正達合夥公司
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Publication of TW201204704A publication Critical patent/TW201204704A/zh
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Publication of TWI428325B publication Critical patent/TWI428325B/zh

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/23Preparation of halogenated hydrocarbons by dehalogenation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/26Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/30Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by a Diels-Alder synthesis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/04Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups
    • C07C209/06Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms
    • C07C209/10Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms with formation of amino groups bound to carbon atoms of six-membered aromatic rings or from amines having nitrogen atoms bound to carbon atoms of six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/24Halogenated aromatic hydrocarbons with unsaturated side chains
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C29/00Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
    • C07C29/132Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C35/00Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C35/48Halogenated derivatives
    • C07C35/52Alcohols with a condensed ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/27Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
    • C07C45/29Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D303/00Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02Compounds containing oxirane rings
    • C07D303/12Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/16Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by esterified hydroxyl radicals
    • C07D303/17Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by esterified hydroxyl radicals containing oxirane rings condensed with carbocyclic ring systems having three or more relevant rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/56Ring systems containing bridged rings
    • C07C2603/58Ring systems containing bridged rings containing three rings
    • C07C2603/60Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Epoxy Compounds (AREA)
TW100113507A 2010-04-20 2011-04-19 製備吡唑羧醯胺之方法 TWI428325B (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP10160438 2010-04-20

Publications (2)

Publication Number Publication Date
TW201204704A TW201204704A (en) 2012-02-01
TWI428325B true TWI428325B (zh) 2014-03-01

Family

ID=44072655

Family Applications (1)

Application Number Title Priority Date Filing Date
TW100113507A TWI428325B (zh) 2010-04-20 2011-04-19 製備吡唑羧醯胺之方法

Country Status (13)

Country Link
US (1) US8519152B2 (https=)
EP (1) EP2560959B1 (https=)
JP (1) JP5684896B2 (https=)
CN (1) CN102906072B (https=)
AR (1) AR080922A1 (https=)
BR (1) BR112012026631B1 (https=)
ES (1) ES2513540T3 (https=)
IL (1) IL222398A (https=)
MX (1) MX2012012005A (https=)
PY (1) PY1115670A (https=)
TW (1) TWI428325B (https=)
UY (1) UY33340A (https=)
WO (1) WO2011131545A1 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI480041B (zh) * 2010-04-20 2015-04-11 先正達合夥公司 用於製備吡唑羧醯胺之方法

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI534126B (zh) * 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法
GB201403438D0 (en) * 2014-02-27 2014-04-16 Syngenta Participations Ag Polymorphs
KR20250036910A (ko) 2022-07-22 2025-03-14 신젠타 크롭 프로텍션 아게 이종환식 아미드 유도체의 고체 형태
CN116143635B (zh) * 2022-12-01 2025-02-25 江苏七洲绿色科技研究院有限公司 一种9-二氯亚甲基-5-氨基-苯并降冰片烯的制备方法
PY2503719A (es) 2024-01-26 2025-08-05 Syngenta Crop Protection Ag Proceso químico

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH075487B2 (ja) 1985-11-14 1995-01-25 住友化学工業株式会社 1―ブロモ―2―クロロ―4―フルオロベンゼンの製造法
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
US7223879B2 (en) 1998-07-10 2007-05-29 Massachusetts Institute Of Technology Ligands for metals and improved metal-catalyzed processes based thereon
US7732469B2 (en) 2005-10-25 2010-06-08 Syngenta Crop Protection, Inc. Heterocyclic amide derivatives useful as microbiocides
WO2007124907A2 (en) 2006-04-27 2007-11-08 Syngenta Participations Ag Heterocyclyl-carboxylic acid (benzonorbornene-5-yl)amide derivatives as fungicides for agrochemical use
CN101528034B (zh) 2006-10-25 2011-11-09 辛根塔有限公司 生产经取代的溴苯的方法
BRPI0923527A2 (pt) * 2008-12-24 2016-08-09 Syngenta Ltd métodos de preparo de fungicidas

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI480041B (zh) * 2010-04-20 2015-04-11 先正達合夥公司 用於製備吡唑羧醯胺之方法

Also Published As

Publication number Publication date
AR080922A1 (es) 2012-05-16
US8519152B2 (en) 2013-08-27
CN102906072A (zh) 2013-01-30
IL222398A (en) 2017-01-31
BR112012026631A2 (pt) 2015-09-15
US20130035496A1 (en) 2013-02-07
TW201204704A (en) 2012-02-01
JP2013525317A (ja) 2013-06-20
JP5684896B2 (ja) 2015-03-18
WO2011131545A1 (en) 2011-10-27
CN102906072B (zh) 2014-07-02
BR112012026631B1 (pt) 2017-07-25
EP2560959A1 (en) 2013-02-27
EP2560959B1 (en) 2014-08-20
PY1115670A (es) 2014-09-01
MX2012012005A (es) 2012-12-17
UY33340A (es) 2011-12-01
ES2513540T3 (es) 2014-10-27

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