TWI394570B - 作為凝血因子ＩＸａ的抑制劑之異絲胺酸衍生物 - Google Patents

作為凝血因子ＩＸａ的抑制劑之異絲胺酸衍生物 Download PDF

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TWI394570B
TWI394570B TW096133788A TW96133788A TWI394570B TW I394570 B TWI394570 B TW I394570B TW 096133788 A TW096133788 A TW 096133788A TW 96133788 A TW96133788 A TW 96133788A TW I394570 B TWI394570 B TW I394570B
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hydroxy
amino
phenylethyl
benzimidazol
het
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TW096133788A
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Chinese (zh)
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TW200829245A (en
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Henning Steinhagen
Markus Follmann
Jochen Goerlitzer
Herman Schreuder
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Sanofi Aventis
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  • Organic Chemistry (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Diabetes (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
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TW096133788A 2006-09-13 2007-09-11 作為凝血因子ＩＸａ的抑制劑之異絲胺酸衍生物 TWI394570B (zh)

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CA2477604A1 (en) 2002-03-13 2003-09-25 Signum Biosciences, Inc. Modulation of protein methylation and phosphoprotein phosphate
US7923041B2 (en) 2005-02-03 2011-04-12 Signum Biosciences, Inc. Compositions and methods for enhancing cognitive function
EP1843734A4 (en) 2005-02-03 2008-09-10 Signum Biosciences Inc COMPOSITIONS AND METHOD FOR INTENSIFYING COGNITIVE FUNCTIONS
CA2662626C (en) * 2006-09-07 2016-07-26 Industrial Research Limited Acyclic amine inhibitors of 5'-methylthioadenosine phosphorylase and nucleosidase
CN102014897B (zh) 2008-04-21 2015-08-05 西格纳姆生物科学公司 化合物、组合物和其制备方法
TW201033184A (en) 2008-12-05 2010-09-16 Mochida Pharm Co Ltd Morpholinone compounds as factor IXa inhibitors
EP2473491B1 (en) * 2009-08-31 2013-07-17 Mochida Pharmaceutical Co., Ltd. Morpholinone compounds as factor ixa inhibitors
EP3131897B8 (en) 2014-04-16 2022-08-03 Merck Sharp & Dohme LLC Factor ixa inhibitors
CN109627218B (zh) * 2018-11-27 2022-03-29 深圳市龙华区中心医院 一种抗凝小分子化合物及其应用和包含其的药物

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US20050137168A1 (en) * 2003-12-19 2005-06-23 Gobbi Luca C. Heterocyclyl substituted 1-alkoxy acetic acid amides

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AR063708A1 (es) 2009-02-11
US8097758B2 (en) 2012-01-17
WO2008031509A1 (de) 2008-03-20
CL2007002652A1 (es) 2008-02-08
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CA2663544A1 (en) 2008-03-20
MX2009002047A (es) 2009-03-06
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MA30707B1 (fr) 2009-09-01
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AU2007297013A1 (en) 2008-03-20
CN101516834B (zh) 2013-04-03
TW200829245A (en) 2008-07-16
RU2009113602A (ru) 2010-10-20
IL197504A (en) 2013-06-27
RU2446157C2 (ru) 2012-03-27
EP2069289B1 (de) 2013-10-02
JP2010503625A (ja) 2010-02-04
AU2007297013B2 (en) 2012-05-31
EP2069289A1 (de) 2009-06-17
US20090233949A1 (en) 2009-09-17
SG174080A1 (en) 2011-09-29
IL197504A0 (en) 2009-12-24
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