TW429254B - Novel pyrimidin-4-one and pyrimidin-4-thione as fungicide - Google Patents

Novel pyrimidin-4-one and pyrimidin-4-thione as fungicide

Info

Publication number
TW429254B
TW429254B TW087114037A TW87114037A TW429254B TW 429254 B TW429254 B TW 429254B TW 087114037 A TW087114037 A TW 087114037A TW 87114037 A TW87114037 A TW 87114037A TW 429254 B TW429254 B TW 429254B
Authority
TW
Taiwan
Prior art keywords
halogen
c6alkyl
mono
pyrimidin
c6alkoxy
Prior art date
Application number
TW087114037A
Other languages
English (en)
Chinese (zh)
Inventor
Harald Walter
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of TW429254B publication Critical patent/TW429254B/zh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/90Oxygen atoms with acyclic radicals attached in position 2 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/91Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/92Oxygen atoms with hetero atoms directly attached to nitrogen atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/28Halogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/36Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Health & Medical Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
TW087114037A 1997-09-12 1998-08-25 Novel pyrimidin-4-one and pyrimidin-4-thione as fungicide TW429254B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9719411.2A GB9719411D0 (en) 1997-09-12 1997-09-12 New Pesticides

Publications (1)

Publication Number Publication Date
TW429254B true TW429254B (en) 2001-04-11

Family

ID=10818960

Family Applications (1)

Application Number Title Priority Date Filing Date
TW087114037A TW429254B (en) 1997-09-12 1998-08-25 Novel pyrimidin-4-one and pyrimidin-4-thione as fungicide

Country Status (26)

Country Link
US (1) US6277858B1 (https=)
EP (1) EP1015434B1 (https=)
JP (1) JP2001516749A (https=)
KR (1) KR100585571B1 (https=)
CN (1) CN1270593A (https=)
AR (1) AR015439A1 (https=)
AT (1) ATE216370T1 (https=)
AU (1) AU743717B2 (https=)
BR (1) BR9812439A (https=)
CA (1) CA2301694A1 (https=)
DE (1) DE69804981T2 (https=)
DK (1) DK1015434T3 (https=)
EG (1) EG22051A (https=)
ES (1) ES2175804T3 (https=)
GB (1) GB9719411D0 (https=)
GT (1) GT199800142A (https=)
HN (1) HN1998000139A (https=)
HU (1) HUP0002423A3 (https=)
IL (1) IL134779A0 (https=)
NZ (1) NZ503261A (https=)
PL (1) PL339053A1 (https=)
PT (1) PT1015434E (https=)
TR (1) TR200000713T2 (https=)
TW (1) TW429254B (https=)
WO (1) WO1999014202A2 (https=)
ZA (1) ZA988336B (https=)

Families Citing this family (45)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR9809598A (pt) * 1997-05-08 2000-07-04 Agrevo Uk Ltd Uso de compostos, e, composto.
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
GB9824331D0 (en) * 1998-11-06 1998-12-30 Novartis Ag Organic compounds
GB0021786D0 (en) * 2000-09-05 2000-10-18 Zeneca Ltd Fungicidal formulations
AU2002227243A1 (en) * 2000-12-11 2002-06-24 E.I. Du Pont De Nemours And Company Quinazolinones and pyridinopyrimidinones for controlling invertebrate pests
TW200306155A (en) 2002-03-19 2003-11-16 Du Pont Benzamides and advantageous compositions thereof for use as fungicides
KR100967280B1 (ko) * 2002-06-11 2010-07-01 이 아이 듀폰 디 네모아 앤드 캄파니 흰가루병을 방제하는데 유용한 융합된 피리미디논과디니트로페놀 화합물의 혼합물
PT1511380E (pt) * 2002-06-11 2006-12-29 Du Pont Mistura de pirimidinonas fundidas e compostos dinitrofenólicos úteis para controlar oídios
DE10347090A1 (de) 2003-10-10 2005-05-04 Bayer Cropscience Ag Synergistische fungizide Wirkstoffkombinationen
DE10349501A1 (de) 2003-10-23 2005-05-25 Bayer Cropscience Ag Synergistische fungizide Wirkstoffkombinationen
CN1898254A (zh) * 2003-10-30 2007-01-17 马萨诸塞州立大学 肽合成的新偶联剂
WO2005061518A1 (en) * 2003-12-19 2005-07-07 Merck & Co., Inc. Mitotic kinesin inhibitors
JP2007517066A (ja) * 2003-12-31 2007-06-28 サイオス・インコーポレーテツド ピリドピリミドンの製造方法
DE102004049761A1 (de) 2004-10-12 2006-04-13 Bayer Cropscience Ag Fungizide Wirkstoffkombinationen
DE102005015677A1 (de) 2005-04-06 2006-10-12 Bayer Cropscience Ag Synergistische fungizide Wirkstoffkombinationen
DE102005026482A1 (de) 2005-06-09 2006-12-14 Bayer Cropscience Ag Wirkstoffkombinationen
CN104170838B (zh) 2005-06-09 2016-03-30 拜尔农作物科学股份公司 活性物质结合物
CN100335481C (zh) * 2005-10-11 2007-09-05 华中师范大学 一类具有杀菌除草活性的多取代吡啶并[4,3-d]嘧啶及制备
DE102006023263A1 (de) * 2006-05-18 2007-11-22 Bayer Cropscience Ag Synergistische Wirkstoffkombinationen
WO2008013622A2 (en) 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
CL2007003256A1 (es) 2006-11-15 2008-07-25 Du Pont Mezcla fungicida que comprende al menos tres compuestos diferentes; composicion fungicida que comprende dicha mezcla; y metodo para controlar una enfermedad en plantas causada por el patogeno fungico vegetal que comprende aplicar una cantidad de la m
JP5337711B2 (ja) 2007-01-25 2013-11-06 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 殺菌性アミド
DE102007045920B4 (de) 2007-09-26 2018-07-05 Bayer Intellectual Property Gmbh Synergistische Wirkstoffkombinationen
US8349870B2 (en) 2008-01-25 2013-01-08 E I Du Pont De Nemours And Company Fungicidal hetercyclic compounds
CN101531638B (zh) * 2008-03-13 2011-12-28 中国科学院广州生物医药与健康研究院 用作雌激素相关受体调节剂的化合物及其应用
CN101628913B (zh) * 2008-07-18 2013-01-23 中国科学院广州生物医药与健康研究院 用作雌激素相关受体调节剂的化合物及其应用
AU2009322486A1 (en) 2008-12-02 2010-06-10 E. I. Du Pont De Nemours And Company Fungicidal heterocyclic compounds
AR075713A1 (es) 2009-03-03 2011-04-20 Du Pont Pirazoles fungicidas
WO2010108507A2 (de) 2009-03-25 2010-09-30 Bayer Cropscience Ag Synergistische wirkstoffkombinationen
CN102510721B (zh) 2009-07-16 2014-11-19 拜尔农作物科学股份公司 含苯基三唑的协同活性物质结合物
EP2462120A1 (en) 2009-08-07 2012-06-13 E. I. du Pont de Nemours and Company Fungicidal diphenyl-substituted pyridazines
TW201116212A (en) 2009-10-29 2011-05-16 Du Pont Heterobicycle-substituted azolyl benzene fungicides
WO2011051958A1 (en) 2009-10-30 2011-05-05 E.I. Du Pont De Nemours And Company Fungicidal pyrazolones
BR112012016733A2 (pt) 2010-01-07 2015-09-01 Du Pont "composto, composição fungicida e método"
CN102285971B (zh) * 2010-06-21 2013-12-18 中国中化股份有限公司 吡唑基喹唑啉酮类化合物及其应用
WO2012023143A1 (en) 2010-08-19 2012-02-23 E. I. Du Pont De Nemours And Company Fungicidal pyrazoles
CN103130730B (zh) * 2011-11-24 2015-04-08 南开大学 喹唑啉类衍生物及其制备方法、抗hiv活性和抗tmv活性
CN104151255B (zh) * 2014-07-22 2016-07-13 清华大学 一种多取代喹唑啉亚胺衍生物及其制备方法
EP2910126A1 (en) 2015-05-05 2015-08-26 Bayer CropScience AG Active compound combinations having insecticidal properties
JP7114076B2 (ja) 2015-12-22 2022-08-08 シャイ・セラピューティクス・エルエルシー がん及び炎症性疾患の処置のための化合物
WO2017207395A1 (en) 2016-06-02 2017-12-07 Bayer Cropscience Aktiengesellschaft Isothiazolopyridones, processes for their preparation and their use as fungicides
EP3464296B1 (en) 2016-06-02 2020-10-14 Bayer CropScience Aktiengesellschaft Isothiazolopyridones, processes for their preparation and their use as herbicides and/or plant growth regulators
PL3529246T3 (pl) 2016-10-24 2024-03-25 Fmc Corporation Oksadiazole o działaniu grzybobójczym
JP7514005B2 (ja) 2017-06-21 2024-07-10 シャイ・セラピューティクス・エルエルシー がん、炎症性疾患、ラソパシー、及び線維性疾患の治療のためのrasスーパーファミリーと相互作用する化合物
JP7407461B2 (ja) 2018-12-19 2024-01-04 シャイ・セラピューティクス・エルエルシー がん、炎症性疾患、ras病、及び線維性疾患の処置のためのrasスーパーファミリーと相互作用する化合物

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3714354A (en) * 1971-07-06 1973-01-30 Pfizer Bronchodilator activity of substituted quinazolinecarboxylic acid esters
BE793594A (fr) * 1972-01-03 1973-07-02 Pfizer Nouvelles 6,7-dimethoxyquinazolines utiles comme analgesiques et tranquillisants
GB8820129D0 (en) * 1988-08-24 1988-09-28 Schering Agrochemicals Ltd Fungicides
SK140295A3 (en) * 1993-05-12 1996-09-04 Du Pont Condensed bicyclic pyrimidinones, fungicidal agents on their base and inhibition method of plant deseases by using them
US5610301A (en) * 1993-07-01 1997-03-11 American Cyanamid Company Process for the regioselective n-alkylation of quinazolinones
BR9609613A (pt) * 1995-07-05 1999-05-25 Du Pont Composto composição fungicida e método de controle de doenças de plantas
BR9809598A (pt) * 1997-05-08 2000-07-04 Agrevo Uk Ltd Uso de compostos, e, composto.

Also Published As

Publication number Publication date
EP1015434A2 (en) 2000-07-05
ES2175804T3 (es) 2002-11-16
KR100585571B1 (ko) 2006-06-02
NZ503261A (en) 2002-03-28
KR20010023894A (ko) 2001-03-26
HUP0002423A3 (en) 2001-02-28
DE69804981T2 (de) 2002-11-28
CA2301694A1 (en) 1999-03-25
EG22051A (en) 2002-06-30
DK1015434T3 (da) 2002-08-05
CN1270593A (zh) 2000-10-18
HUP0002423A2 (hu) 2000-11-28
WO1999014202A2 (en) 1999-03-25
PL339053A1 (en) 2000-12-04
PT1015434E (pt) 2002-08-30
ZA988336B (en) 1999-02-12
BR9812439A (pt) 2000-09-26
AU9742998A (en) 1999-04-05
ATE216370T1 (de) 2002-05-15
HN1998000139A (es) 1999-06-02
US6277858B1 (en) 2001-08-21
WO1999014202B1 (en) 1999-06-17
AU743717B2 (en) 2002-01-31
WO1999014202A3 (en) 1999-05-14
AR015439A1 (es) 2001-05-02
GT199800142A (es) 2000-03-02
GB9719411D0 (en) 1997-11-12
IL134779A0 (en) 2001-04-30
DE69804981D1 (de) 2002-05-23
JP2001516749A (ja) 2001-10-02
EP1015434B1 (en) 2002-04-17
TR200000713T2 (tr) 2000-08-21

Similar Documents

Publication Publication Date Title
TW429254B (en) Novel pyrimidin-4-one and pyrimidin-4-thione as fungicide
MY102741A (en) Imidazole compounds and biocidal composition comprising the same for controlling harmful organisms
ATE239727T1 (de) Fungizide trifluoromethylalkylamino- triazolopyrimidine-derivate
EP1134214A4 (en) PICOLINAMIDE DERIVATIVES AND PESTICIDES CONTAINING THESE DERIVATIVES AS ACTIVE INGREDIENT
WO1998005652A3 (en) Arthropodicidal and fungicidal cyclic amides
PL373026A1 (en) 5-substituted-alkylaminopyrazole derivatives as pesticides
WO2005046672A3 (fr) Utilisation d’inhibiteurs de glucosidase pour une therapie de la mucoviscidose
HUT54867A (en) Fungicidal compositions comprising imidazole derivatives
IL64314A (en) 2-oxoazetidine derivatives,their production and antimicrobial and beta-lactamase inhibitory compositions containing them
EP0757987A4 (en) PYRAZOLECARBOXYLIC ACID DERIVATIVE AND PLANT DISEASE CONTROL AGENT
GB9819317D0 (en) Organic compounds
ES2078651T3 (es) Compuesto de piridinsulfonamida sustituida o una sal del mismo, procedimiento para su preparacion y herbicida que lo contiene.
WO1991019703A3 (en) Fungicidal iminooxazolidinones
NO20061355L (no) Fungicide blandinger for kontroll av rispatogener
WO1998017631A3 (en) Substituted oxime-ethers and their use as pesticides
AU2003235359A1 (en) Biguanide derivative and therapeutic agent for diabetes containing the same
WO2004060856A3 (en) Organic activator
NZ221330A (en) Fungicidal compositions containing benzimidazole derivatives for use against benomyl-resistant fungi
SE8801738D0 (sv) Forfarande for bekempning av mergborrar
JPS5732207A (en) Herbicidal composition
AU1287892A (en) Method of inhibiting the progressive development of diabetes mellitus
PT816355E (pt) Derivados espiro-heterociclicos
JPS56147703A (en) Fungicidal composition for agricultural and horticultural use
MD424G2 (ro) Derivaţi ai amidei
WO2003005823A3 (de) Bromnitrothienyldioxane

Legal Events

Date Code Title Description
GD4A Issue of patent certificate for granted invention patent
MM4A Annulment or lapse of patent due to non-payment of fees