TW227000B - - Google Patents

Info

Publication number
TW227000B
TW227000B TW081100891A TW81100891A TW227000B TW 227000 B TW227000 B TW 227000B TW 081100891 A TW081100891 A TW 081100891A TW 81100891 A TW81100891 A TW 81100891A TW 227000 B TW227000 B TW 227000B
Authority
TW
Taiwan
Prior art keywords
pct
sec
date
ring
fused
Prior art date
Application number
TW081100891A
Other languages
English (en)
Chinese (zh)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of TW227000B publication Critical patent/TW227000B/zh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Prostheses (AREA)
  • Steroid Compounds (AREA)
  • Cosmetics (AREA)
TW081100891A 1991-02-13 1992-02-10 TW227000B (OSRAM)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB919102997A GB9102997D0 (en) 1991-02-13 1991-02-13 Therapeutic agents

Publications (1)

Publication Number Publication Date
TW227000B true TW227000B (OSRAM) 1994-07-21

Family

ID=10689943

Family Applications (1)

Application Number Title Priority Date Filing Date
TW081100891A TW227000B (OSRAM) 1991-02-13 1992-02-10

Country Status (29)

Country Link
US (1) US5358953A (OSRAM)
EP (1) EP0572425B1 (OSRAM)
JP (1) JP2506541B2 (OSRAM)
KR (1) KR970005302B1 (OSRAM)
CN (1) CN1040326C (OSRAM)
AT (1) ATE109482T1 (OSRAM)
AU (1) AU650322B2 (OSRAM)
BR (1) BR9205615A (OSRAM)
CA (1) CA2099381C (OSRAM)
CZ (1) CZ280504B6 (OSRAM)
DE (1) DE69200304T2 (OSRAM)
DK (1) DK0572425T3 (OSRAM)
EG (1) EG20085A (OSRAM)
ES (1) ES2059212T3 (OSRAM)
FI (1) FI933531A7 (OSRAM)
GB (1) GB9102997D0 (OSRAM)
HU (2) HUT65947A (OSRAM)
IE (1) IE65125B1 (OSRAM)
IL (1) IL100887A (OSRAM)
MX (1) MX9200589A (OSRAM)
MY (1) MY108437A (OSRAM)
NO (1) NO300592B1 (OSRAM)
NZ (1) NZ241597A (OSRAM)
PL (1) PL169304B1 (OSRAM)
RU (1) RU2114845C1 (OSRAM)
TW (1) TW227000B (OSRAM)
WO (1) WO1992014734A1 (OSRAM)
YU (1) YU48238B (OSRAM)
ZA (1) ZA921005B (OSRAM)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2042421B1 (es) * 1992-05-22 1994-08-01 Uriach & Cia Sa J Procedimiento para la obtencion de la 8-cloro-11-*1-*(5-metil-3-piridil)metil*-4-piperidiliden*-6,11-dihidro-5h-benzo*5,6*ciclohepta*1,2-b*piridina.
US5753671A (en) * 1994-08-10 1998-05-19 British Biotech Pharmaceuticals Limited Imidazopyridine derivatives as dual histamine (H1) and platelet activating factor (PAF) antagonists
ES2087038B1 (es) * 1994-11-07 1997-03-16 Uriach & Cia Sa J Nuevas piperidinas con actividad antagonista del paf.
US5567711A (en) * 1995-04-19 1996-10-22 Abbott Laboratories Indole-3-carbonyl and indole-3-sulfonyl derivatives as platelet activating factor antagonists
GB9508748D0 (en) * 1995-04-28 1995-06-14 British Biotech Pharm Benzimidazole derivatives
MX9707187A (es) * 1995-08-05 1997-11-29 British Biotech Pharm Derivados de imidazopiridina.
SE9801526D0 (sv) * 1998-04-29 1998-04-29 Astra Ab New compounds
AU2001279313B2 (en) 2000-08-04 2007-03-01 Ampio Pharmaceuticals, Inc. Method of using diketopiperazines and composition containing them
ES2572454T3 (es) 2003-05-15 2016-05-31 Ampio Pharmaceuticals Inc Tratamiento de enfermedades mediadas por los linfocitos T
US7687515B2 (en) * 2006-01-17 2010-03-30 N.V. Organon 6-phenyl-1H-imidazo[4,5-c]pyridine-4-carbonitrile derivatives
CA2713293A1 (en) 2008-01-30 2009-08-06 Nippon Zoki Pharmaceutical Co., Ltd. Piperidine derivative
EP2300011A4 (en) 2008-05-27 2012-06-20 Dmi Life Sciences Inc THERAPEUTIC PROCESSES AND COMPOUNDS
CN103619839B (zh) * 2011-06-28 2016-06-01 福建省闽东力捷迅药业有限公司 抗-变态反应的苯并环庚并噻吩衍生物
EA028343B1 (ru) 2011-10-10 2017-11-30 Ампио Фармасьютикалз, Инк. Лечение дегенеративного заболевания сустава
AU2012323320B2 (en) 2011-10-10 2017-05-11 Ampio Pharmaceuticals, Inc. Implantable medical devices with increased immune tolerance, and methods for making and implanting
EP2771007B1 (en) * 2011-10-28 2018-04-04 Ampio Pharmaceuticals, Inc. Treatment of rhinitis
MX2015010937A (es) 2013-03-15 2015-10-29 Ampio Pharmaceuticals Inc Composiciones para la movilizacion, autodireccion, expansion y diferenciacion de celulas madre y metodos para usar las mismas.
WO2016028790A1 (en) 2014-08-18 2016-02-25 Ampio Pharmaceuticals, Inc. Treatment of joint conditions
US11389512B2 (en) 2015-06-22 2022-07-19 Ampio Pharmaceuticals, Inc. Use of low molecular weight fractions of human serum albumin in treating diseases
CN113880801A (zh) * 2020-07-03 2022-01-04 合肥医工医药股份有限公司 一类三环化合物、其制备方法及其医药用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL132137C (OSRAM) * 1963-04-24
EP0404797B1 (en) * 1988-03-15 1995-02-01 G.D. Searle & Co. 1H/3H-[4-(N,N-CYCLOALKYL AND/OR BRANCHED-ALKYLCARBOXAMIDO) -BENZYL]IMIDAZO[4,5-c]PYRIDINES AS PAF ANTAGONISTS
CA1341370C (en) * 1988-04-28 2002-06-18 John J. Powinski Fused polycyclic compounds, methods of manufacture, and their use as paf antagonists, antihistamines and/or antiinflammatory agents
US5250681A (en) * 1988-06-02 1993-10-05 Ajinomoto Co., Inc. Piperidine derivatives and hypotensives containing the same
US5114919A (en) * 1990-02-26 1992-05-19 Merck & Co., Inc. Adjuncts in cancer chemotherapy
ATE112567T1 (de) * 1990-05-09 1994-10-15 Pfizer Imidazo(4,5-c>pyridine als paf antagonisten.

Also Published As

Publication number Publication date
PL169304B1 (pl) 1996-06-28
ATE109482T1 (de) 1994-08-15
JPH06504992A (ja) 1994-06-09
EG20085A (en) 1997-05-31
FI933531A0 (fi) 1993-08-10
MY108437A (en) 1996-09-30
GB9102997D0 (en) 1991-03-27
DE69200304D1 (de) 1994-09-08
AU650322B2 (en) 1994-06-16
IL100887A (en) 1996-01-19
KR970005302B1 (ko) 1997-04-15
YU48238B (sh) 1997-08-22
NO300592B1 (no) 1997-06-23
AU1168392A (en) 1992-09-15
WO1992014734A1 (en) 1992-09-03
NO932889D0 (no) 1993-08-13
FI933531L (fi) 1993-08-10
DE69200304T2 (de) 1994-12-08
IE920449A1 (en) 1992-08-12
NZ241597A (en) 1993-04-28
MX9200589A (es) 1992-10-01
HU9302327D0 (en) 1993-10-28
EP0572425B1 (en) 1994-08-03
US5358953A (en) 1994-10-25
HU211202A9 (en) 1995-11-28
FI933531A7 (fi) 1993-08-10
HUT65947A (en) 1994-08-29
YU14392A (sh) 1994-11-15
CN1040326C (zh) 1998-10-21
IL100887A0 (en) 1992-11-15
RU2114845C1 (ru) 1998-07-10
BR9205615A (pt) 1994-05-17
JP2506541B2 (ja) 1996-06-12
CA2099381A1 (en) 1992-08-14
CZ280504B6 (cs) 1996-02-14
EP0572425A1 (en) 1993-12-08
NO932889L (no) 1993-08-13
DK0572425T3 (da) 1994-09-12
CA2099381C (en) 1996-07-09
ZA921005B (en) 1993-08-12
CN1064275A (zh) 1992-09-09
CS42592A3 (en) 1992-09-16
IE65125B1 (en) 1995-10-04
ES2059212T3 (es) 1994-11-01

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