TW203049B - - Google Patents

Download PDF

Info

Publication number
TW203049B
TW203049B TW080102725A TW80102725A TW203049B TW 203049 B TW203049 B TW 203049B TW 080102725 A TW080102725 A TW 080102725A TW 80102725 A TW80102725 A TW 80102725A TW 203049 B TW203049 B TW 203049B
Authority
TW
Taiwan
Prior art keywords
group
compound
same
page
alkyl
Prior art date
Application number
TW080102725A
Other languages
English (en)
Chinese (zh)
Original Assignee
Yamanouchi Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd
Application granted granted Critical
Publication of TW203049B publication Critical patent/TW203049B/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
TW080102725A 1990-04-13 1991-04-10 TW203049B (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP9845590 1990-04-13
JP28549390 1990-10-23

Publications (1)

Publication Number Publication Date
TW203049B true TW203049B (nl) 1993-04-01

Family

ID=26439622

Family Applications (1)

Application Number Title Priority Date Filing Date
TW080102725A TW203049B (nl) 1990-04-13 1991-04-10

Country Status (10)

Country Link
US (1) US5162318A (nl)
EP (1) EP0454330A1 (nl)
KR (1) KR910018360A (nl)
CN (1) CN1060837A (nl)
AU (1) AU7500891A (nl)
CA (1) CA2040235A1 (nl)
FI (1) FI911776A (nl)
HU (1) HUT57735A (nl)
IE (1) IE911251A1 (nl)
TW (1) TW203049B (nl)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9418326D0 (en) * 1994-09-12 1994-11-02 Lilly Industries Ltd Pharmaceutical compounds
GB2308362A (en) * 1995-12-19 1997-06-25 Lilly Industries Ltd Pharmaceutical indole derivatives
FR2767827A1 (fr) * 1997-09-03 1999-02-26 Adir Nouveaux derives de l'indole et de l'indazole, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US6498154B1 (en) 1999-05-04 2002-12-24 Wyeth Cyclic regimens using quinazolinone and benzoxazine derivatives
US6380235B1 (en) * 1999-05-04 2002-04-30 American Home Products Corporation Benzimidazolones and analogues
US6391907B1 (en) 1999-05-04 2002-05-21 American Home Products Corporation Indoline derivatives
US6358947B1 (en) 1999-05-04 2002-03-19 American Home Products Corporation Tetracyclic progesterone receptor modulator compounds and methods
US6355648B1 (en) 1999-05-04 2002-03-12 American Home Products Corporation Thio-oxindole derivatives
US6358948B1 (en) 1999-05-04 2002-03-19 American Home Products Corporation Quinazolinone and benzoxazine derivatives as progesterone receptor modulators
US6319912B1 (en) 1999-05-04 2001-11-20 American Home Products Corporation Cyclic regimens using 2,1-benzisothiazoline 2,2-dioxides
US6380178B1 (en) 1999-05-04 2002-04-30 American Home Products Corporation Cyclic regimens using cyclocarbamate and cyclic amide derivatives
US6462032B1 (en) 1999-05-04 2002-10-08 Wyeth Cyclic regimens utilizing indoline derivatives
US6444668B1 (en) 1999-05-04 2002-09-03 Wyeth Combination regimens using progesterone receptor modulators
US6399593B1 (en) 1999-05-04 2002-06-04 Wyeth Cyclic regimens using cyclic urea and cyclic amide derivatives
US6369056B1 (en) 1999-05-04 2002-04-09 American Home Products Corporation Cyclic urea and cyclic amide derivatives
US6423699B1 (en) 1999-05-04 2002-07-23 American Home Products Corporation Combination therapies using benzimidazolones
US6509334B1 (en) 1999-05-04 2003-01-21 American Home Products Corporation Cyclocarbamate derivatives as progesterone receptor modulators
US6306851B1 (en) 1999-05-04 2001-10-23 American Home Products Corporation Cyclocarbamate and cyclic amide derivatives
US6407101B1 (en) 1999-05-04 2002-06-18 American Home Products Corporation Cyanopyrroles
US6417214B1 (en) 1999-05-04 2002-07-09 Wyeth 3,3-substituted indoline derivatives
US6329416B1 (en) 1999-05-04 2001-12-11 American Home Products Corporation Combination regimens using 3,3-substituted indoline derivatives
US6339098B1 (en) 1999-05-04 2002-01-15 American Home Products Corporation 2,1-benzisothiazoline 2,2-dioxides
UA73119C2 (en) 2000-04-19 2005-06-15 American Home Products Corpoir Derivatives of cyclic thiocarbamates, pharmaceutical composition including noted derivatives of cyclic thiocarbamates and active ingredients of medicines as modulators of progesterone receptors
ES2367539T3 (es) 2001-12-21 2011-11-04 X-Ceptor Therapeutics, Inc. Moduladores heterocíclicos de receptores nucleares.
US7115644B2 (en) * 2002-09-13 2006-10-03 Boehringer Ingelheim Pharmaceuticals Inc. Heterocyclic compounds
EP1904483A1 (en) 2005-07-13 2008-04-02 F. Hoffmann-Roche AG Benzimidazole derivatives as 5-ht6,5-ht24
AU2021268614A1 (en) * 2020-05-06 2022-12-08 Merck Sharp & Dohme Llc IL4I1 inhibitors and methods of use

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2609645A1 (de) * 1976-03-09 1977-09-15 Boehringer Sohn Ingelheim Aminoalkylheterocyclen
DE2644833A1 (de) * 1976-10-05 1978-04-20 Boehringer Sohn Ingelheim Neue 1-aryloxy-2-hydroxy-3-alkylenaminopropane und verfahren zu ihrer herstellung
US4200641A (en) * 1976-12-21 1980-04-29 Janssen Pharmaceutica, N.V. 1-[(Heterocyclyl)-alkyl]-4-diarylmethoxy piperidine derivatives
US4359468A (en) * 1981-02-25 1982-11-16 Boehringer Ingelheim Ltd. Antiallergic N-[4-(indolyl)-piperidino-alkyl]-benzimidazolones
US4492708A (en) * 1982-09-27 1985-01-08 Eli Lilly And Company Antiviral benzimidazoles
JPS62252721A (ja) * 1986-04-24 1987-11-04 Kissei Pharmaceut Co Ltd 消化性潰瘍治療剤
FR2643903A1 (fr) * 1989-03-03 1990-09-07 Union Pharma Scient Appl Nouveaux derives de benzimidazole, leurs procedes de preparation, intermediaires de synthese, compositions pharmaceutiques les contenant, utiles notamment pour le traitement des maladies cardiovasculaires, et des ulceres duodenaux

Also Published As

Publication number Publication date
HU911226D0 (en) 1991-10-28
CN1060837A (zh) 1992-05-06
EP0454330A1 (en) 1991-10-30
US5162318A (en) 1992-11-10
KR910018360A (ko) 1991-11-30
IE911251A1 (en) 1991-10-23
HUT57735A (en) 1991-12-30
FI911776A0 (fi) 1991-04-12
FI911776A (fi) 1991-10-14
AU7500891A (en) 1991-10-17
CA2040235A1 (en) 1991-10-14

Similar Documents

Publication Publication Date Title
TW203049B (nl)
ES2249913T3 (es) Derivados de imidazo-piridina que inhiben la secrecion de acido gastrico.
US4841047A (en) 4-benzyl-1-(2H)-phthalazinone-derivates
ES2694829T3 (es) Derivados de benzotriazol trisustituido como inhibidores de dihidroorotato oxigenasa
AU773504B2 (en) Derivatives of pyrimido(6,1-a)isoquinolin-4-one
BG62618B1 (bg) Асиметрично заместени ксантини с аденозинантагонистичнисвойства, метод за тяхното получаване и междинни съединения затази цел, приложение на тези съединения като фармакологичнисредства, фармацевтични смеси, които ги съдържат, и метод затяхното получаване
PT85692B (pt) Processo para a preparacao de derivados de benzimidazois (1h-imidazol-1-ilmetil)-substituidos e de composicoes farmaceuticas que os contem
PT1689751E (pt) Novas 5,7-diaminopirazolo[4,3-d]pirimidinas com actividade inibidora de pde-5
JPH05155858A (ja) トロンボキサン受容体アンタゴニストである新規ベンズイミダゾールおよびアザベンズイミダゾール誘導体、それらの製造方法、およびそれらを含む合成中間体および薬剤組成物
JPS6293274A (ja) 新規アミド誘導体及びその製法
JPS60501708A (ja) アロプリノ−ル　プロドラツグ類
JPH0655728B2 (ja) ヒスタミン誘導体及びその製造方法並びに該誘導体を含有する医薬
US4761411A (en) Dihydrobenzopyrrolobenzodiazepines useful for treating pyschoses
JPH06507620A (ja) イミダゾベンゾキノン類およびこれを有効成分とする高血圧・鬱血性心不全の予防・治療剤
HU177422B (en) Process for preparing new 6-phenyl-s-triazolo/4,3-a/pyrido/2,3-f/ /1,4/-diazepines
US4258059A (en) Amino-benzamides
CA3169832A1 (en) Use of jak inhibitors in preparation of drugs for treatment of jak kinase related diseases
JPH01501477A (ja) 抗葉酸剤
KR880001719B1 (ko) 1,4,9,10-테트라하이드로-피라졸로[4,3-e]-피리도[3,2-b][1,4]디아제핀-10-온의 제조 방법
PT93457A (pt) Processo para a preparacao de um derivado de triazina e de composicoes farmaceuticas que os contem
PT88244B (pt) Processo para a preparacao de derivados de tetrazole antagonistas de leucotrienos
TW206230B (nl)
CA1141765A (en) Benzimidazole derivatives
JPS60166651A (ja) 新規ジアミド化合物
ES2322463T3 (es) Preocedimiento para preparar derivados de imidazol sustituidos y productos intermedios utilizados en el procedimiento.