TW202208337A - Enpp1之亞胺基硫烷酮抑制劑 - Google Patents

Enpp1之亞胺基硫烷酮抑制劑 Download PDF

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TW202208337A
TW202208337A TW110115908A TW110115908A TW202208337A TW 202208337 A TW202208337 A TW 202208337A TW 110115908 A TW110115908 A TW 110115908A TW 110115908 A TW110115908 A TW 110115908A TW 202208337 A TW202208337 A TW 202208337A
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compound
pharmaceutically acceptable
acceptable salt
methyl
mmol
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TW110115908A
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Chinese (zh)
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德里克 A 柯根
莎拉 貝蒂戈爾
新森 蘇
皮奧特 尼采爾
伯科姆 里昂 范
羅格 福爾默
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美商佛拉斯托醫療公司
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Publication of TW202208337A publication Critical patent/TW202208337A/zh

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TW110115908A 2020-05-04 2021-05-03 Enpp1之亞胺基硫烷酮抑制劑 TW202208337A (zh)

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US202063019853P 2020-05-04 2020-05-04
US63/019,853 2020-05-04
US202063093709P 2020-10-19 2020-10-19
US63/093,709 2020-10-19

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EP (1) EP4146344A1 (https=)
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KR (1) KR20230019431A (https=)
CN (1) CN115996912A (https=)
AU (1) AU2021268606A1 (https=)
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BR112022023112A2 (pt) * 2020-05-14 2023-01-17 Vir Biotechnology Inc Moduladores de enpp1 e usos dos mesmos
US12091412B2 (en) 2020-06-16 2024-09-17 Volastra Therapeutics, Inc. Heterocyclic inhibitors of ENPP1
EP4236928A4 (en) 2020-10-30 2024-08-28 1Cbio, Inc. ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE 1 (ENPP1) INHIBITORS AND THEIR USES
WO2023086638A1 (en) * 2021-11-15 2023-05-19 Vir Biotechnology, Inc. Enpp1 modulators and uses thereof
JP2024545511A (ja) * 2021-12-09 2024-12-09 バラ セラピューティクス,インコーポレイテッド メニン-mll相互作用の阻害剤
EP4514331A1 (en) 2022-04-29 2025-03-05 Petragen, Inc. Inhibitors of enpp1 and modulation of bone growth
WO2023225001A1 (en) * 2022-05-16 2023-11-23 Vir Biotechnology, Inc. Naphthyridine based enpp1 modulators and uses thereof
CN119677742A (zh) * 2022-08-01 2025-03-21 斯拉瓦蒂人工智能科技私人有限公司 一种新型外核苷酸焦磷酸酶/磷酸二酯酶1(enpp1)抑制剂及其用途
WO2024127343A1 (en) * 2022-12-16 2024-06-20 Sravathi Ai Technology Private Limited Inhibitors of ectonucleotide pyrophosphatase / phosphodiesterase 1 (enpp-1)
WO2025207514A1 (en) * 2024-03-25 2025-10-02 Riboscience Llc Bicyclic heteroaryl sulfanediimine derivatives as ectonucleotide pyrophosphatase phosphodiesterase 1 inhibitors

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