TW201622721A - Ｓ１ｐ調節劑之立即釋放劑量療法 - Google Patents

Ｓ１ｐ調節劑之立即釋放劑量療法 Download PDF

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Publication number
TW201622721A
TW201622721A TW104111330A TW104111330A TW201622721A TW 201622721 A TW201622721 A TW 201622721A TW 104111330 A TW104111330 A TW 104111330A TW 104111330 A TW104111330 A TW 104111330A TW 201622721 A TW201622721 A TW 201622721A
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TW
Taiwan
Prior art keywords
day
dosage form
patient
treatment
immediate release
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TW104111330A
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English (en)
Chinese (zh)
Inventor
菲利普 米契爾 蕾恩 波洛特
法蘭克 道可
艾力克 勒崗紐斯
艾梅瑞克 瑞諾德
艾利克 沃史托
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諾華公司
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52988364&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TW201622721(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 諾華公司 filed Critical 諾華公司
Publication of TW201622721A publication Critical patent/TW201622721A/zh

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
TW104111330A 2014-04-10 2015-04-08 Ｓ１ｐ調節劑之立即釋放劑量療法 TW201622721A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201461977816P 2014-04-10 2014-04-10

Publications (1)

Publication Number Publication Date
TW201622721A true TW201622721A (zh) 2016-07-01

Family

ID=52988364

Family Applications (1)

Application Number Title Priority Date Filing Date
TW104111330A TW201622721A (zh) 2014-04-10 2015-04-08 Ｓ１ｐ調節劑之立即釋放劑量療法

Country Status (16)

Country Link
US (4) US20170027907A1 (OSRAM)
EP (3) EP4074312A1 (OSRAM)
JP (1) JP6674903B2 (OSRAM)
KR (2) KR20160141841A (OSRAM)
CN (2) CN106456552A (OSRAM)
AU (2) AU2015246036A1 (OSRAM)
CA (1) CA2943598C (OSRAM)
CL (1) CL2016002562A1 (OSRAM)
IL (2) IL305337A (OSRAM)
MX (1) MX2016013245A (OSRAM)
PH (1) PH12016501965A1 (OSRAM)
RU (2) RU2020107732A (OSRAM)
SG (1) SG11201607894RA (OSRAM)
TW (1) TW201622721A (OSRAM)
WO (1) WO2015155709A1 (OSRAM)
ZA (1) ZA201606519B (OSRAM)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO2699580T3 (OSRAM) 2014-01-24 2018-02-24
RU2020107732A (ru) * 2014-04-10 2020-03-30 Новартис Аг Схема дозирования модулятора s1p с немедленным высвобождением
US11434200B2 (en) 2017-03-09 2022-09-06 Novartis Ag Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof
US11629124B2 (en) 2017-03-09 2023-04-18 Novartis Ag Solid forms comprising an oxime ether compound, compositions and methods of use thereof
CA3074416A1 (en) * 2017-09-29 2019-04-04 Novartis Ag Dosing regimen of siponimod
CN111107845A (zh) * 2017-09-29 2020-05-05 诺华股份有限公司 西尼莫德的给药方案
SI3758708T1 (sl) 2018-03-01 2025-04-30 Astrazeneca Ab Farmacevtski sestavki, ki vsebujejo (2S)-{(1S)-1-ciano-2-[4-(3-metil-2-okso-2,3-dihidro-1,3-benzoksazol-5-il)fenil]etil}-1,4-oksazepan-2-karboksamid
AU2019306532A1 (en) 2018-07-17 2021-03-04 Insmed Incorporated Certain (2S)-N-[(1S)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating Lupus Nephritis
CN109908095A (zh) * 2019-04-08 2019-06-21 肇庆学院 一种西尼莫德片剂及制备方法
KR20220093330A (ko) 2019-10-31 2022-07-05 이도르시아 파마슈티컬스 리미티드 Cxcr7 안타고니스트와 s1p1 수용체 조절인자의 조합
US11135197B2 (en) 2020-02-07 2021-10-05 Argentum Pharmaceuticals Llc Dosage regimen of an S1P receptor modulator
CN120584108A (zh) 2023-01-06 2025-09-02 英斯梅德股份有限公司 新型可逆dpp1抑制剂及其用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104803902A (zh) * 2008-12-18 2015-07-29 诺华股份有限公司 1-(4-{1-[(e)-4-环己基-3-三氟甲基-苄氧基亚氨基]-乙基}-2-乙基-苄基)-氮杂环丁烷-3-甲酸的半富马酸盐
UY32352A (es) * 2008-12-22 2010-07-30 Novartis Ag Régimen de dosificación para un agonista de los receptores de s1p
CN105213372A (zh) * 2008-12-22 2016-01-06 诺华股份有限公司 S1p受体激动剂的给药方案
PH12012500520A1 (en) * 2009-09-29 2012-10-22 Novartis Ag Dosage regimen of an s1p receptor modulator
JO3619B1 (ar) * 2011-01-07 2020-08-27 Novartis Ag صياغات مثبطة للمناعة
WO2012095853A1 (en) * 2011-01-10 2012-07-19 Novartis Pharma Ag Modified release formulations comprising sip receptor modulators
SG10201602279PA (en) * 2011-10-21 2016-04-28 Novartis Ag Dosage regimen for an s1p receptor modulator or agonist
RU2020107732A (ru) * 2014-04-10 2020-03-30 Новартис Аг Схема дозирования модулятора s1p с немедленным высвобождением

Also Published As

Publication number Publication date
RU2016143979A3 (OSRAM) 2018-11-12
AU2020203107A1 (en) 2020-05-28
PH12016501965A1 (en) 2017-01-09
MX2016013245A (es) 2017-01-16
CA2943598A1 (en) 2015-10-15
EP4074312A1 (en) 2022-10-19
IL305337A (en) 2023-10-01
IL247986A0 (en) 2016-11-30
EP3129020A1 (en) 2017-02-15
CN116650467A (zh) 2023-08-29
KR20220156981A (ko) 2022-11-28
RU2020107732A (ru) 2020-03-30
US20170027907A1 (en) 2017-02-02
EP3831378A1 (en) 2021-06-09
CL2016002562A1 (es) 2017-07-28
US20190054065A1 (en) 2019-02-21
ZA201606519B (en) 2017-11-29
WO2015155709A1 (en) 2015-10-15
AU2020203107B2 (en) 2021-10-21
RU2016143979A (ru) 2018-05-14
JP2017510607A (ja) 2017-04-13
SG11201607894RA (en) 2016-10-28
CN106456552A (zh) 2017-02-22
CA2943598C (en) 2023-03-07
RU2715734C2 (ru) 2020-03-03
US20220016076A1 (en) 2022-01-20
US20250041266A1 (en) 2025-02-06
KR20160141841A (ko) 2016-12-09
JP6674903B2 (ja) 2020-04-01
AU2015246036A1 (en) 2016-10-13

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