TW201536284A - 使用黃嘌呤氧化酶抑制劑之治療方法與組成物 - Google Patents
使用黃嘌呤氧化酶抑制劑之治療方法與組成物 Download PDFInfo
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- TW201536284A TW201536284A TW103119057A TW103119057A TW201536284A TW 201536284 A TW201536284 A TW 201536284A TW 103119057 A TW103119057 A TW 103119057A TW 103119057 A TW103119057 A TW 103119057A TW 201536284 A TW201536284 A TW 201536284A
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
- A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Immunology (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
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|---|---|---|---|
| US201361829759P | 2013-05-31 | 2013-05-31 | |
| US201361839609P | 2013-06-26 | 2013-06-26 |
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| TW201536284A true TW201536284A (zh) | 2015-10-01 |
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| TW103119057A TW201536284A (zh) | 2013-05-31 | 2014-05-30 | 使用黃嘌呤氧化酶抑制劑之治療方法與組成物 |
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| Country | Link |
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| US (2) | US20140357683A1 (enExample) |
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| TW (1) | TW201536284A (enExample) |
| WO (1) | WO2014194226A2 (enExample) |
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| RU2018118603A (ru) * | 2015-10-28 | 2019-11-28 | Сан Фармасьютикал Индастриз Лимитед | Фармацевтические композиции диметилфумарата |
| CN105769766B (zh) * | 2016-03-24 | 2018-07-06 | 长沙佰顺生物科技有限公司 | 一种托匹司他纳米乳及其制备方法 |
| JP7108384B2 (ja) * | 2016-07-13 | 2022-07-28 | 日本ケミファ株式会社 | ２－［３－シアノ－４－（２－メチルプロポキシ）フェニル］－４－メチルチアゾール－５－カルボン酸の口腔内崩壊錠 |
| WO2018017368A1 (en) * | 2016-07-18 | 2018-01-25 | Arthrosi Therapeutics, Llc | Compounds, compositions and methods for treating or preventing a sympton associated with gout or hyperuricemia |
| IL283663B2 (en) | 2018-12-06 | 2025-12-01 | Arthrosi Therapeutics Inc | Crystalline forms of (3,5-dibromo-4-hydroxyphenyl)(2-(1-hydroxyethyl)benzofuran-3-yl-4,5,6,7-d4)methanone and pharmaceutical composition comprsing them |
| US12419854B2 (en) | 2018-12-06 | 2025-09-23 | Arthrosi Therapeutics, Inc. | Methods for treating or preventing gout or hyperuricemia |
| US20220323441A1 (en) * | 2019-06-04 | 2022-10-13 | Nippon Chemiphar Co., Ltd. | Therapeutic for gout or hyperuricemia |
| MX2023014357A (es) * | 2021-06-15 | 2023-12-15 | Lg Chemical Ltd | Una composicion farmaceutica que comprende acido 1-(3-ciano-1-isopropil-indol-5-il)pirazol-4-carboxilo. |
| CN115252567A (zh) * | 2022-07-08 | 2022-11-01 | 广西纯正堂制药有限公司 | 非布司他渗透泵缓释片及其制备方法 |
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| GB1478759A (en) | 1974-11-18 | 1977-07-06 | Alza Corp | Process for forming outlet passageways in pills using a laser |
| US4200098A (en) | 1978-10-23 | 1980-04-29 | Alza Corporation | Osmotic system with distribution zone for dispensing beneficial agent |
| US5286497A (en) | 1991-05-20 | 1994-02-15 | Carderm Capital L.P. | Diltiazem formulation |
| US5573776A (en) | 1992-12-02 | 1996-11-12 | Alza Corporation | Oral osmotic device with hydrogel driving member |
| US5544163A (en) | 1994-03-08 | 1996-08-06 | Excel, Inc. | Expandable telecommunications system |
| PT1488790E (pt) | 2002-03-28 | 2014-10-10 | Teijin Pharma Ltd | Preparação sólida contendo uma forma de cristal único a de um derivado de ácido tiazolcarboxílico |
| JP4914210B2 (ja) | 2004-06-14 | 2012-04-11 | 日本ケミファ株式会社 | 縮合ピリミジン誘導体、及びキサンチンオキシダーゼ阻害剤 |
| JP5040656B2 (ja) | 2005-10-07 | 2012-10-03 | アステラス製薬株式会社 | トリアリールカルボン酸誘導体 |
| CA2675443A1 (en) * | 2007-01-19 | 2008-07-24 | Takeda Pharmaceuticals North America, Inc. | Methods for preventing or reducing the number of gout flares using xanthine oxidoreductase inhibitors and anti-inflammatory agents |
| HRP20130846T1 (hr) | 2009-03-31 | 2013-11-22 | Kissei Pharmaceutical Co., Ltd. | Derivati indolizina i njihova uporaba u medicinske svrhe |
| CN101773498B (zh) * | 2009-12-30 | 2012-06-20 | 青岛黄海制药有限责任公司 | 一种含有非布司他的口服缓控释制剂的制备方法 |
| CA2802831C (en) | 2010-06-16 | 2018-11-20 | Teijin Pharma Limited | Controlled release coat-core tablet |
| TW201202249A (en) | 2010-06-16 | 2012-01-16 | Takeda Pharmaceuticals North America Inc | Novel modified release dosage forms of xanthine oxidoreductase inhibitor or xanthine oxidase inhibitors |
| CN102641255A (zh) * | 2012-05-08 | 2012-08-22 | 南方医科大学 | 一种治疗痛风的非布索坦渗透泵控释片及其制备方法 |
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2014
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- 2014-05-30 SG SG10201709955PA patent/SG10201709955PA/en unknown
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- 2014-05-30 SG SG11201509738RA patent/SG11201509738RA/en unknown
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- 2014-05-30 CA CA2913755A patent/CA2913755A1/en not_active Abandoned
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2015
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2017
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2019
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Also Published As
| Publication number | Publication date |
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| JP2019108356A (ja) | 2019-07-04 |
| PH12015502679A1 (en) | 2016-03-07 |
| CA2913755A1 (en) | 2014-12-04 |
| WO2014194226A2 (en) | 2014-12-04 |
| SG11201509738RA (en) | 2015-12-30 |
| JP2016520133A (ja) | 2016-07-11 |
| CN105579037A (zh) | 2016-05-11 |
| US20180311217A1 (en) | 2018-11-01 |
| SG10201709955PA (en) | 2018-01-30 |
| MX2015016494A (es) | 2016-11-18 |
| US20140357683A1 (en) | 2014-12-04 |
| WO2014194226A3 (en) | 2015-05-14 |
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