TW201325606A - 用氯化鈉穩定化之依那西普調配物 - Google Patents

用氯化鈉穩定化之依那西普調配物 Download PDF

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Publication number
TW201325606A
TW201325606A TW101138560A TW101138560A TW201325606A TW 201325606 A TW201325606 A TW 201325606A TW 101138560 A TW101138560 A TW 101138560A TW 101138560 A TW101138560 A TW 101138560A TW 201325606 A TW201325606 A TW 201325606A
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Taiwan
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weight
composition
peak
etanercept
hic
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TW101138560A
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English (en)
Chinese (zh)
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Mark Manning
Brian Murphy
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Coherus Biosciences Inc
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Publication of TW201325606A publication Critical patent/TW201325606A/zh

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/177—Receptors; Cell surface antigens; Cell surface determinants
    • A61K38/1793—Receptors; Cell surface antigens; Cell surface determinants for cytokines; for lymphokines; for interferons
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    • A61K38/19—Cytokines; Lymphokines; Interferons
    • A61K38/191—Tumor necrosis factors [TNF], e.g. lymphotoxin [LT], i.e. TNF-beta
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    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
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    • C—CHEMISTRY; METALLURGY
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    • C07K14/705—Receptors; Cell surface antigens; Cell surface determinants
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    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
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    • C07K14/705—Receptors; Cell surface antigens; Cell surface determinants
    • C07K14/715—Receptors; Cell surface antigens; Cell surface determinants for cytokines; for lymphokines; for interferons
    • C07K14/7151—Receptors; Cell surface antigens; Cell surface determinants for cytokines; for lymphokines; for interferons for tumor necrosis factor [TNF], for lymphotoxin [LT]
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    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/81—Protease inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K2319/00—Fusion polypeptide
    • C07K2319/30—Non-immunoglobulin-derived peptide or protein having an immunoglobulin constant or Fc region, or a fragment thereof, attached thereto

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  • Health & Medical Sciences (AREA)
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  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Dermatology (AREA)
  • Cell Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Toxicology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Reproductive Health (AREA)
  • Inorganic Chemistry (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Hematology (AREA)
TW101138560A 2011-10-18 2012-10-18 用氯化鈉穩定化之依那西普調配物 TW201325606A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161548518P 2011-10-18 2011-10-18
US201261669480P 2012-07-09 2012-07-09

Publications (1)

Publication Number Publication Date
TW201325606A true TW201325606A (zh) 2013-07-01

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ID=48136153

Family Applications (6)

Application Number Title Priority Date Filing Date
TW101138560A TW201325606A (zh) 2011-10-18 2012-10-18 用氯化鈉穩定化之依那西普調配物
TW101138565A TWI644681B (zh) 2011-10-18 2012-10-18 用金屬離子穩定化之依那西普調配物
TW101138564A TW201325608A (zh) 2011-10-18 2012-10-18 用糖及多元醇之組合穩定化之依那西普調配物
TW101138566A TWI619504B (zh) 2011-10-18 2012-10-18 用美洛明穩定化之依那西普調配物
TW101138561A TW201325607A (zh) 2011-10-18 2012-10-18 用胺基酸穩定化之依那西普調配物
TW101138567A TWI595883B (zh) 2011-10-18 2012-10-18 用木糖醇穩定化之依那西普調配物

Family Applications After (5)

Application Number Title Priority Date Filing Date
TW101138565A TWI644681B (zh) 2011-10-18 2012-10-18 用金屬離子穩定化之依那西普調配物
TW101138564A TW201325608A (zh) 2011-10-18 2012-10-18 用糖及多元醇之組合穩定化之依那西普調配物
TW101138566A TWI619504B (zh) 2011-10-18 2012-10-18 用美洛明穩定化之依那西普調配物
TW101138561A TW201325607A (zh) 2011-10-18 2012-10-18 用胺基酸穩定化之依那西普調配物
TW101138567A TWI595883B (zh) 2011-10-18 2012-10-18 用木糖醇穩定化之依那西普調配物

Country Status (28)

Country Link
US (21) US9302002B2 (https=)
EP (6) EP2768854A4 (https=)
JP (6) JP6220788B2 (https=)
KR (7) KR20140079491A (https=)
CN (6) CN104010657A (https=)
AR (6) AR088383A1 (https=)
AU (6) AU2012326171B2 (https=)
BR (6) BR112014009146A8 (https=)
CA (6) CA2851642A1 (https=)
CY (1) CY1121843T1 (https=)
DK (1) DK2768525T3 (https=)
EA (6) EA025267B1 (https=)
ES (1) ES2734070T3 (https=)
HK (3) HK1200718A1 (https=)
HR (1) HRP20191215T1 (https=)
HU (1) HUE045624T2 (https=)
IL (6) IL231826A0 (https=)
IN (3) IN2014CN02527A (https=)
LT (1) LT2768525T (https=)
MX (7) MX2014004725A (https=)
PL (1) PL2768525T3 (https=)
PT (1) PT2768525T (https=)
RS (1) RS59179B1 (https=)
SG (6) SG11201401576WA (https=)
SI (1) SI2768525T1 (https=)
SM (1) SMT201900422T1 (https=)
TW (6) TW201325606A (https=)
WO (6) WO2013059408A1 (https=)

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