TW201102378A - Polymorphic form D of bazedoxifene acetate and methods of preparing same - Google Patents
Polymorphic form D of bazedoxifene acetate and methods of preparing same Download PDFInfo
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- TW201102378A TW201102378A TW099120246A TW99120246A TW201102378A TW 201102378 A TW201102378 A TW 201102378A TW 099120246 A TW099120246 A TW 099120246A TW 99120246 A TW99120246 A TW 99120246A TW 201102378 A TW201102378 A TW 201102378A
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- acetate
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Rheumatology (AREA)
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- Hematology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT001109A ITMI20091109A1 (it) | 2009-06-23 | 2009-06-23 | Forma polimorfa d di bazedoxifene acetato e metodi per la sua preparazione |
| US24496109P | 2009-09-23 | 2009-09-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW201102378A true TW201102378A (en) | 2011-01-16 |
Family
ID=42035899
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW099120246A TW201102378A (en) | 2009-06-23 | 2010-06-22 | Polymorphic form D of bazedoxifene acetate and methods of preparing same |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US8063041B2 (enExample) |
| EP (1) | EP2445876A1 (enExample) |
| JP (4) | JP2011037832A (enExample) |
| AR (1) | AR077203A1 (enExample) |
| CA (1) | CA2766618A1 (enExample) |
| IT (1) | ITMI20091109A1 (enExample) |
| TW (1) | TW201102378A (enExample) |
| WO (1) | WO2010151541A1 (enExample) |
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| TWI577285B (zh) | 2007-08-13 | 2017-04-11 | 孟山都科技有限責任公司 | 控制植物寄生性線蟲的化合物及方法以及被覆有該化合物之種子 |
| EP2616463A4 (en) * | 2010-09-14 | 2014-01-08 | Reddys Lab Ltd Dr | PREPARATION OF CRYSTALLINE BAZEDOXIFES AND THEIR SALTS |
| WO2013182169A1 (en) | 2012-06-07 | 2013-12-12 | Zentiva, K. S. | Process of preparation of an antioxidant-free polymorphically and chemically stable formulation of bazedoxifene acetate |
| WO2013182170A1 (en) | 2012-06-07 | 2013-12-12 | Zentiva, K. S. | Enhancement of dissolution rate from pharmaceutical composition comprising bazedoxifene acetate |
| UA118254C2 (uk) | 2012-12-04 | 2018-12-26 | Монсанто Текнолоджи Ллс | Нематоцидні водні композиції концентрату суспензії |
| CN103864664A (zh) * | 2012-12-18 | 2014-06-18 | 江苏柯菲平医药有限公司 | 巴多昔芬乙酸盐新晶型及其制备方法 |
| CN103864665B (zh) * | 2014-03-04 | 2016-03-02 | 苏州特瑞药业有限公司 | 醋酸巴多昔芬的制备方法 |
| CN104370796B (zh) * | 2014-11-21 | 2016-09-14 | 扬子江药业集团有限公司 | 一种醋酸巴多昔芬多晶型b的制备方法 |
| JP6863547B2 (ja) | 2015-06-18 | 2021-04-21 | エステトラ ソシエテ プリーヴ ア レスポンサビリテ リミテ | エステトロール成分を含有する口腔内崩壊性投与単位 |
| GEP20217243B (en) | 2015-06-18 | 2021-04-26 | Sprl Estetra | Orodispersible dosage unit containing an estetrol component |
| CA3178291A1 (en) | 2016-08-05 | 2018-04-12 | Estetra Srl | Method for the management of dysmenorrhea and menstrual pain |
| KR20190096462A (ko) | 2018-01-08 | 2019-08-20 | (주)휴온스 | 바제독시펜 아세테이트 결정형 d형을 포함하는 안정성이 증가된 약제학적 조성물 및 그 제조방법 |
| JOP20200260A1 (ar) * | 2018-04-19 | 2019-10-19 | Estetra Sprl | مركبات واستخداماتها للتخفيف من الأعراض المصاحبة لانقطاع الطمث |
| TWI801561B (zh) | 2018-04-19 | 2023-05-11 | 比利時商依思特拉私人有限責任公司 | 化合物及其用於緩解絕經相關症狀的用途 |
| CN109851547B (zh) * | 2018-12-27 | 2020-09-08 | 北京鑫开元医药科技有限公司 | 一种醋酸巴多昔芬晶型d的制备方法及用途 |
| KR20190132311A (ko) | 2019-11-15 | 2019-11-27 | (주)휴온스 | 바제독시펜 아세테이트 결정형 d형을 포함하는 안정성이 증가된 약제학적 조성물 및 그 제조방법 |
| CN111004165A (zh) * | 2019-12-03 | 2020-04-14 | 南京正济医药研究有限公司 | 一种醋酸巴多昔芬晶型a的制备方法 |
| TWI893101B (zh) | 2020-04-16 | 2025-08-11 | 比利時商埃斯特拉有限責任公司 | 具有降低之副作用之避孕組成物 |
| US11246874B1 (en) | 2021-04-20 | 2022-02-15 | Oxygen Biotech LLC | Treatment of COVID-19 |
| CN113244240A (zh) * | 2021-05-26 | 2021-08-13 | 深圳市人民医院 | 醋酸巴多昔芬在治疗急性髓系白血病药物中的应用 |
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|---|---|---|---|---|
| US2772508A (en) | 1954-04-28 | 1956-12-04 | Claude A Greenlee | Fish line pullaway sinker |
| ATE206701T1 (de) | 1996-04-19 | 2001-10-15 | American Home Prod | Östrogene verbindungen |
| US5998402A (en) * | 1996-04-19 | 1999-12-07 | American Home Products Corporation | 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents |
| US6479535B1 (en) | 1998-05-15 | 2002-11-12 | Wyeth | 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indole and estrogen formulations |
| AR029538A1 (es) | 2000-07-06 | 2003-07-02 | Wyeth Corp | Composiciones farmaceuticas de agentes estrogenicos |
| NZ537051A (en) | 2002-06-13 | 2007-11-30 | Wyeth Corp | Use of bazedoxifene in an extended dosage treatment regimen |
| JP2007532560A (ja) * | 2004-04-07 | 2007-11-15 | ワイス | バゼドキシフェンアセテートの結晶多形 |
| TW200536845A (en) * | 2004-04-07 | 2005-11-16 | Wyeth Corp | Crystalline polymorph of bazedoxifene acetate |
| MXPA06011685A (es) * | 2004-04-08 | 2006-12-14 | Wyeth Corp | Formulaciones de dispersiones solidas de acetato de bazedoxifeno. |
| CN101304731B (zh) | 2005-08-24 | 2012-06-20 | 惠氏公司 | 醋酸苯卓昔芬制剂及其生产方法 |
| CZ302358B6 (cs) * | 2007-07-25 | 2011-03-30 | Zentiva, A. S. | Nové soli bazedoxifenu |
-
2009
- 2009-06-23 IT IT001109A patent/ITMI20091109A1/it unknown
-
2010
- 2010-06-22 EP EP10728533A patent/EP2445876A1/en not_active Withdrawn
- 2010-06-22 US US12/820,593 patent/US8063041B2/en active Active
- 2010-06-22 CA CA2766618A patent/CA2766618A1/en not_active Abandoned
- 2010-06-22 WO PCT/US2010/039488 patent/WO2010151541A1/en not_active Ceased
- 2010-06-22 TW TW099120246A patent/TW201102378A/zh unknown
- 2010-06-22 JP JP2010141370A patent/JP2011037832A/ja active Pending
- 2010-06-23 AR ARP100102214A patent/AR077203A1/es not_active Application Discontinuation
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2015
- 2015-12-04 JP JP2015237242A patent/JP2016033165A/ja active Pending
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2017
- 2017-05-22 JP JP2017100527A patent/JP2017137360A/ja active Pending
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2018
- 2018-07-30 JP JP2018142063A patent/JP2018162327A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JP2011037832A (ja) | 2011-02-24 |
| ITMI20091109A1 (it) | 2010-12-24 |
| US20110021504A1 (en) | 2011-01-27 |
| WO2010151541A1 (en) | 2010-12-29 |
| AR077203A1 (es) | 2011-08-10 |
| US8063041B2 (en) | 2011-11-22 |
| JP2016033165A (ja) | 2016-03-10 |
| CA2766618A1 (en) | 2010-12-29 |
| JP2017137360A (ja) | 2017-08-10 |
| WO2010151541A8 (en) | 2011-05-12 |
| JP2018162327A (ja) | 2018-10-18 |
| EP2445876A1 (en) | 2012-05-02 |
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