TW200722098A - Facially amphiphilic polymers and oligomers, compositions thereof, and use thereof in pharmaceutical compositions for treating cancer - Google Patents

Facially amphiphilic polymers and oligomers, compositions thereof, and use thereof in pharmaceutical compositions for treating cancer

Info

Publication number
TW200722098A
TW200722098A TW095106642A TW95106642A TW200722098A TW 200722098 A TW200722098 A TW 200722098A TW 095106642 A TW095106642 A TW 095106642A TW 95106642 A TW95106642 A TW 95106642A TW 200722098 A TW200722098 A TW 200722098A
Authority
TW
Taiwan
Prior art keywords
compositions
oligomers
amphiphilic polymers
treating cancer
pharmaceutical compositions
Prior art date
Application number
TW095106642A
Other languages
English (en)
Chinese (zh)
Inventor
William Frank Degrado
Gregory N Tew
Lachelle S Arnt
Original Assignee
Univ Pennsylvania
Univ Massachusetts
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Pennsylvania, Univ Massachusetts filed Critical Univ Pennsylvania
Publication of TW200722098A publication Critical patent/TW200722098A/zh

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/10—Peptides having 12 to 20 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Indole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
TW095106642A 2005-02-25 2006-02-27 Facially amphiphilic polymers and oligomers, compositions thereof, and use thereof in pharmaceutical compositions for treating cancer TW200722098A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US65609205P 2005-02-25 2005-02-25

Publications (1)

Publication Number Publication Date
TW200722098A true TW200722098A (en) 2007-06-16

Family

ID=36941658

Family Applications (2)

Application Number Title Priority Date Filing Date
TW095106642A TW200722098A (en) 2005-02-25 2006-02-27 Facially amphiphilic polymers and oligomers, compositions thereof, and use thereof in pharmaceutical compositions for treating cancer
TW101108505A TW201231063A (en) 2005-02-25 2006-02-27 Facially amphiphilic polymers and oligomers, compositions thereof, and use thereof in pharmaceutical compositions for treating cancer

Family Applications After (1)

Application Number Title Priority Date Filing Date
TW101108505A TW201231063A (en) 2005-02-25 2006-02-27 Facially amphiphilic polymers and oligomers, compositions thereof, and use thereof in pharmaceutical compositions for treating cancer

Country Status (8)

Country Link
US (1) US20060241052A1 (https=)
EP (5) EP2301349A2 (https=)
JP (1) JP2008531585A (https=)
KR (1) KR20080004475A (https=)
AU (1) AU2006218805A1 (https=)
CA (1) CA2599205A1 (https=)
TW (2) TW200722098A (https=)
WO (1) WO2006093813A2 (https=)

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EP2471526A3 (en) 2003-03-17 2012-12-12 The Trustees Of The University Of Pennsylvania Facially amphiphillic polymers and oligomers and uses thereof
CN1922133A (zh) 2004-01-23 2007-02-28 宾夕法尼亚州大学理事会 表面两亲性聚芳基和聚芳基炔基聚合物和低聚物及其用途
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RU2530899C2 (ru) 2008-07-28 2014-10-20 Селлсьютикс Корпорейшн Противомалярийные соединения
TWI478915B (zh) 2008-10-27 2015-04-01 Cellceutix Corp 宿主防禦之合成模擬物及其用途
CA2746421A1 (en) * 2008-12-10 2010-06-17 Polymedix, Inc. Antimicrobial molecules for treating multi-drug resistant and extensively drug resistant strains of mycobacterium
KR101094299B1 (ko) 2009-12-17 2011-12-19 삼성모바일디스플레이주식회사 선형 증발원 및 이를 포함하는 증착 장치
EP2709619B1 (en) 2011-05-16 2017-10-11 Cellceutix Corporation Compounds for use in treatment of mucositis
AU2012352621A1 (en) 2011-12-13 2014-07-24 Cellceutix Corporation Cyclic compounds and methods of making and using the same
MX2014008763A (es) * 2012-01-18 2015-04-13 Cellceutix Corp Compuestos y metodos para tratar infecciones por candidosis y aspergillus.
CN109305926B (zh) * 2018-10-18 2021-06-25 吉林大学 一种可形成分子内氢键的芳酰胺类金属配体及其制备方法与应用
WO2021248008A1 (en) 2020-06-05 2021-12-09 Innovation Pharmaceuticals Inc. Arylamide compounds for treatment and prevention of viral infections

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Also Published As

Publication number Publication date
EP1855704A2 (en) 2007-11-21
EP2301349A2 (en) 2011-03-30
JP2008531585A (ja) 2008-08-14
CA2599205A1 (en) 2006-09-08
EP2298074A3 (en) 2011-10-26
EP2298074A2 (en) 2011-03-23
WO2006093813A3 (en) 2007-11-22
EP1855704A4 (en) 2009-12-02
KR20080004475A (ko) 2008-01-09
US20060241052A1 (en) 2006-10-26
WO2006093813A2 (en) 2006-09-08
AU2006218805A1 (en) 2006-09-08
EP2433628A1 (en) 2012-03-28
TW201231063A (en) 2012-08-01
EP2433627A1 (en) 2012-03-28

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