TW200604137A - Coupling process for generating reactive boron-containing derivatives of n-substituted pyrrole-2-carbonitriles to produce biaryls - Google Patents

Coupling process for generating reactive boron-containing derivatives of n-substituted pyrrole-2-carbonitriles to produce biaryls

Info

Publication number
TW200604137A
TW200604137A TW094113123A TW94113123A TW200604137A TW 200604137 A TW200604137 A TW 200604137A TW 094113123 A TW094113123 A TW 094113123A TW 94113123 A TW94113123 A TW 94113123A TW 200604137 A TW200604137 A TW 200604137A
Authority
TW
Taiwan
Prior art keywords
carbonitriles
boron
coupling process
containing derivatives
substituted pyrrole
Prior art date
Application number
TW094113123A
Other languages
English (en)
Inventor
Bogdan Kazimierz Wilk
Arkadiy Zinoviy Rubezhov
Jean Louise Helom
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of TW200604137A publication Critical patent/TW200604137A/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TW094113123A 2004-04-27 2005-04-25 Coupling process for generating reactive boron-containing derivatives of n-substituted pyrrole-2-carbonitriles to produce biaryls TW200604137A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56563604P 2004-04-27 2004-04-27
US64765605P 2005-01-27 2005-01-27

Publications (1)

Publication Number Publication Date
TW200604137A true TW200604137A (en) 2006-02-01

Family

ID=34967855

Family Applications (1)

Application Number Title Priority Date Filing Date
TW094113123A TW200604137A (en) 2004-04-27 2005-04-25 Coupling process for generating reactive boron-containing derivatives of n-substituted pyrrole-2-carbonitriles to produce biaryls

Country Status (7)

Country Link
US (2) US7446211B2 (zh)
AR (1) AR049631A1 (zh)
PA (1) PA8631101A1 (zh)
PE (1) PE20060331A1 (zh)
SV (1) SV2005002092A (zh)
TW (1) TW200604137A (zh)
WO (1) WO2005105817A2 (zh)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA06012402A (es) 2004-04-27 2007-01-17 Wyeth Corp Carbamato y tiocarbamato biarilos ciclicos que contienen cianopirrol y metodos para preparar los mismos.
US7446211B2 (en) 2004-04-27 2008-11-04 Wyeth Coupling process for generating reactive boron-containing derivatives of N-substituted pyrrole-2-carbonitriles to produce biaryls
GT200500185A (es) * 2004-08-09 2006-04-10 Moduladores del receptor de progesterona que comprenden derivados de pirrol-oxindol y sus usos
CA2575737C (en) * 2004-08-13 2013-09-24 Wyeth Tanaproget derivatives, metabolites, and uses thereof
EP1877059B8 (en) 2005-04-28 2010-05-19 Wyeth a Corporation of the State of Delaware Micronized tanaproget and compostions containing same
BRPI0610156A2 (pt) * 2005-04-28 2016-08-16 Wyeth Corp forma micronizada de um composto, forma purificada i do composto, kit, padrão de referência, e, método de preparaçao de uma composição farmacêutica.
CN101166736B (zh) 2005-04-28 2013-02-06 惠氏公司 他那普戈特的多晶型ⅱ
ATE460937T1 (de) 2005-04-28 2010-04-15 Wyeth Corp Mikronisierte tanaproget zusammensetzungen und verfahren zu ihrer herstellung
PE20070220A1 (es) 2005-07-29 2007-03-19 Wyeth Corp Proceso para la sintesis de moduladores del receptor de progesterona
US20070213526A1 (en) * 2006-03-07 2007-09-13 Wyeth Purification of progesterone receptor modulators
AU2008211047B2 (en) 2007-01-29 2013-07-25 Wako Pure Chemical Industries, Ltd. Reagent for organic synthesis reaction containing organic triol borate salt
US20080319204A1 (en) * 2007-06-25 2008-12-25 Wyeth Process for the synthesis of progesterone receptor modulators
US20090170823A1 (en) * 2007-12-20 2009-07-02 Duramed Pharmaceuticals, Inc. Dosage Regimens and Pharmaceutical Compositions and Packages for Emergency Contraception
WO2021226269A1 (en) 2020-05-05 2021-11-11 Nuvalent, Inc. Heteroaromatic macrocyclic ether chemotherapeutic agents
EP4146626A4 (en) 2020-05-05 2024-05-29 Nuvalent Inc CHEMOTHERAPEUTIC AGENTS BASED ON HETEROAROMATIC MACROCYCLIC ETHERS

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MX9206628A (es) * 1991-11-22 1993-05-01 Boehringer Ingelheim Pharma Ester de prolinaboronato y metodo para su preparacion.
KR960704886A (ko) 1993-09-10 1996-10-09 베르너 발데크 포토크롬 화합물, 그의 제조 방법과 제조 중간체 및 그의 용도 (Photochromic Compounds, Methods and Intermediates for Producing Them and Their Use)
EP1192189B1 (en) 1999-02-22 2004-09-29 Eastman Chemical Company Catalysts containing n-pyrrolyl substituted nitrogen donors
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US7446211B2 (en) 2004-04-27 2008-11-04 Wyeth Coupling process for generating reactive boron-containing derivatives of N-substituted pyrrole-2-carbonitriles to produce biaryls

Also Published As

Publication number Publication date
SV2005002092A (es) 2005-12-13
PA8631101A1 (es) 2006-09-08
WO2005105817A3 (en) 2006-01-12
PE20060331A1 (es) 2006-05-16
US7446211B2 (en) 2008-11-04
WO2005105817A2 (en) 2005-11-10
US8129523B2 (en) 2012-03-06
US20050272702A1 (en) 2005-12-08
AR049631A1 (es) 2006-08-23
US20090054663A1 (en) 2009-02-26

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