SV2005002092A - " proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos " ref. am - 101481salvo. - Google Patents

" proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos " ref. am - 101481salvo.

Info

Publication number
SV2005002092A
SV2005002092A SV2005002092A SV2005002092A SV2005002092A SV 2005002092 A SV2005002092 A SV 2005002092A SV 2005002092 A SV2005002092 A SV 2005002092A SV 2005002092 A SV2005002092 A SV 2005002092A SV 2005002092 A SV2005002092 A SV 2005002092A
Authority
SV
El Salvador
Prior art keywords
boro
content
pirrol
carbonitrile
biarilos
Prior art date
Application number
SV2005002092A
Other languages
English (en)
Inventor
Bogdan Kazimierz Wilk
Arkadiy Zinoviy Rubezhov
Jean Louise Helom
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of SV2005002092A publication Critical patent/SV2005002092A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Abstract

SE PRESENTA UNA PREPARACION CONVENIENTE DE COMPUESTOS CON CONTENIDO DE BORO COMPUESTOS DE PIRROLCARBONITRILO CON CONTENIDO DE BORO, COMPUESTOS DE PIRROL-2-CARBONITRILO N-SUSTITUIDOS CON CONTENIDO DE BORO Y DERIVADOS DE LOS MISMOS. LA PRESENTE INVENCION PRESENTA ASIMISMO EL USO DE ESTOS COMPUESTOS CON CONTENIDO DE BORO Y DERIVADOS DE LOS MISMOS EN REACCIONES DE ACOPLAMIENTO PARA LA PRODUCCION DE COMPUESTOS DE BIARILO
SV2005002092A 2004-04-27 2005-04-25 " proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos " ref. am - 101481salvo. SV2005002092A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56563604P 2004-04-27 2004-04-27
US64765605P 2005-01-27 2005-01-27

Publications (1)

Publication Number Publication Date
SV2005002092A true SV2005002092A (es) 2005-12-13

Family

ID=34967855

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2005002092A SV2005002092A (es) 2004-04-27 2005-04-25 " proceso de acoplamiento para la generacion de derivados reactivos de pirrol-2-carbonitrilo n-sustituidos con contenido de boro para producir biarilos " ref. am - 101481salvo.

Country Status (7)

Country Link
US (2) US7446211B2 (es)
AR (1) AR049631A1 (es)
PA (1) PA8631101A1 (es)
PE (1) PE20060331A1 (es)
SV (1) SV2005002092A (es)
TW (1) TW200604137A (es)
WO (1) WO2005105817A2 (es)

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BRPI0510278A (pt) 2004-04-27 2007-10-30 Wyeth Corp método para produzir compostos, produto, e, composto
AR049631A1 (es) 2004-04-27 2006-08-23 Wyeth Corp Proceso de acoplamiento para la generacion de derivados reactivos de pirrol -2- carbonitrilo n- sustituidos con contenido de boro para producir biarilos
GT200500185A (es) * 2004-08-09 2006-04-10 Moduladores del receptor de progesterona que comprenden derivados de pirrol-oxindol y sus usos
US7569679B2 (en) * 2004-08-13 2009-08-04 Wyeth Tanaproget derivatives, metabolites, and uses thereof
DK1896034T3 (da) 2005-04-28 2010-05-17 Wyeth Corp Mikroniserede tanaproget-sammensætninger og fremgangsmåder til fremstilling af disse
MX2007013469A (es) 2005-04-28 2008-01-22 Wyeth Corp Forma ii polimorfa de tanaproget.
US7786297B2 (en) * 2005-04-28 2010-08-31 Wyeth Llc Purified form of tanaproget
EP1877059B8 (en) 2005-04-28 2010-05-19 Wyeth a Corporation of the State of Delaware Micronized tanaproget and compostions containing same
PE20070220A1 (es) 2005-07-29 2007-03-19 Wyeth Corp Proceso para la sintesis de moduladores del receptor de progesterona
US20070213526A1 (en) * 2006-03-07 2007-09-13 Wyeth Purification of progesterone receptor modulators
WO2008093637A1 (ja) 2007-01-29 2008-08-07 Wako Pure Chemical Industries, Ltd. 有機トリオールボレート塩を含んでなる有機合成反応用試薬
US20080319204A1 (en) * 2007-06-25 2008-12-25 Wyeth Process for the synthesis of progesterone receptor modulators
WO2009082478A1 (en) 2007-12-20 2009-07-02 Duramed Pharmaceuticals, Inc. Dosage regimens and pharmaceutical compositions and packages for emergency contraception
JP2023525040A (ja) 2020-05-05 2023-06-14 ヌバレント， インク． ヘテロ芳香族大環状エーテル化学療法剤
CN115916754A (zh) 2020-05-05 2023-04-04 纽威伦特公司 杂芳族大环醚化学治疗剂

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Also Published As

Publication number Publication date
US20090054663A1 (en) 2009-02-26
TW200604137A (en) 2006-02-01
PE20060331A1 (es) 2006-05-16
WO2005105817A3 (en) 2006-01-12
PA8631101A1 (es) 2006-09-08
US8129523B2 (en) 2012-03-06
WO2005105817A2 (en) 2005-11-10
US7446211B2 (en) 2008-11-04
AR049631A1 (es) 2006-08-23
US20050272702A1 (en) 2005-12-08

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