BR0112861A - Processo para o preparo de 2-(4-piridil)amino-6-dialquilóxifenil-pirido[2,3-d]pirimi din-7-onas - Google Patents
Processo para o preparo de 2-(4-piridil)amino-6-dialquilóxifenil-pirido[2,3-d]pirimi din-7-onasInfo
- Publication number
- BR0112861A BR0112861A BR0112861-2A BR0112861A BR0112861A BR 0112861 A BR0112861 A BR 0112861A BR 0112861 A BR0112861 A BR 0112861A BR 0112861 A BR0112861 A BR 0112861A
- Authority
- BR
- Brazil
- Prior art keywords
- pyrido
- pyridyl
- amino
- dialkyloxyphenyl
- pyrimidin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
Abstract
"PROCESSO PARA O PREPARO DE 2-(4-PIRIDIL)AMINO-6-DIALQUILóXIFENIL-PIRIDO[2,3-D]PIRIMI DIN-7-ONAS". Processo para o preparo de 2-piridilamino-pirido[2,3-d]pirimidinas da Fórmula (II) em que Ar é arila, R' e R" são hidrogênio, alquila, alcóxi e R^ 2^ é alquila.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US22308400P | 2000-08-04 | 2000-08-04 | |
PCT/US2001/022001 WO2002012237A2 (en) | 2000-08-04 | 2001-07-12 | Process for preparing 2-(4-pyridyl)amino-6-dialkyloxyphenyl-pyrido[2,3-d]pyrimidin-7-ones |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0112861A true BR0112861A (pt) | 2003-07-01 |
Family
ID=22834962
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0112861-2A BR0112861A (pt) | 2000-08-04 | 2001-07-12 | Processo para o preparo de 2-(4-piridil)amino-6-dialquilóxifenil-pirido[2,3-d]pirimi din-7-onas |
Country Status (9)
Country | Link |
---|---|
US (1) | US6960662B2 (pt) |
EP (1) | EP1307451A2 (pt) |
JP (1) | JP2004505974A (pt) |
AR (1) | AR030571A1 (pt) |
AU (1) | AU2001278908A1 (pt) |
BR (1) | BR0112861A (pt) |
CA (1) | CA2417937A1 (pt) |
MX (1) | MXPA03000289A (pt) |
WO (1) | WO2002012237A2 (pt) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AP1333A (en) * | 2000-08-04 | 2004-11-28 | Warner Lambert Co | 2-(4-pyridyl) amino-6-dialkoxyphenyl-pyrido [2,3-d] pyrimidin-7-ones. |
JP2005507392A (ja) * | 2000-08-04 | 2005-03-17 | ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー | 2−(4−ピリジル)アミノ−6−ジアルキルオキシフェニルピリド〔2,3−d〕ピリミジン−7−オン類の製造方法 |
US7196090B2 (en) * | 2002-07-25 | 2007-03-27 | Warner-Lambert Company | Kinase inhibitors |
US7098332B2 (en) | 2002-12-20 | 2006-08-29 | Hoffmann-La Roche Inc. | 5,8-Dihydro-6H-pyrido[2,3-d]pyrimidin-7-ones |
GB0230019D0 (en) * | 2002-12-23 | 2003-01-29 | Syngenta Ltd | Fungicides |
CA2555724A1 (en) * | 2004-02-18 | 2005-09-09 | Warner-Lambert Company Llc | 2-(pyridin-3-ylamino)-pyrido[2,3-d]pyrimidin-7-ones |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1336904C (en) | 1987-08-26 | 1995-09-05 | Mitsuyuki Takesue | Pyrimidines and their pharmaceutically acceptable salts thereof |
DE4408404A1 (de) | 1994-03-12 | 1995-09-14 | Huels Chemische Werke Ag | Verfahren zur Herstellung von Chlorpyrimidinen |
US5801183A (en) | 1995-01-27 | 1998-09-01 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon | Aza and aza (N-oxy) analogs of glycine/NMDA receptor antagonists |
IL117923A (en) | 1995-05-03 | 2000-06-01 | Warner Lambert Co | Anti-cancer pharmaceutical compositions containing polysubstituted pyrido¬2,3-d¾pyrimidine derivatives and certain such novel compounds |
US5620981A (en) * | 1995-05-03 | 1997-04-15 | Warner-Lambert Company | Pyrido [2,3-D]pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation |
US5945422A (en) * | 1997-02-05 | 1999-08-31 | Warner-Lambert Company | N-oxides of amino containing pyrido 2,3-D! pyrimidines |
CZ301369B6 (cs) | 1998-03-13 | 2010-02-03 | Syngenta Participations Ag | Herbicidne aktivní deriváty 3-hydroxy-4-aryl-5-oxopyrazolinu |
PL343112A1 (en) | 1998-03-31 | 2001-07-30 | Warner Lambert Co | Quinolones as serine protease inhibitors |
AP1333A (en) * | 2000-08-04 | 2004-11-28 | Warner Lambert Co | 2-(4-pyridyl) amino-6-dialkoxyphenyl-pyrido [2,3-d] pyrimidin-7-ones. |
JP2005507392A (ja) * | 2000-08-04 | 2005-03-17 | ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー | 2−(4−ピリジル)アミノ−6−ジアルキルオキシフェニルピリド〔2,3−d〕ピリミジン−7−オン類の製造方法 |
DE60303009T2 (de) * | 2002-01-22 | 2006-07-13 | Warner-Lambert Co. Llc | 2-(pyridin-2-ylamino)-pyrido[2,3-d]pyrimidin-7-one |
-
2001
- 2001-07-12 JP JP2002518212A patent/JP2004505974A/ja active Pending
- 2001-07-12 AU AU2001278908A patent/AU2001278908A1/en not_active Abandoned
- 2001-07-12 WO PCT/US2001/022001 patent/WO2002012237A2/en active Application Filing
- 2001-07-12 EP EP01957137A patent/EP1307451A2/en not_active Withdrawn
- 2001-07-12 CA CA002417937A patent/CA2417937A1/en not_active Abandoned
- 2001-07-12 BR BR0112861-2A patent/BR0112861A/pt not_active IP Right Cessation
- 2001-07-12 US US10/343,805 patent/US6960662B2/en not_active Expired - Fee Related
- 2001-07-12 MX MXPA03000289A patent/MXPA03000289A/es active IP Right Grant
- 2001-08-03 AR ARP010103717A patent/AR030571A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2002012237A2 (en) | 2002-02-14 |
AR030571A1 (es) | 2003-08-27 |
AU2001278908A1 (en) | 2002-02-18 |
US20030216415A1 (en) | 2003-11-20 |
JP2004505974A (ja) | 2004-02-26 |
CA2417937A1 (en) | 2002-02-14 |
US6960662B2 (en) | 2005-11-01 |
EP1307451A2 (en) | 2003-05-07 |
WO2002012237A3 (en) | 2002-05-10 |
MXPA03000289A (es) | 2003-06-06 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7O E 8O ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2021 DE 29/09/2009. |