BR0112861A - Processo para o preparo de 2-(4-piridil)amino-6-dialquilóxifenil-pirido[2,3-d]pirimi din-7-onas - Google Patents

Processo para o preparo de 2-(4-piridil)amino-6-dialquilóxifenil-pirido[2,3-d]pirimi din-7-onas

Info

Publication number
BR0112861A
BR0112861A BR0112861-2A BR0112861A BR0112861A BR 0112861 A BR0112861 A BR 0112861A BR 0112861 A BR0112861 A BR 0112861A BR 0112861 A BR0112861 A BR 0112861A
Authority
BR
Brazil
Prior art keywords
pyrido
pyridyl
amino
dialkyloxyphenyl
pyrimidin
Prior art date
Application number
BR0112861-2A
Other languages
English (en)
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of BR0112861A publication Critical patent/BR0112861A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

"PROCESSO PARA O PREPARO DE 2-(4-PIRIDIL)AMINO-6-DIALQUILóXIFENIL-PIRIDO[2,3-D]PIRIMI DIN-7-ONAS". Processo para o preparo de 2-piridilamino-pirido[2,3-d]pirimidinas da Fórmula (II) em que Ar é arila, R' e R" são hidrogênio, alquila, alcóxi e R^ 2^ é alquila.
BR0112861-2A 2000-08-04 2001-07-12 Processo para o preparo de 2-(4-piridil)amino-6-dialquilóxifenil-pirido[2,3-d]pirimi din-7-onas BR0112861A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22308400P 2000-08-04 2000-08-04
PCT/US2001/022001 WO2002012237A2 (en) 2000-08-04 2001-07-12 Process for preparing 2-(4-pyridyl)amino-6-dialkyloxyphenyl-pyrido[2,3-d]pyrimidin-7-ones

Publications (1)

Publication Number Publication Date
BR0112861A true BR0112861A (pt) 2003-07-01

Family

ID=22834962

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0112861-2A BR0112861A (pt) 2000-08-04 2001-07-12 Processo para o preparo de 2-(4-piridil)amino-6-dialquilóxifenil-pirido[2,3-d]pirimi din-7-onas

Country Status (9)

Country Link
US (1) US6960662B2 (pt)
EP (1) EP1307451A2 (pt)
JP (1) JP2004505974A (pt)
AR (1) AR030571A1 (pt)
AU (1) AU2001278908A1 (pt)
BR (1) BR0112861A (pt)
CA (1) CA2417937A1 (pt)
MX (1) MXPA03000289A (pt)
WO (1) WO2002012237A2 (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AP1333A (en) * 2000-08-04 2004-11-28 Warner Lambert Co 2-(4-pyridyl) amino-6-dialkoxyphenyl-pyrido [2,3-d] pyrimidin-7-ones.
JP2005507392A (ja) * 2000-08-04 2005-03-17 ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー 2−(4−ピリジル)アミノ−6−ジアルキルオキシフェニルピリド〔2,3−d〕ピリミジン−7−オン類の製造方法
US7196090B2 (en) * 2002-07-25 2007-03-27 Warner-Lambert Company Kinase inhibitors
US7098332B2 (en) 2002-12-20 2006-08-29 Hoffmann-La Roche Inc. 5,8-Dihydro-6H-pyrido[2,3-d]pyrimidin-7-ones
GB0230019D0 (en) * 2002-12-23 2003-01-29 Syngenta Ltd Fungicides
CA2555724A1 (en) * 2004-02-18 2005-09-09 Warner-Lambert Company Llc 2-(pyridin-3-ylamino)-pyrido[2,3-d]pyrimidin-7-ones

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1336904C (en) 1987-08-26 1995-09-05 Mitsuyuki Takesue Pyrimidines and their pharmaceutically acceptable salts thereof
DE4408404A1 (de) 1994-03-12 1995-09-14 Huels Chemische Werke Ag Verfahren zur Herstellung von Chlorpyrimidinen
US5801183A (en) 1995-01-27 1998-09-01 State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon Aza and aza (N-oxy) analogs of glycine/NMDA receptor antagonists
IL117923A (en) 1995-05-03 2000-06-01 Warner Lambert Co Anti-cancer pharmaceutical compositions containing polysubstituted pyrido¬2,3-d¾pyrimidine derivatives and certain such novel compounds
US5620981A (en) * 1995-05-03 1997-04-15 Warner-Lambert Company Pyrido [2,3-D]pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation
US5945422A (en) * 1997-02-05 1999-08-31 Warner-Lambert Company N-oxides of amino containing pyrido 2,3-D! pyrimidines
CZ301369B6 (cs) 1998-03-13 2010-02-03 Syngenta Participations Ag Herbicidne aktivní deriváty 3-hydroxy-4-aryl-5-oxopyrazolinu
PL343112A1 (en) 1998-03-31 2001-07-30 Warner Lambert Co Quinolones as serine protease inhibitors
AP1333A (en) * 2000-08-04 2004-11-28 Warner Lambert Co 2-(4-pyridyl) amino-6-dialkoxyphenyl-pyrido [2,3-d] pyrimidin-7-ones.
JP2005507392A (ja) * 2000-08-04 2005-03-17 ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー 2−(4−ピリジル)アミノ−6−ジアルキルオキシフェニルピリド〔2,3−d〕ピリミジン−7−オン類の製造方法
DE60303009T2 (de) * 2002-01-22 2006-07-13 Warner-Lambert Co. Llc 2-(pyridin-2-ylamino)-pyrido[2,3-d]pyrimidin-7-one

Also Published As

Publication number Publication date
WO2002012237A2 (en) 2002-02-14
AR030571A1 (es) 2003-08-27
AU2001278908A1 (en) 2002-02-18
US20030216415A1 (en) 2003-11-20
JP2004505974A (ja) 2004-02-26
CA2417937A1 (en) 2002-02-14
US6960662B2 (en) 2005-11-01
EP1307451A2 (en) 2003-05-07
WO2002012237A3 (en) 2002-05-10
MXPA03000289A (es) 2003-06-06

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7O E 8O ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2021 DE 29/09/2009.