TW200529848A

TW200529848A - 1h-imidazo[4,5-c]quinoline derivatives in the treatment of protein kinase dependent diseases

1h-imidazo[4,5-c]quinoline derivatives in the treatment of protein kinase dependent diseases Download PDF

Info

Publication number: TW200529848A
Authority: TW; Taiwan
Prior art keywords: phenyl; imidazo; group; ylethynyl; methyl
Prior art date: 2003-11-21

Application number

TW093135753A

Other languages

English (en)

Chinese (zh)

Inventor

Hans-Georg Capraro

Pascal Furet

Carlos Garcia-Echeverria

Frederic Stauffer

Original Assignee

Novartis Ag

Priority date

2003-11-21

Filing date

2004-11-19

Publication date

2005-09-16

2004-11-19 Application filed by Novartis Ag filed Critical Novartis Ag

2005-09-16 Publication of TW200529848A publication Critical patent/TW200529848A/zh

Links

208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title claims abstract description 87
201000010099 disease Diseases 0.000 title claims abstract description 84
238000011282 treatment Methods 0.000 title claims abstract description 60
102000001253 Protein Kinase Human genes 0.000 title claims abstract description 43
108060006633 protein kinase Proteins 0.000 title claims abstract description 43
230000001419 dependent effect Effects 0.000 title claims abstract description 39
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238000000034 method Methods 0.000 claims abstract description 49
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IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims description 164
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229910052757 nitrogen Inorganic materials 0.000 claims description 86
239000001257 hydrogen Substances 0.000 claims description 74
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