TR201902673T4 - Medetomidin sentezinde yararlı olan 3-arilbütanlar gibi bileşiklerin hazırlanması için işlemler. - Google Patents

Medetomidin sentezinde yararlı olan 3-arilbütanlar gibi bileşiklerin hazırlanması için işlemler. Download PDF

Info

Publication number
TR201902673T4
TR201902673T4 TR2019/02673T TR201902673T TR201902673T4 TR 201902673 T4 TR201902673 T4 TR 201902673T4 TR 2019/02673 T TR2019/02673 T TR 2019/02673T TR 201902673 T TR201902673 T TR 201902673T TR 201902673 T4 TR201902673 T4 TR 201902673T4
Authority
TR
Turkey
Prior art keywords
preparation
arylbutanes
medetomidine
synthesis
processes
Prior art date
Application number
TR2019/02673T
Other languages
English (en)
Turkish (tr)
Inventor
Eklund Lars
Eek Margus
Ekambaram Ramesh
Maasalu Ants
Original Assignee
I Tech Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by I Tech Ab filed Critical I Tech Ab
Publication of TR201902673T4 publication Critical patent/TR201902673T4/tr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01Sulfonic acids
    • C07C309/02Sulfonic acids having sulfo groups bound to acyclic carbon atoms
    • C07C309/24Sulfonic acids having sulfo groups bound to acyclic carbon atoms of a carbon skeleton containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • C07C45/455Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation with carboxylic acids or their derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/45Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C249/00Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C249/02Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of compounds containing imino groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/62Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by hydrogenation of carbon-to-carbon double or triple bonds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/63Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/78Separation; Purification; Stabilisation; Use of additives
    • C07C45/86Use of additives, e.g. for stabilisation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C47/00Compounds having —CHO groups
    • C07C47/20Unsaturated compounds having —CHO groups bound to acyclic carbon atoms
    • C07C47/228Unsaturated compounds having —CHO groups bound to acyclic carbon atoms containing six-membered aromatic rings, e.g. phenylacetaldehyde
    • C07C47/232Unsaturated compounds having —CHO groups bound to acyclic carbon atoms containing six-membered aromatic rings, e.g. phenylacetaldehyde having unsaturation outside the aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C07D233/58Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/14Esters of phosphoric acids containing P(=O)-halide groups
    • C07F9/1403Esters of phosphoric acids containing P(=O)-halide groups containing the structure Hal-P(=O)-O-unsaturated acyclic group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C47/00Compounds having —CHO groups
    • C07C47/20Unsaturated compounds having —CHO groups bound to acyclic carbon atoms
    • C07C47/228Unsaturated compounds having —CHO groups bound to acyclic carbon atoms containing six-membered aromatic rings, e.g. phenylacetaldehyde
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C47/00Compounds having —CHO groups
    • C07C47/20Unsaturated compounds having —CHO groups bound to acyclic carbon atoms
    • C07C47/24Unsaturated compounds having —CHO groups bound to acyclic carbon atoms containing halogen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
TR2019/02673T 2015-01-30 2016-01-29 Medetomidin sentezinde yararlı olan 3-arilbütanlar gibi bileşiklerin hazırlanması için işlemler. TR201902673T4 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB1501593.6A GB201501593D0 (en) 2015-01-30 2015-01-30 New compounds and processes

Publications (1)

Publication Number Publication Date
TR201902673T4 true TR201902673T4 (tr) 2019-03-21

Family

ID=52705534

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2019/02673T TR201902673T4 (tr) 2015-01-30 2016-01-29 Medetomidin sentezinde yararlı olan 3-arilbütanlar gibi bileşiklerin hazırlanması için işlemler.

Country Status (13)

Country Link
US (1) US10053420B2 (https=)
EP (1) EP3250556B1 (https=)
JP (1) JP6702623B2 (https=)
KR (1) KR102458638B1 (https=)
CN (1) CN107428648B (https=)
DK (1) DK3250556T3 (https=)
ES (1) ES2716748T3 (https=)
GB (1) GB201501593D0 (https=)
HR (1) HRP20190286T1 (https=)
HU (1) HUE042626T2 (https=)
PL (1) PL3250556T3 (https=)
TR (1) TR201902673T4 (https=)
WO (1) WO2016120635A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12050293B2 (en) 2018-12-19 2024-07-30 Pgs Geophysical As Medetomidine compositions having improved anti-fouling characteristics
ES2945827T3 (es) 2020-10-21 2023-07-07 I Tech Ab Compuestos antiincrustantes
KR20240148807A (ko) * 2022-03-22 2024-10-11 옵쉐스트바 스 아그라니첸너이아트볫스트벤너스찌유 "빅-즈다로비예쥐보트니흐" 메데토미딘 및 그 유도체의 제조 방법
WO2026015064A1 (en) 2024-07-09 2026-01-15 I-Tech Ab Antifouling paint composition with improved in-can stability

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2340812C2 (de) 1973-08-11 1982-05-27 Basf Ag, 6700 Ludwigshafen Phenylpropanale sowie ein Verfahren zu deren Herstellung
US4416902A (en) 1982-07-16 1983-11-22 International Flavors & Fragrances Inc. Flavoring with cyclohexenyl-beta-methyl acrolein derivatives
DE19714042A1 (de) 1997-04-05 1998-10-08 Henkel Kgaa Verfahren zur Herstellung aromatischer Aldehyde
WO2007111630A1 (en) * 2005-07-29 2007-10-04 Flexitral, Inc. Compounds which release an odor on a change in ph
CN102458659B (zh) * 2009-06-03 2014-07-09 高砂香料工业株式会社 不对称氢化催化剂
TW201223934A (en) * 2010-11-26 2012-06-16 Lonza Ag 3-(2,3-dimethylphenyl)-2-butenal and its use as perfume
KR101914806B1 (ko) * 2011-01-19 2018-11-02 디에스엠 아이피 어셋츠 비.브이. 탄소-탄소 이중 결합 접촉 수소화에 의한 4-아세톡시-2-메틸부탄알의 제조
WO2012120070A1 (en) * 2011-03-10 2012-09-13 Lonza Ltd Method for preparation of 3-(2,3-dimethylphenyl)-2-butenal
KR101932206B1 (ko) 2011-07-22 2018-12-24 캠브렉스 칼스코가 아베 4-치환 이미다졸의 신규 제조방법
KR101537204B1 (ko) * 2012-05-08 2015-07-22 론자 아게 (론자 엘티디.) 2-(2,3-디메틸페닐)-1-프로파날의 제조 방법
WO2012172120A2 (en) 2012-05-08 2012-12-20 Lonza Ltd 2-(2,3-dimethylphenyl)-1-propanal and its use as perfume
WO2012172119A2 (en) * 2012-05-08 2012-12-20 Lonza Ltd Method for the preparation of medetomidine

Also Published As

Publication number Publication date
CN107428648B (zh) 2021-12-10
WO2016120635A1 (en) 2016-08-04
JP2018505179A (ja) 2018-02-22
KR102458638B1 (ko) 2022-10-24
EP3250556B1 (en) 2018-12-05
EP3250556A1 (en) 2017-12-06
KR20170108080A (ko) 2017-09-26
US10053420B2 (en) 2018-08-21
CN107428648A (zh) 2017-12-01
PL3250556T3 (pl) 2019-05-31
GB201501593D0 (en) 2015-03-18
HUE042626T2 (hu) 2019-07-29
US20180009744A1 (en) 2018-01-11
HRP20190286T1 (hr) 2019-04-05
JP6702623B2 (ja) 2020-06-03
ES2716748T3 (es) 2019-06-14
DK3250556T3 (en) 2019-03-11

Similar Documents

Publication Publication Date Title
BR112016029333A2 (pt) síntese de compostos de carbamoilpiridona policíclico
MX2015002616A (es) Sintesis de bis(fluorosulfonil)imida.
MX2020009401A (es) Ligadores de nucleótidos modificados.
MY184733A (en) Pyrimidine fgfr4 inhibitors
UA113643C2 (xx) N-цикліламіди як нематоциди
CR20160098A (es) Polimorfo de los inhibidores de la syk
WO2015008218A3 (en) Process for the preparation of suvorexant and intermediates useful in the synthesis of suvorexant
BR112017006349A2 (pt) derivados de ácido borônico
EA201591349A1 (ru) Способ получения вортиоксетина
EA201790983A1 (ru) Синтез копанлисиба и его дигидрохлорида
NZ711192A (en) Process for making benzoxazepin compounds
BR112016018851A8 (pt) processo para fornecer um composto de fórmula (iv)
MX2017017022A (es) Metodo para la sintesis de derivados de rapamicina.
AR095727A1 (es) Preparación de intermediarios de pirimidina
AR117002A2 (es) Proceso para la preparación de inhibidores de quinasa c-fms
MX384794B (es) Proceso para la preparacion de 5-fluoro-1h-pirazoles a partir de hexafluoropropeno.
TR201902673T4 (tr) Medetomidin sentezinde yararlı olan 3-arilbütanlar gibi bileşiklerin hazırlanması için işlemler.
CY1121116T1 (el) Νεα μεθοδος για την συνθεση αγομελατινης
EA201490998A1 (ru) Способ получения сложных эфиров (5-фтор-2-метил-3-хинолин-2-илметил-индол-1-ил)-уксусной кислоты
MX386134B (es) Proceso para la preparación de 5-fluoro-1h-pirazoles.
BR112016027455A2 (pt) moduladores ppar
NZ720106A (en) A process for the preparation of regadenoson
EA201491463A1 (ru) Способ получения соединения по новой реакции присоединения михаэля с применением воды или различных кислот в качестве добавки
WO2014173917A8 (en) Synthesis of bace inhibitors
MX2016000487A (es) Piridina-2-carboxamidas como nematicidas.