MX384794B - Proceso para la preparacion de 5-fluoro-1h-pirazoles a partir de hexafluoropropeno. - Google Patents

Proceso para la preparacion de 5-fluoro-1h-pirazoles a partir de hexafluoropropeno.

Info

Publication number
MX384794B
MX384794B MX2016015543A MX2016015543A MX384794B MX 384794 B MX384794 B MX 384794B MX 2016015543 A MX2016015543 A MX 2016015543A MX 2016015543 A MX2016015543 A MX 2016015543A MX 384794 B MX384794 B MX 384794B
Authority
MX
Mexico
Prior art keywords
pyrazoles
fluoro
preparation
hexaflouropropene
compound
Prior art date
Application number
MX2016015543A
Other languages
English (en)
Other versions
MX2016015543A (es
Inventor
Christian Funke
Norbert Lui
Sergii Pazenok
Original Assignee
Elanco Animal Health Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Elanco Animal Health Gmbh filed Critical Elanco Animal Health Gmbh
Publication of MX2016015543A publication Critical patent/MX2016015543A/es
Publication of MX384794B publication Critical patent/MX384794B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C21/00—Acyclic unsaturated compounds containing halogen atoms
    • C07C21/02—Acyclic unsaturated compounds containing halogen atoms containing carbon-to-carbon double bonds
    • C07C21/18—Acyclic unsaturated compounds containing halogen atoms containing carbon-to-carbon double bonds containing fluorine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Un nuevo proceso para la preparación de 5-fluoro 1H-pirazoles de la fórmula general (I) como se describe en este documento y las reacciones adicionales con este compuesto.
MX2016015543A 2014-05-27 2015-05-26 Proceso para la preparacion de 5-fluoro-1h-pirazoles a partir de hexafluoropropeno. MX384794B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP14169990 2014-05-27
PCT/EP2015/061540 WO2015181139A1 (en) 2014-05-27 2015-05-26 Process for the preparation of 5-fluoro-1h-pyrazoles starting from hexafluoropropene

Publications (2)

Publication Number Publication Date
MX2016015543A MX2016015543A (es) 2017-02-27
MX384794B true MX384794B (es) 2025-03-14

Family

ID=50774764

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016015543A MX384794B (es) 2014-05-27 2015-05-26 Proceso para la preparacion de 5-fluoro-1h-pirazoles a partir de hexafluoropropeno.

Country Status (17)

Country Link
US (1) US9957256B2 (es)
EP (1) EP3148984B1 (es)
JP (2) JP2017521372A (es)
KR (1) KR102478643B1 (es)
CN (1) CN106536484A (es)
DK (1) DK3148984T3 (es)
ES (1) ES2745559T3 (es)
HR (1) HRP20191551T1 (es)
HU (1) HUE045704T2 (es)
IL (1) IL248566B (es)
LT (1) LT3148984T (es)
MX (1) MX384794B (es)
PL (1) PL3148984T3 (es)
PT (1) PT3148984T (es)
SI (1) SI3148984T1 (es)
TW (1) TWI694066B (es)
WO (1) WO2015181139A1 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018162312A1 (en) 2017-03-10 2018-09-13 Basf Se Spirocyclic derivatives
WO2018177993A1 (de) 2017-03-31 2018-10-04 Bayer Cropscience Aktiengesellschaft Pyrazole zur bekämpfung von arthropoden
EP3590927A1 (en) 2018-07-05 2020-01-08 Bayer Animal Health GmbH Novel compounds for controlling arthropods
EP3771711A1 (en) 2019-07-29 2021-02-03 Bayer Animal Health GmbH Pyrazole derivatives for controlling arthropods
CR20220112A (es) 2019-08-14 2022-06-21 Vetoquinol Sa Composiciones que comprenden tigolaner para el control de parásitos
EP4157830B1 (en) 2020-05-27 2025-04-30 Vetoquinol SA Method for preparing 2-chloro-n-(1-cyanocyclopropyl)-5-[2'-methyl-5'-(pentafluoroethyl)-4'-(trifluoromethyl)-2'h-1,3'-bipyrazol-4-yl]benzamide
WO2021242581A1 (en) 2020-05-29 2021-12-02 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic heterocyclic compounds

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1228592B (de) 1964-09-09 1966-11-17 Carl Aust Einrichtung zur Erzeugung von Ozon
JPS572696B2 (es) * 1973-05-08 1982-01-18
SU1456419A1 (ru) 1987-06-18 1989-02-07 Институт элементоорганических соединений им.А.Н.Несмеянова Способ получени 1-замещенных 3-пентафторэтил-4-трифторметил-5-фторпиразолов
US5254774A (en) * 1992-12-28 1993-10-19 Minnesota Mining And Manufacturing Company Preparation of hexafluoropropene oligomers
US6774270B1 (en) * 2003-04-01 2004-08-10 3M Innovative Properties Company Method of removing hexafluoropropylene dimers
EP2184273A1 (de) 2008-11-05 2010-05-12 Bayer CropScience AG Halogen-substituierte Verbindungen als Pestizide
CN103221395A (zh) 2010-11-23 2013-07-24 先正达参股股份有限公司 杀虫化合物
CN103261188A (zh) * 2010-12-17 2013-08-21 先正达参股股份有限公司 杀虫化合物
JP2014510049A (ja) * 2011-02-09 2014-04-24 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト 殺虫性化合物
MX350121B (es) * 2011-03-18 2017-08-28 Bayer Ip Gmbh Derivados de n-(3-carbamoilfenil)-1h-pirazol-5-carboxamida y el uso de los mismos para el control de plagas de animales.
CN103483139B (zh) * 2012-06-15 2016-01-27 中化蓝天集团有限公司 一种制备全氟-2-甲基-2-戊烯的方法
WO2014012975A1 (en) * 2012-07-19 2014-01-23 Bayer Cropscience Ag Process for the preparation of 5-fluoro-1h-pyrazoles
CN102992986B (zh) * 2012-09-29 2016-02-03 中国人民武装警察部队学院 全氟乙基异丙基酮的制备方法
CN107473929B (zh) * 2012-10-26 2020-10-30 浙江蓝天环保高科技股份有限公司 一种联产制备全氟-2-甲基-2-戊烯和全氟-4-甲基-2-戊烯的方法

Also Published As

Publication number Publication date
JP2020097612A (ja) 2020-06-25
JP7013501B2 (ja) 2022-01-31
IL248566B (en) 2019-10-31
EP3148984B1 (en) 2019-07-24
CN106536484A (zh) 2017-03-22
PL3148984T3 (pl) 2019-12-31
HRP20191551T1 (hr) 2019-11-29
KR20170008766A (ko) 2017-01-24
US20170190690A1 (en) 2017-07-06
KR102478643B1 (ko) 2022-12-15
US9957256B2 (en) 2018-05-01
ES2745559T3 (es) 2020-03-02
DK3148984T3 (da) 2019-09-23
PT3148984T (pt) 2019-09-30
SI3148984T1 (sl) 2019-12-31
HUE045704T2 (hu) 2020-01-28
LT3148984T (lt) 2019-09-25
TWI694066B (zh) 2020-05-21
JP2017521372A (ja) 2017-08-03
TW201613871A (en) 2016-04-16
MX2016015543A (es) 2017-02-27
IL248566A0 (en) 2016-12-29
WO2015181139A1 (en) 2015-12-03
EP3148984A1 (en) 2017-04-05

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