TR201101807T2 - Rosuvastatin kalsiyumun farmasotik bileşimleri - Google Patents
Rosuvastatin kalsiyumun farmasotik bileşimleriInfo
- Publication number
- TR201101807T2 TR201101807T2 TR2011/01807T TR201101807T TR201101807T2 TR 201101807 T2 TR201101807 T2 TR 201101807T2 TR 2011/01807 T TR2011/01807 T TR 2011/01807T TR 201101807 T TR201101807 T TR 201101807T TR 201101807 T2 TR201101807 T2 TR 201101807T2
- Authority
- TR
- Turkey
- Prior art keywords
- pharmaceutical compositions
- rosuvastatin calcium
- rosuvastatin
- sodium carbonate
- anhydrous sodium
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 229960004796 rosuvastatin calcium Drugs 0.000 title 1
- LALFOYNTGMUKGG-BGRFNVSISA-L rosuvastatin calcium Chemical group [Ca+2].CC(C)C1=NC(N(C)S(C)(=O)=O)=NC(C=2C=CC(F)=CC=2)=C1\C=C\[C@@H](O)C[C@@H](O)CC([O-])=O.CC(C)C1=NC(N(C)S(C)(=O)=O)=NC(C=2C=CC(F)=CC=2)=C1\C=C\[C@@H](O)C[C@@H](O)CC([O-])=O LALFOYNTGMUKGG-BGRFNVSISA-L 0.000 title 1
- CDBYLPFSWZWCQE-UHFFFAOYSA-L Sodium Carbonate Chemical class [Na+].[Na+].[O-]C([O-])=O CDBYLPFSWZWCQE-UHFFFAOYSA-L 0.000 abstract 2
- BPRHUIZQVSMCRT-VEUZHWNKSA-N rosuvastatin Chemical compound CC(C)C1=NC(N(C)S(C)(=O)=O)=NC(C=2C=CC(F)=CC=2)=C1\C=C\[C@@H](O)C[C@@H](O)CC(O)=O BPRHUIZQVSMCRT-VEUZHWNKSA-N 0.000 abstract 2
- 229960000672 rosuvastatin Drugs 0.000 abstract 2
- 159000000007 calcium salts Chemical group 0.000 abstract 1
- 238000004090 dissolution Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Buluş, rosuvastatinin veya farmasötik olarak kabul edilebilir tuzlarının; ağırlıkça %0.5 ile %2 oranında olması gereken susuz sodyum karbonat kullanımının sağlandığı, 0.1 N HCl ortamında dissolüsyon profilleri üzerine etkisi olan, özellikle rosuvastatinin kalsiyum tuzu ile susuz sodyum karbonat tuzunun farmasötik bileşimleri ile ilgilidir.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/IB2008/052595 WO2009156796A1 (en) | 2008-06-27 | 2008-06-27 | Pharmaceutical compositions of rosuvastatin calcium |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR201101807T2 true TR201101807T2 (tr) | 2012-02-21 |
Family
ID=40386506
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2011/01807T TR201101807T2 (tr) | 2008-06-27 | 2008-06-27 | Rosuvastatin kalsiyumun farmasotik bileşimleri |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US20110098315A1 (tr) |
| EP (1) | EP2306982B1 (tr) |
| JP (1) | JP2011525901A (tr) |
| KR (1) | KR101283147B1 (tr) |
| AU (1) | AU2008358622A1 (tr) |
| BR (1) | BRPI0822782A2 (tr) |
| CA (1) | CA2728539A1 (tr) |
| DK (1) | DK2306982T3 (tr) |
| EA (1) | EA201170101A1 (tr) |
| ES (1) | ES2535106T3 (tr) |
| GE (1) | GEP20135735B (tr) |
| IL (1) | IL210102A0 (tr) |
| MA (1) | MA32498B1 (tr) |
| MX (1) | MX2010013834A (tr) |
| PT (1) | PT2306982E (tr) |
| TN (1) | TN2010000585A1 (tr) |
| TR (1) | TR201101807T2 (tr) |
| WO (1) | WO2009156796A1 (tr) |
| ZA (1) | ZA201009057B (tr) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8609138B2 (en) * | 2010-06-30 | 2013-12-17 | Mochida Pharmaceutical Co., Ltd. | ω3 fatty acid compound preparation |
| RO129060B1 (ro) * | 2013-04-25 | 2014-11-28 | Antibiotice S.A. | Compoziţie farmaceutică stabilă cu rosuvastatină calcică amorfă |
| KR102240429B1 (ko) * | 2013-05-06 | 2021-04-15 | 한미약품 주식회사 | 로수바스타틴 또는 이의 약학적으로 허용되는 염이 함유된 필름 코팅층을 포함하는 복합 제형 |
| KR20150079373A (ko) | 2013-12-30 | 2015-07-08 | 한미약품 주식회사 | 에제티미브 및 로수바스타틴을 포함하는 경구용 복합제제 |
| CN107072997A (zh) | 2014-11-11 | 2017-08-18 | 盐野义制药株式会社 | 含有对光不稳定的药物的多层片剂 |
| JP6108635B2 (ja) * | 2015-05-14 | 2017-04-05 | ダイト株式会社 | ロスバスタチン含有口腔内速崩壊錠 |
| HRP20251674T1 (hr) | 2019-07-31 | 2026-02-13 | Intas Pharmaceuticals Ltd. | Farmaceutski pripravak koji sadrži inhibitore hmg coa reduktaze i fenofibrat |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU217629B (hu) * | 1991-12-12 | 2000-03-28 | Novartis Ag. | Eljárás fluvasztatint tartalmazó stabilizált gyógyszerkészítmények előállítására |
| GB0001621D0 (en) * | 2000-01-26 | 2000-03-15 | Astrazeneca Ab | Pharmaceutical compositions |
| AU2003227691B2 (en) * | 2002-05-03 | 2008-05-15 | Hexal Ag | Stable pharmaceutical formulation for a combination of a statin and an ace inhibitor |
| US20040132771A1 (en) * | 2002-12-20 | 2004-07-08 | Pfizer Inc | Compositions of choleseteryl ester transfer protein inhibitors and HMG-CoA reductase inhibitors |
| JP4839221B2 (ja) * | 2003-11-07 | 2011-12-21 | ジェイ ジェイ ファーマ,インコーポレイテッド | Hdlを高める併用療法用複合物 |
| WO2006134604A1 (en) * | 2005-06-15 | 2006-12-21 | Hetero Drugs Limited | Combination composition of cholesterol absorption inhibitor and 3-hydroxy-3-methylglutaryl-coenzyme a (hmg-coa) reductase inhibitor |
| US20070202159A1 (en) * | 2006-02-02 | 2007-08-30 | Mathur Rajeev S | Pharmaceutical composition comprising stabilized statin particles |
| WO2008005543A2 (en) * | 2006-07-06 | 2008-01-10 | Teva Pharmaceutical Industries Ltd. | Compositions with controlled pharmacokinetics |
| WO2008062476A2 (en) * | 2006-10-31 | 2008-05-29 | Glenmark Pharmaceutical Limited | Pharmaceutical composition comprising rosuvastatin or pharmaceutically accepatble salts thereof |
-
2008
- 2008-06-27 AU AU2008358622A patent/AU2008358622A1/en not_active Abandoned
- 2008-06-27 BR BRPI0822782A patent/BRPI0822782A2/pt not_active IP Right Cessation
- 2008-06-27 MX MX2010013834A patent/MX2010013834A/es not_active Application Discontinuation
- 2008-06-27 CA CA2728539A patent/CA2728539A1/en not_active Abandoned
- 2008-06-27 US US12/997,248 patent/US20110098315A1/en not_active Abandoned
- 2008-06-27 GE GEAP200812071A patent/GEP20135735B/en unknown
- 2008-06-27 EA EA201170101A patent/EA201170101A1/ru unknown
- 2008-06-27 WO PCT/IB2008/052595 patent/WO2009156796A1/en not_active Ceased
- 2008-06-27 DK DK08776549T patent/DK2306982T3/en active
- 2008-06-27 EP EP08776549.1A patent/EP2306982B1/en not_active Not-in-force
- 2008-06-27 ES ES08776549.1T patent/ES2535106T3/es active Active
- 2008-06-27 JP JP2011515641A patent/JP2011525901A/ja active Pending
- 2008-06-27 PT PT87765491T patent/PT2306982E/pt unknown
- 2008-06-27 TR TR2011/01807T patent/TR201101807T2/tr unknown
- 2008-06-27 KR KR1020107029131A patent/KR101283147B1/ko not_active Expired - Fee Related
-
2010
- 2010-12-17 TN TNP2010000585A patent/TN2010000585A1/fr unknown
- 2010-12-17 ZA ZA2010/09057A patent/ZA201009057B/en unknown
- 2010-12-19 IL IL210102A patent/IL210102A0/en unknown
-
2011
- 2011-01-21 MA MA33550A patent/MA32498B1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL210102A0 (en) | 2011-02-28 |
| ZA201009057B (en) | 2012-01-25 |
| BRPI0822782A2 (pt) | 2015-09-29 |
| TN2010000585A1 (en) | 2012-05-24 |
| PT2306982E (pt) | 2015-05-18 |
| KR20110027711A (ko) | 2011-03-16 |
| CA2728539A1 (en) | 2009-12-30 |
| WO2009156796A1 (en) | 2009-12-30 |
| JP2011525901A (ja) | 2011-09-29 |
| GEP20135735B (en) | 2013-01-25 |
| EP2306982B1 (en) | 2015-01-07 |
| AU2008358622A1 (en) | 2009-12-30 |
| ES2535106T3 (es) | 2015-05-05 |
| MA32498B1 (fr) | 2011-07-03 |
| KR101283147B1 (ko) | 2013-07-05 |
| DK2306982T3 (en) | 2015-04-20 |
| MX2010013834A (es) | 2011-02-21 |
| EA201170101A1 (ru) | 2011-08-30 |
| US20110098315A1 (en) | 2011-04-28 |
| EP2306982A1 (en) | 2011-04-13 |
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