TR199901128T2 - N-(aril/heteroarilasetil) amino asit esterler, bunu ihtiva eden farmasötik bilesimler ve bu tür bilesikler kullanarak -amiloit peptit salinimini ve/veya bunun sentezlenmesini inhibe etme yöntemleri. - Google Patents

N-(aril/heteroarilasetil) amino asit esterler, bunu ihtiva eden farmasötik bilesimler ve bu tür bilesikler kullanarak -amiloit peptit salinimini ve/veya bunun sentezlenmesini inhibe etme yöntemleri.

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Publication number
TR199901128T2
TR199901128T2 TR1999/01128T TR9901128T TR199901128T2 TR 199901128 T2 TR199901128 T2 TR 199901128T2 TR 1999/01128 T TR1999/01128 T TR 1999/01128T TR 9901128 T TR9901128 T TR 9901128T TR 199901128 T2 TR199901128 T2 TR 199901128T2
Authority
TR
Turkey
Prior art keywords
synthesis
pharmaceutical compositions
compounds
amyloid peptide
inhibit
Prior art date
Application number
TR1999/01128T
Other languages
English (en)
Inventor
Wu Jing
D. Thorsett Eugene
S. Nissen Jeffrey
E. Mabry Thomas
H. Latimer Lee
John Verghese
Y. Fang Lawrence
E. Audia James
Original Assignee
Elan Pharmaceuticals, Inc.
Eli Lilly And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Elan Pharmaceuticals, Inc., Eli Lilly And Company filed Critical Elan Pharmaceuticals, Inc.
Publication of TR199901128T2 publication Critical patent/TR199901128T2/tr

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    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
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Abstract

Ilisikte, -amiloit peptit salinimini ve/veya bunun sentezine inhibe eden ve buna bagli olarak Alzheimer hastaliginin tedavisinde faydali olan bilesikler verilmektedir. Yine ilisikte -amiloit peptit salinimini ve/veya bunun sentezini inhibe eden bir bilesik ihtiva eden bir bilesik ihtiva eden farmasötik bilesimler ve bu tür farmasötik bilesimler kullanarak Alzheimer hastaligini hem profilaktik, hem terapötik tedavisine iliskin yöntemler verilmektedir.
TR1999/01128T 1996-11-22 1997-11-20 N-(aril/heteroarilasetil) amino asit esterler, bunu ihtiva eden farmasötik bilesimler ve bu tür bilesikler kullanarak -amiloit peptit salinimini ve/veya bunun sentezlenmesini inhibe etme yöntemleri. TR199901128T2 (tr)

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NO992463L (no) 1999-07-19
CA2267065A1 (en) 1998-05-28
BR9713404A (pt) 2000-01-25
KR20000069074A (ko) 2000-11-25
JP2001505204A (ja) 2001-04-17
EP0951464B1 (en) 2005-05-11
DE69733272D1 (de) 2005-06-16
ID21956A (id) 1999-08-19
HUP0000492A3 (en) 2000-06-28
AU739035B2 (en) 2001-10-04
DE69733272T2 (de) 2006-01-26
NZ334950A (en) 2001-03-30
NO992463D0 (no) 1999-05-21
CN1237960A (zh) 1999-12-08
EP0951464A1 (en) 1999-10-27
IL129238A0 (en) 2000-02-17
ATE295346T1 (de) 2005-05-15
AU5249898A (en) 1998-06-10
WO1998022430A1 (en) 1998-05-28

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