TNSN96141A1 - Formulations pharmaceutiques et procede pour leur production - Google Patents

Formulations pharmaceutiques et procede pour leur production

Info

Publication number
TNSN96141A1
TNSN96141A1 TNTNSN96141A TNSN96141A TNSN96141A1 TN SN96141 A1 TNSN96141 A1 TN SN96141A1 TN TNSN96141 A TNTNSN96141 A TN TNSN96141A TN SN96141 A TNSN96141 A TN SN96141A TN SN96141 A1 TNSN96141 A1 TN SN96141A1
Authority
TN
Tunisia
Prior art keywords
formulation
production
pharmaceutical formulations
administration
hydroxypropylmethylcellulose
Prior art date
Application number
TNTNSN96141A
Other languages
English (en)
Inventor
James Macrae Ross
Sarah Smith Janet
Original Assignee
Pfizer Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Res & Dev filed Critical Pfizer Res & Dev
Publication of TNSN96141A1 publication Critical patent/TNSN96141A1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

L’INVENTION CONCERNE UNE FORMULATION PHARMACEUTIQUE A LIBERATION CONTROLEE POUR L’ADMINISTRATION ORALE. CETTE FORMULATION CONSISTE EN UN COMPOSE MEDICAMENTEUX ACTIF, UN POLYMERE D’OXYDE D’ETHYLENE DE BAS POIDS MOLECULAIRE, DE L’HYDROXYPROPYLMETHYLCELLULOSE, DES EXCIPIENTS DE COMPRESSION ET, FACULTATIVEMENT, UN OU PLUSIEURS POLYMERES ENTERIQUES. APPLICATION : OBTENTION DE FORMULATION A VITESSE CONSTANTE DE LIBERATION POUR L'ADMINISTRATION DE DIVERS MEDICAMENTS.
TNTNSN96141A 1995-11-21 1996-11-20 Formulations pharmaceutiques et procede pour leur production TNSN96141A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9523752.5A GB9523752D0 (en) 1995-11-21 1995-11-21 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
TNSN96141A1 true TNSN96141A1 (fr) 2005-03-15

Family

ID=10784188

Family Applications (1)

Application Number Title Priority Date Filing Date
TNTNSN96141A TNSN96141A1 (fr) 1995-11-21 1996-11-20 Formulations pharmaceutiques et procede pour leur production

Country Status (29)

Country Link
EP (1) EP0862437A1 (fr)
JP (1) JPH10513481A (fr)
KR (1) KR19990071505A (fr)
CN (1) CN1215993A (fr)
AP (1) AP718A (fr)
AR (1) AR004335A1 (fr)
AU (1) AU709560B2 (fr)
BG (1) BG102438A (fr)
BR (1) BR9611626A (fr)
CA (1) CA2232715A1 (fr)
CO (1) CO4480020A1 (fr)
CZ (1) CZ155498A3 (fr)
GB (1) GB9523752D0 (fr)
HR (1) HRP960554A2 (fr)
HU (1) HUP9903734A3 (fr)
IS (1) IS4706A (fr)
MA (1) MA26410A1 (fr)
MX (1) MX9804008A (fr)
NO (1) NO982302L (fr)
NZ (1) NZ322053A (fr)
OA (1) OA10687A (fr)
PE (1) PE22898A1 (fr)
PL (1) PL326981A1 (fr)
SK (1) SK63098A3 (fr)
TN (1) TNSN96141A1 (fr)
TR (1) TR199800902T2 (fr)
WO (1) WO1997018814A1 (fr)
YU (1) YU62096A (fr)
ZA (1) ZA969722B (fr)

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AU759825B2 (en) * 1997-12-16 2003-05-01 Pfizer Products Inc. Combination effective for the treatment of impotence
AU736951C (en) 1998-03-19 2003-02-20 Bristol-Myers Squibb Company Biphasic controlled release delivery system for high solubility pharmaceuticals and method
GT199900061A (es) * 1998-05-15 2000-10-14 Pfizer Formulaciones farmaceuticas.
EP0987020A1 (fr) * 1998-09-04 2000-03-22 Pharma Pass LLC Composition contenant du metoprolol et procédé de préparation
EP0974343B1 (fr) * 1998-07-22 2004-09-29 Pharma Pass II LLC Procédé de préparation d'une composition solide contentant du metoprolol
CO5140079A1 (es) * 1998-10-14 2002-03-22 Novartis Ag Composicion farmaceutica de liberacion sostenida y metodo para liberar un agente farmaceuticamente activo de liberacion sostenida y metodo para liberar un agente far- maceuticamente activo
UA67802C2 (uk) * 1998-10-23 2004-07-15 Пфайзер Рісьоч Енд Дівелепмент Компані, Н.В./С.А. Фармацевтична композиція з контрольованим вивільненням інгібітора цгмф фде-5 (варіанти), спосіб її одержання та спосіб лікування еректильної дисфункції
US20030059467A1 (en) * 2001-09-14 2003-03-27 Pawan Seth Pharmaceutical composition comprising doxasozin
US7612112B2 (en) 2001-10-25 2009-11-03 Depomed, Inc. Methods of treatment using a gastric retained gabapentin dosage
TWI312285B (en) 2001-10-25 2009-07-21 Depomed Inc Methods of treatment using a gastric retained gabapentin dosage
US6723340B2 (en) 2001-10-25 2004-04-20 Depomed, Inc. Optimal polymer mixtures for gastric retentive tablets
US8329217B2 (en) 2001-11-06 2012-12-11 Osmotica Kereskedelmi Es Szolgaltato Kft Dual controlled release dosage form
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
WO2005037247A2 (fr) * 2003-10-17 2005-04-28 Ranbaxy Laboratories Limited Formulations matricielles de doxazosine a administration orale
US20050255157A1 (en) * 2004-05-11 2005-11-17 Glenmark Pharmaceuticals Limited Sustained release, mucoadhesive vaginal pharmaceutical compositions
KR100574554B1 (ko) * 2004-05-28 2006-04-27 한미약품 주식회사 니아신의 경구투여용 서방성 조성물
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
KR100679111B1 (ko) * 2004-11-20 2007-02-07 대우약품공업주식회사 독사조신을 포함하는 서방성 정제
CA2619035A1 (fr) * 2005-08-22 2007-03-01 Novartis Ag Compositions pharmaceutiques
US20090176882A1 (en) 2008-12-09 2009-07-09 Depomed, Inc. Gastric retentive gabapentin dosage forms and methods for using same
CA2597740C (fr) 2006-04-26 2012-10-16 Supernus Pharmaceuticals, Inc. Preparations a liberation modifiee contenant de l'oxcarbazepine et derives connexes
CA2810839A1 (fr) 2006-05-04 2007-11-15 Boehringer Ingelheim International Gmbh Polymorphes
EP1852108A1 (fr) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG Compositions d'inhibiteurs de la DPP IV
PE20110235A1 (es) 2006-05-04 2011-04-14 Boehringer Ingelheim Int Combinaciones farmaceuticas que comprenden linagliptina y metmorfina
CN100396282C (zh) * 2006-07-25 2008-06-25 山东省医药工业研究所 甲磺酸多沙唑嗪缓释胶囊及制备方法
SA07280459B1 (ar) 2006-08-25 2011-07-20 بيورديو فارما إل. بي. أشكال جرعة صيدلانية للتناول عن طريق الفم مقاومة للعبث تشتمل على مسكن شبه أفيوني
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PE20091730A1 (es) 2008-04-03 2009-12-10 Boehringer Ingelheim Int Formulaciones que comprenden un inhibidor de dpp4
BRPI0916997A2 (pt) 2008-08-06 2020-12-15 Boehringer Ingelheim International Gmbh Inibidor de dpp-4 e seu uso
US20200155558A1 (en) 2018-11-20 2020-05-21 Boehringer Ingelheim International Gmbh Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
KR101004205B1 (ko) 2008-12-17 2010-12-24 동아제약주식회사 유데나필 함유 서방성 제제를 제조하기 위한 제어방출 조성물
EP2395983B1 (fr) 2009-02-13 2020-04-08 Boehringer Ingelheim International GmbH Composition pharmaceutique contenant un inhibiteur sglt2 en combinaison avec un inhibiteur dpp-iv et optioenellement un autre agent antidiabetique
US9901551B2 (en) 2009-04-20 2018-02-27 Ambra Bioscience Llc Chemosensory receptor ligand-based therapies
EP2421524B1 (fr) 2009-04-20 2018-08-08 Elcelyx Therapeutics, Inc. Thérapies à base de ligand de récepteur chimiosensible
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CN107115530A (zh) 2009-11-27 2017-09-01 勃林格殷格翰国际有限公司 基因型糖尿病患者利用dpp‑iv抑制剂例如利拉利汀的治疗
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WO2013174767A1 (fr) 2012-05-24 2013-11-28 Boehringer Ingelheim International Gmbh Dérivé de xanthine en tant qu'inhibiteur de la dpp-4 à utiliser dans la modification de l'apport alimentaire et dans la régulation des préférences alimentaires
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Also Published As

Publication number Publication date
EP0862437A1 (fr) 1998-09-09
NO982302D0 (no) 1998-05-20
BG102438A (en) 1999-01-29
YU62096A (sh) 1999-03-04
AP9600883A0 (en) 1997-01-31
JPH10513481A (ja) 1998-12-22
PL326981A1 (en) 1998-11-09
CN1215993A (zh) 1999-05-05
GB9523752D0 (en) 1996-01-24
OA10687A (en) 2002-11-27
NZ322053A (en) 1999-11-29
IS4706A (is) 1998-03-31
ZA969722B (en) 1998-05-20
AR004335A1 (es) 1998-11-04
NO982302L (no) 1998-07-17
AP718A (en) 1999-01-06
HRP960554A2 (en) 1998-02-28
WO1997018814A1 (fr) 1997-05-29
TR199800902T2 (xx) 1998-09-21
MA26410A1 (fr) 2004-12-20
MX9804008A (es) 1998-09-30
KR19990071505A (ko) 1999-09-27
BR9611626A (pt) 1999-06-01
CA2232715A1 (fr) 1997-05-29
HUP9903734A2 (hu) 2000-03-28
SK63098A3 (en) 1999-05-07
AU709560B2 (en) 1999-09-02
CO4480020A1 (es) 1997-07-09
CZ155498A3 (cs) 1999-03-17
AU7572196A (en) 1997-06-11
HUP9903734A3 (en) 2000-04-28
PE22898A1 (es) 1998-05-07

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