TNSN87101A1 - Compose b - lactamique, son procede de preparation, composition medicinale pour la therapie des maladies infectieuses bacteriennes le contenant, et intermediaires pour la synthese - Google Patents
Compose b - lactamique, son procede de preparation, composition medicinale pour la therapie des maladies infectieuses bacteriennes le contenant, et intermediaires pour la syntheseInfo
- Publication number
- TNSN87101A1 TNSN87101A1 TNTNSN87101A TNSN87101A TNSN87101A1 TN SN87101 A1 TNSN87101 A1 TN SN87101A1 TN TNSN87101 A TNTNSN87101 A TN TNSN87101A TN SN87101 A TNSN87101 A TN SN87101A TN SN87101 A1 TNSN87101 A1 TN SN87101A1
- Authority
- TN
- Tunisia
- Prior art keywords
- compound
- synthesis
- lactamique
- intermediates
- therapy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/36—Methylene radicals, substituted by sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
- C07D501/34—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
CETTE INVENTION CONCERNE UN NOUVEAU COMPOSE B - LACTAMIQUE, PLUS PARTICULIEREMENT UN COMPOSE NOUVEAU DE LA SERIE DES CEPHALOSPORINES UTILE EN TANT QU'ANTIBIOTIQUE, UN PROCEDE POUR LE PREPARER, UN INTERMEDIAIRE DE SYNTHESE ET SON EMPLOI
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP16986086 | 1986-07-21 | ||
JP27318286 | 1986-11-17 |
Publications (1)
Publication Number | Publication Date |
---|---|
TNSN87101A1 true TNSN87101A1 (fr) | 1990-01-01 |
Family
ID=26493073
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TNTNSN87101A TNSN87101A1 (fr) | 1986-07-21 | 1987-08-19 | Compose b - lactamique, son procede de preparation, composition medicinale pour la therapie des maladies infectieuses bacteriennes le contenant, et intermediaires pour la synthese |
Country Status (17)
Country | Link |
---|---|
US (1) | US4966900A (fr) |
EP (1) | EP0254495A3 (fr) |
KR (1) | KR880001677A (fr) |
CN (1) | CN87104995A (fr) |
AU (1) | AU597695B2 (fr) |
DK (1) | DK378187A (fr) |
FI (1) | FI872879A (fr) |
HU (1) | HU198944B (fr) |
IL (1) | IL83194A0 (fr) |
MA (1) | MA21148A1 (fr) |
MC (2) | MC1838A1 (fr) |
NZ (1) | NZ221052A (fr) |
OA (1) | OA08639A (fr) |
PH (1) | PH25108A (fr) |
PT (1) | PT85375B (fr) |
TN (1) | TNSN87101A1 (fr) |
ZW (1) | ZW13387A1 (fr) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MC1921A1 (fr) * | 1987-04-10 | 1989-04-06 | Sankei Yakuhin Kk | Derives acyles |
DK170088A (da) * | 1987-04-10 | 1988-10-11 | Hoffmann La Roche | Acylderivater |
FI883320A (fi) * | 1987-08-07 | 1989-02-08 | Sankei Yakuhin Kk | --laktam, dess framstaellning och mellanprodukter foer dess framstaellning. |
US5073550A (en) * | 1987-08-14 | 1991-12-17 | Hoffmann-La Roche Inc. | Cephalosphorins with sulfur-containing oxyimino side chain |
US5138066A (en) * | 1987-08-14 | 1992-08-11 | Hoffmann-La Roche, Inc. | Intermediates for cephalosporins with sulfur-containing oxyimino side chain |
EP0303172A3 (fr) * | 1987-08-14 | 1991-05-15 | F. Hoffmann-La Roche Ag | Oxyimino-céphalosporines |
US4904775A (en) * | 1988-05-16 | 1990-02-27 | E. R. Squibb & Sons, Inc. | Heteroaroylhydrazide derivatives of monocyclic beta-lactam antibiotics |
CA2024282A1 (fr) * | 1989-09-21 | 1991-03-22 | Peter H. Ermann | Derives hydrazide heterocycliques de beta-lactam monocyclique antibiotique |
US5077432A (en) * | 1990-01-22 | 1991-12-31 | E. R. Squibb & Sons, Inc. | Monobactam hydrazides containing catechol sulfonic acid groups |
US5030724A (en) * | 1990-01-22 | 1991-07-09 | E. R. Squibb & Sons, Inc. | Monobactam hydrazides containing catechol sulfonic acid groups |
ZA918014B (en) * | 1990-11-05 | 1992-07-29 | Squibb & Sons Inc | Heteroaroyl derivatives of monocyclic beta-lactam antibiotics |
IL99898A (en) * | 1990-11-09 | 1996-10-31 | Eisai Co Ltd | 7-Noble-3- Compounds Transformed Carbamoylloxy |
US5250691A (en) * | 1991-09-09 | 1993-10-05 | E. R. Squibb & Sons, Inc. | Heteroaryl derivatives of monocyclic beta-lactam antibiotics |
CN102659713B (zh) * | 2012-05-07 | 2014-03-05 | 山东金城柯瑞化学有限公司 | 头孢地尼侧链酸活性酯的制备方法 |
CN109721618A (zh) * | 2017-10-30 | 2019-05-07 | 刘力 | 头孢匹胺新化合物及其组合物和用途 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GR63088B (en) * | 1976-04-14 | 1979-08-09 | Takeda Chemical Industries Ltd | Preparation process of novel cephalosporins |
US4091671A (en) * | 1977-01-05 | 1978-05-30 | Mclees Donald J | Electronic fluid level sensor |
JPS5874680A (ja) * | 1981-10-01 | 1983-05-06 | Kyowa Hakko Kogyo Co Ltd | β−ラクタム化合物 |
DE150507T1 (de) * | 1983-12-29 | 1987-02-26 | Mochida Pharmaceutical Co., Ltd., Tokio/Tokyo, Jp | Cephalosporinverbindungen, verfahren zu ihrer herstellung und pharmazeutishe praeparate. |
US4610824A (en) * | 1984-10-09 | 1986-09-09 | E. R. Squibb & Sons, Inc. | Hydrazide derivatives of monocyclic beta-lactam antibiotics |
AU586215B2 (en) * | 1985-01-21 | 1989-07-06 | Nippon Pharmaceutical Development Institute Company Limited | Novel ```-lactam antibiotics |
US4826834A (en) * | 1985-09-27 | 1989-05-02 | Takeda Chemical Industries, Ltd. | Cephem compounds |
JPS63132893A (ja) * | 1986-11-25 | 1988-06-04 | Mochida Pharmaceut Co Ltd | 新規セフアロスポリン誘導体、その製法およびそれらを有効成分とする抗菌剤 |
DK170088A (da) * | 1987-04-10 | 1988-10-11 | Hoffmann La Roche | Acylderivater |
MC1921A1 (fr) * | 1987-04-10 | 1989-04-06 | Sankei Yakuhin Kk | Derives acyles |
-
1987
- 1987-06-30 FI FI872879A patent/FI872879A/fi not_active Application Discontinuation
- 1987-07-13 NZ NZ221052A patent/NZ221052A/xx unknown
- 1987-07-15 IL IL83194A patent/IL83194A0/xx unknown
- 1987-07-17 EP EP87306330A patent/EP0254495A3/fr not_active Withdrawn
- 1987-07-17 ZW ZW133/87A patent/ZW13387A1/xx unknown
- 1987-07-17 HU HU873267A patent/HU198944B/hu unknown
- 1987-07-17 MC MC881900A patent/MC1838A1/fr unknown
- 1987-07-20 KR KR1019870007818A patent/KR880001677A/ko not_active Application Discontinuation
- 1987-07-20 PH PH35560A patent/PH25108A/en unknown
- 1987-07-20 DK DK378187A patent/DK378187A/da not_active Application Discontinuation
- 1987-07-20 OA OA59168A patent/OA08639A/xx unknown
- 1987-07-20 US US07/075,412 patent/US4966900A/en not_active Expired - Fee Related
- 1987-07-20 AU AU75917/87A patent/AU597695B2/en not_active Ceased
- 1987-07-20 MA MA21280A patent/MA21148A1/fr unknown
- 1987-07-21 CN CN198787104995A patent/CN87104995A/zh active Pending
- 1987-07-21 PT PT85375A patent/PT85375B/pt not_active IP Right Cessation
- 1987-08-19 TN TNTNSN87101A patent/TNSN87101A1/fr unknown
-
1988
- 1988-06-09 MC MC88210K patent/MC210A7/fr unknown
Also Published As
Publication number | Publication date |
---|---|
KR880001677A (ko) | 1988-04-26 |
IL83194A0 (en) | 1987-12-31 |
ZW13387A1 (en) | 1988-05-18 |
NZ221052A (en) | 1989-09-27 |
HUT45540A (en) | 1988-07-28 |
HU198944B (en) | 1989-12-28 |
EP0254495A3 (fr) | 1989-11-29 |
US4966900A (en) | 1990-10-30 |
FI872879A (fi) | 1988-01-22 |
MC1838A1 (fr) | 1988-06-03 |
EP0254495A2 (fr) | 1988-01-27 |
PT85375B (pt) | 1990-04-30 |
OA08639A (en) | 1988-11-30 |
CN87104995A (zh) | 1988-03-09 |
PH25108A (en) | 1991-02-19 |
FI872879A0 (fi) | 1987-06-30 |
DK378187D0 (da) | 1987-07-20 |
MA21148A1 (fr) | 1988-10-01 |
PT85375A (en) | 1987-08-01 |
DK378187A (da) | 1988-01-22 |
AU7591787A (en) | 1988-01-28 |
AU597695B2 (en) | 1990-06-07 |
MC210A7 (fr) | 1989-06-30 |
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