FI872879A0 - --laktamfoerening, foerfarande foer dess framstaellning, denna innehaollande laekemedelskomposition foer behandling av sjukdom med bakterieinfektion samt mellanprodukter foer dess syntes. - Google Patents

--laktamfoerening, foerfarande foer dess framstaellning, denna innehaollande laekemedelskomposition foer behandling av sjukdom med bakterieinfektion samt mellanprodukter foer dess syntes.

Info

Publication number
FI872879A0
FI872879A0 FI872879A FI872879A FI872879A0 FI 872879 A0 FI872879 A0 FI 872879A0 FI 872879 A FI872879 A FI 872879A FI 872879 A FI872879 A FI 872879A FI 872879 A0 FI872879 A0 FI 872879A0
Authority
FI
Finland
Prior art keywords
foer
dess
sjukdom
laktamfoerening
laekemedelskomposition
Prior art date
Application number
FI872879A
Other languages
English (en)
Other versions
FI872879A (fi
Inventor
Shigeo Shimizu
Hiroyuki Takano
Original Assignee
Sankei Yakuhin Kk
Nippon Pharma Dev Inst
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankei Yakuhin Kk, Nippon Pharma Dev Inst filed Critical Sankei Yakuhin Kk
Publication of FI872879A0 publication Critical patent/FI872879A0/fi
Publication of FI872879A publication Critical patent/FI872879A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • C07D501/34Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI872879A 1986-07-21 1987-06-30 --laktamfoerening, foerfarande foer dess framstaellning, denna innehaollande laekemedelskomposition foer behandling av sjukdom med bakterieinfektion samt mellanprodukter foer dess syntes. FI872879A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP16986086 1986-07-21
JP27318286 1986-11-17

Publications (2)

Publication Number Publication Date
FI872879A0 true FI872879A0 (fi) 1987-06-30
FI872879A FI872879A (fi) 1988-01-22

Family

ID=26493073

Family Applications (1)

Application Number Title Priority Date Filing Date
FI872879A FI872879A (fi) 1986-07-21 1987-06-30 --laktamfoerening, foerfarande foer dess framstaellning, denna innehaollande laekemedelskomposition foer behandling av sjukdom med bakterieinfektion samt mellanprodukter foer dess syntes.

Country Status (17)

Country Link
US (1) US4966900A (fi)
EP (1) EP0254495A3 (fi)
KR (1) KR880001677A (fi)
CN (1) CN87104995A (fi)
AU (1) AU597695B2 (fi)
DK (1) DK378187A (fi)
FI (1) FI872879A (fi)
HU (1) HU198944B (fi)
IL (1) IL83194A0 (fi)
MA (1) MA21148A1 (fi)
MC (2) MC1838A1 (fi)
NZ (1) NZ221052A (fi)
OA (1) OA08639A (fi)
PH (1) PH25108A (fi)
PT (1) PT85375B (fi)
TN (1) TNSN87101A1 (fi)
ZW (1) ZW13387A1 (fi)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MC1921A1 (fr) * 1987-04-10 1989-04-06 Sankei Yakuhin Kk Derives acyles
DK170088A (da) * 1987-04-10 1988-10-11 Hoffmann La Roche Acylderivater
FI883320A (fi) * 1987-08-07 1989-02-08 Sankei Yakuhin Kk --laktam, dess framstaellning och mellanprodukter foer dess framstaellning.
US5073550A (en) * 1987-08-14 1991-12-17 Hoffmann-La Roche Inc. Cephalosphorins with sulfur-containing oxyimino side chain
US5138066A (en) * 1987-08-14 1992-08-11 Hoffmann-La Roche, Inc. Intermediates for cephalosporins with sulfur-containing oxyimino side chain
EP0303172A3 (de) * 1987-08-14 1991-05-15 F. Hoffmann-La Roche Ag Oxyimino-Cephalosporine
US4904775A (en) * 1988-05-16 1990-02-27 E. R. Squibb & Sons, Inc. Heteroaroylhydrazide derivatives of monocyclic beta-lactam antibiotics
CA2024282A1 (en) * 1989-09-21 1991-03-22 Peter H. Ermann Heterocyclic hydrazide derivatives of monocyclic beta-lactam antibiotics
US5077432A (en) * 1990-01-22 1991-12-31 E. R. Squibb & Sons, Inc. Monobactam hydrazides containing catechol sulfonic acid groups
US5030724A (en) * 1990-01-22 1991-07-09 E. R. Squibb & Sons, Inc. Monobactam hydrazides containing catechol sulfonic acid groups
ZA918014B (en) * 1990-11-05 1992-07-29 Squibb & Sons Inc Heteroaroyl derivatives of monocyclic beta-lactam antibiotics
IL99898A (en) * 1990-11-09 1996-10-31 Eisai Co Ltd 7-Noble-3- Compounds Transformed Carbamoylloxy
US5250691A (en) * 1991-09-09 1993-10-05 E. R. Squibb & Sons, Inc. Heteroaryl derivatives of monocyclic beta-lactam antibiotics
CN102659713B (zh) * 2012-05-07 2014-03-05 山东金城柯瑞化学有限公司 头孢地尼侧链酸活性酯的制备方法
CN109721618A (zh) * 2017-10-30 2019-05-07 刘力 头孢匹胺新化合物及其组合物和用途

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR63088B (en) * 1976-04-14 1979-08-09 Takeda Chemical Industries Ltd Preparation process of novel cephalosporins
US4091671A (en) * 1977-01-05 1978-05-30 Mclees Donald J Electronic fluid level sensor
JPS5874680A (ja) * 1981-10-01 1983-05-06 Kyowa Hakko Kogyo Co Ltd β−ラクタム化合物
DE150507T1 (de) * 1983-12-29 1987-02-26 Mochida Pharmaceutical Co., Ltd., Tokio/Tokyo, Jp Cephalosporinverbindungen, verfahren zu ihrer herstellung und pharmazeutishe praeparate.
US4610824A (en) * 1984-10-09 1986-09-09 E. R. Squibb & Sons, Inc. Hydrazide derivatives of monocyclic beta-lactam antibiotics
AU586215B2 (en) * 1985-01-21 1989-07-06 Nippon Pharmaceutical Development Institute Company Limited Novel ```-lactam antibiotics
US4826834A (en) * 1985-09-27 1989-05-02 Takeda Chemical Industries, Ltd. Cephem compounds
JPS63132893A (ja) * 1986-11-25 1988-06-04 Mochida Pharmaceut Co Ltd 新規セフアロスポリン誘導体、その製法およびそれらを有効成分とする抗菌剤
DK170088A (da) * 1987-04-10 1988-10-11 Hoffmann La Roche Acylderivater
MC1921A1 (fr) * 1987-04-10 1989-04-06 Sankei Yakuhin Kk Derives acyles

Also Published As

Publication number Publication date
KR880001677A (ko) 1988-04-26
IL83194A0 (en) 1987-12-31
ZW13387A1 (en) 1988-05-18
NZ221052A (en) 1989-09-27
HUT45540A (en) 1988-07-28
HU198944B (en) 1989-12-28
EP0254495A3 (en) 1989-11-29
US4966900A (en) 1990-10-30
FI872879A (fi) 1988-01-22
MC1838A1 (fr) 1988-06-03
EP0254495A2 (en) 1988-01-27
PT85375B (pt) 1990-04-30
OA08639A (en) 1988-11-30
CN87104995A (zh) 1988-03-09
PH25108A (en) 1991-02-19
TNSN87101A1 (fr) 1990-01-01
DK378187D0 (da) 1987-07-20
MA21148A1 (fr) 1988-10-01
PT85375A (en) 1987-08-01
DK378187A (da) 1988-01-22
AU7591787A (en) 1988-01-28
AU597695B2 (en) 1990-06-07
MC210A7 (fr) 1989-06-30

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Legal Events

Date Code Title Description
FD Application lapsed

Owner name: SANKEI PHARMACEUTICAL COMPANY LIMITED

Owner name: NIPPON PHARMACEUTICAL DEVELOPMENT