SV2003001098A - Formulacion farmaceutica de sabor enmascarado y procedimiento para su preparacion - Google Patents

Formulacion farmaceutica de sabor enmascarado y procedimiento para su preparacion

Info

Publication number
SV2003001098A
SV2003001098A SV2002001098A SV2002001098A SV2003001098A SV 2003001098 A SV2003001098 A SV 2003001098A SV 2002001098 A SV2002001098 A SV 2002001098A SV 2002001098 A SV2002001098 A SV 2002001098A SV 2003001098 A SV2003001098 A SV 2003001098A
Authority
SV
El Salvador
Prior art keywords
procedure
preparation
pharmaceutical formulation
flavor
masked flavor
Prior art date
Application number
SV2002001098A
Other languages
English (en)
Inventor
Philippe Becourt
Josiane Chauvin
Detlev Schwabe
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of SV2003001098A publication Critical patent/SV2003001098A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1635Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

LA INVENCION SE REFIERE A UNA FORMULACION FARMACEUTICA EN FORMA DE POLVO, DESTINADA A SER ADMINISTRADA EN SUSPENSION ACUOSA POR VIA ORAL, QUE TIENE EL SABOR ENMASCRADO, QUE ICNLUYE POR LO MENOS UN POLIMERO CELULOSICO, UN POLIMERO METACRILICO Y UN PRINCIPIO ACTIVO DISTRIBUIDO DE MANERA HOMOGENEA Y EN ESTADO MOLECULAR EN UNA MATRIZ ATOMIZADA, ASI COMO UN AGENTE ALCALINO Y UN AGENTE ABSORBENTE, EL PROCEDIMIENTO PRA SU PREPARACION, ASI COMO A UN METODO DE ENMASCARAMIENTO DEL SABOR DE PRODUCTOS FARMACEUTICOS.
SV2002001098A 2001-06-21 2002-06-19 Formulacion farmaceutica de sabor enmascarado y procedimiento para su preparacion SV2003001098A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0108157A FR2826274B1 (fr) 2001-06-21 2001-06-21 Formulation pharmaceutique au gout masque et son procede de preparation

Publications (1)

Publication Number Publication Date
SV2003001098A true SV2003001098A (es) 2003-03-18

Family

ID=8864587

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2002001098A SV2003001098A (es) 2001-06-21 2002-06-19 Formulacion farmaceutica de sabor enmascarado y procedimiento para su preparacion

Country Status (42)

Country Link
US (2) US7138138B2 (es)
EP (1) EP1401397B1 (es)
JP (1) JP4880871B2 (es)
CN (1) CN1239149C (es)
AP (1) AP1595A (es)
AR (1) AR036096A1 (es)
AT (1) ATE290366T1 (es)
AU (1) AU2002329311B2 (es)
BG (1) BG66314B1 (es)
BR (1) BRPI0208998A2 (es)
CA (1) CA2452239C (es)
CO (1) CO5540278A2 (es)
CZ (1) CZ299947B6 (es)
DE (1) DE60203178T2 (es)
EA (1) EA006016B1 (es)
EC (1) ECSP034915A (es)
ES (1) ES2236574T3 (es)
FR (1) FR2826274B1 (es)
GT (2) GT200200115A (es)
HK (1) HK1067558A1 (es)
HR (1) HRP20031067B1 (es)
HU (1) HUP0400799A3 (es)
IL (2) IL159404A0 (es)
JO (1) JO2325B1 (es)
MA (1) MA27042A1 (es)
MX (1) MXPA03011756A (es)
MY (1) MY134340A (es)
NO (1) NO332258B1 (es)
NZ (1) NZ530042A (es)
OA (1) OA12635A (es)
PA (1) PA8548301A1 (es)
PE (1) PE20030201A1 (es)
PL (1) PL202090B1 (es)
PT (1) PT1401397E (es)
SK (1) SK285865B6 (es)
SV (1) SV2003001098A (es)
TN (1) TNSN03141A1 (es)
TW (1) TWI228049B (es)
UA (1) UA77960C2 (es)
UY (1) UY27341A1 (es)
WO (1) WO2003000225A2 (es)
ZA (1) ZA200309479B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7384921B2 (en) * 2004-02-20 2008-06-10 Enanta Pharmaceuticals, Inc. Polymorphic forms of 6-11 bicyclic ketolide derivatives
GB2419094A (en) 2004-10-12 2006-04-19 Sandoz Ag Pharmaceutical composition of unpleasnt tasing active substances
FR2882522B1 (fr) * 2005-02-25 2007-04-13 Aventis Pharma Sa Composition pharmaceutique solide comprenant de la telithromycine
US7384922B2 (en) * 2005-05-04 2008-06-10 Enanta Pharmaceuticals, Inc. 6-11 bridged oxime erythromycin derivatives
US20060264386A1 (en) * 2005-05-17 2006-11-23 Rongqi Sun Pharmaceutical formulations of 6-11 bicyclic ketolide derivatives and related macrolides and methods for preparation thereof
KR101387249B1 (ko) * 2006-02-03 2014-05-21 에보니크 룀 게엠베하 물에 난용성인 유효 성분과 중합체의 혼합물을 함유하는제약 조성물
US20100226979A1 (en) * 2006-03-21 2010-09-09 Jubilant Organosys Limited Taste Masked Phamaceutical Composition for Oral Solid Dosage form and Process for Preparing the Same Using Magnesium Aluminium Silicate
US20080181932A1 (en) * 2007-01-30 2008-07-31 Drugtech Corporation Compositions for oral delivery of pharmaceuticals
KR100935893B1 (ko) * 2007-09-11 2010-01-07 국방과학연구소 1,1'-다이메틸-5,5’-바이테트라졸의 합성방법
WO2009055557A1 (en) 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
WO2010069330A2 (en) 2008-12-16 2010-06-24 Carlsberg A/S Coating of hydroxylated surfaces by gas phase grafting
CA2868262A1 (en) 2012-03-27 2013-10-03 Cempra Pharmaceuticals, Inc. Parenteral formulations for administering macrolide antibiotics
DE102012014848A1 (de) * 2012-07-27 2012-10-31 Heilerde-Gesellschaft Luvos Just GmbH & Co. KG Heilerde-Zubereitung
KR20170039689A (ko) * 2014-08-05 2017-04-11 셈프라 파마슈티컬스, 인크. 항균제의 분말 경구 현탁제 제형
CN114209661B (zh) * 2022-02-21 2022-04-29 北京罗诺强施医药技术研发中心有限公司 呈细粒形式的固体药物组合物

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2930409A1 (de) * 1979-07-26 1981-02-12 Bayer Ag Spruehtrocknung von mikrokapseldispersionen
JPS63150220A (ja) * 1986-12-15 1988-06-22 Dainippon Pharmaceut Co Ltd 経口用固形製剤の製造方法
US4808411A (en) * 1987-06-05 1989-02-28 Abbott Laboratories Antibiotic-polymer compositions
US5084278A (en) * 1989-06-02 1992-01-28 Nortec Development Associates, Inc. Taste-masked pharmaceutical compositions
ZA945944B (en) * 1993-08-13 1996-02-08 Eurand America Inc Procedure for encapsulating nsaids
AUPN969796A0 (en) * 1996-05-07 1996-05-30 F.H. Faulding & Co. Limited Taste masked liquid suspensions
EP1027036A2 (en) * 1997-10-03 2000-08-16 ELAN CORPORATION, Plc Taste masked formulations
IN191239B (es) * 1999-06-11 2003-10-11 Ranbaxy Lab Ltd
US6555569B2 (en) * 2000-03-07 2003-04-29 Pfizer Inc. Use of heteroaryl substituted N-(indole-2-carbonyl-) amides for treatment of infection
KR100502031B1 (ko) * 2000-08-22 2005-07-25 바실리어 파마슈티카 아게 항균 활성을 갖는 신규한 매크롤라이드

Also Published As

Publication number Publication date
CA2452239C (fr) 2011-07-19
UY27341A1 (es) 2003-01-31
AU2002329311B2 (en) 2007-02-01
HRP20031067A2 (en) 2004-04-30
HUP0400799A2 (hu) 2004-08-30
FR2826274B1 (fr) 2003-09-26
OA12635A (fr) 2006-06-15
US20070014857A1 (en) 2007-01-18
US20040142029A1 (en) 2004-07-22
IL159404A0 (en) 2004-06-01
BRPI0208998A2 (pt) 2017-06-06
PL202090B1 (pl) 2009-06-30
ZA200309479B (en) 2005-04-26
CZ20033441A3 (en) 2004-03-17
PL366803A1 (en) 2005-02-07
EA200400061A1 (ru) 2004-06-24
CN1529585A (zh) 2004-09-15
JO2325B1 (en) 2006-06-28
JP4880871B2 (ja) 2012-02-22
ATE290366T1 (de) 2005-03-15
IL159404A (en) 2007-08-19
JP2004534810A (ja) 2004-11-18
UA77960C2 (en) 2007-02-15
NO332258B1 (no) 2012-08-13
DE60203178D1 (de) 2005-04-14
BG66314B1 (bg) 2013-04-30
AR036096A1 (es) 2004-08-11
EA006016B1 (ru) 2005-08-25
MXPA03011756A (es) 2004-07-01
HUP0400799A3 (en) 2012-08-28
MY134340A (en) 2007-12-31
WO2003000225A3 (fr) 2003-03-13
EP1401397B1 (fr) 2005-03-09
AP2003002927A0 (en) 2003-12-31
HRP20031067B1 (en) 2011-10-31
SK285865B6 (sk) 2007-10-04
EP1401397A2 (fr) 2004-03-31
ECSP034915A (es) 2004-02-26
SK15922003A3 (sk) 2004-05-04
TWI228049B (en) 2005-02-21
CZ299947B6 (cs) 2009-01-07
CO5540278A2 (es) 2005-07-29
PA8548301A1 (es) 2003-09-05
NO20035581D0 (no) 2003-12-15
DE60203178T2 (de) 2006-01-26
AP1595A (en) 2006-04-12
BG108458A (bg) 2005-02-28
US7138138B2 (en) 2006-11-21
MA27042A1 (fr) 2004-12-20
PE20030201A1 (es) 2003-03-12
WO2003000225A2 (fr) 2003-01-03
NZ530042A (en) 2005-09-30
FR2826274A1 (fr) 2002-12-27
TNSN03141A1 (fr) 2005-12-23
CA2452239A1 (fr) 2003-01-03
GT200200115AA (es) 2005-01-12
CN1239149C (zh) 2006-02-01
GT200200115A (es) 2003-02-27
ES2236574T3 (es) 2005-07-16
HK1067558A1 (en) 2005-04-15
PT1401397E (pt) 2005-05-31

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