AR034900A1 - Uso de una cantidad eficaz de un inhibidor de pde4 y un agente anticolinergico, bien en forma combinada sola o por separado, composiciones farmaceuticas que los comprenden, metodo para prepararlas, y uso de una composicion que comprende una cantidad eficaz de un inhibidor de pde4, una cantidad efica - Google Patents
Uso de una cantidad eficaz de un inhibidor de pde4 y un agente anticolinergico, bien en forma combinada sola o por separado, composiciones farmaceuticas que los comprenden, metodo para prepararlas, y uso de una composicion que comprende una cantidad eficaz de un inhibidor de pde4, una cantidad eficaInfo
- Publication number
- AR034900A1 AR034900A1 ARP020102810A ARP020102810A AR034900A1 AR 034900 A1 AR034900 A1 AR 034900A1 AR P020102810 A ARP020102810 A AR P020102810A AR P020102810 A ARP020102810 A AR P020102810A AR 034900 A1 AR034900 A1 AR 034900A1
- Authority
- AR
- Argentina
- Prior art keywords
- effective amount
- pde4 inhibitor
- composition
- separately
- agent
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Uso de una cantidad eficaz de un inhibidor de PDE4 y un agente anticolinérgico, bien en forma combinada sola o por separado, para la fabricación de composiciones farmacéuticas para la profilaxis, tratamiento o reducción de los empeoramientos asociados con una enfermedad pulmonar. Una composición para la profilaxis, tratamiento o reducción de los empeoramientos asociados a una enfermedad pulmonar, que comprende una cantidad eficaz de un inhibidor de PDE4, una cantidad eficaz de un agente anticolinérgico y un excipiente farmacéuticamente aceptable. Un método para preparar dichas composiciones que comprende mezclar una cantidad eficaz de un inhibidor de PDE4 y un agente anticolinérgico con un excipiente farmacéuticamente aceptable. Uso de una composición que comprende una cantidad eficaz de un inhibidor de PDE4, una cantidad eficaz de un agente anticolinérgico y un excipiente farmacéuticamente aceptable para la fabricación de un medicamento para la profilaxis, tratamiento o reducción de los empeoramientos asociados con una enfermedad pulmonar.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0118373.0A GB0118373D0 (en) | 2001-07-27 | 2001-07-27 | Novel therapeutic method |
Publications (1)
Publication Number | Publication Date |
---|---|
AR034900A1 true AR034900A1 (es) | 2004-03-24 |
Family
ID=9919332
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP020102810A AR034900A1 (es) | 2001-07-27 | 2002-07-25 | Uso de una cantidad eficaz de un inhibidor de pde4 y un agente anticolinergico, bien en forma combinada sola o por separado, composiciones farmaceuticas que los comprenden, metodo para prepararlas, y uso de una composicion que comprende una cantidad eficaz de un inhibidor de pde4, una cantidad efica |
Country Status (18)
Country | Link |
---|---|
US (1) | US20040180918A1 (es) |
EP (1) | EP1411914A2 (es) |
JP (1) | JP2004538302A (es) |
KR (1) | KR20040029384A (es) |
CN (1) | CN1551763A (es) |
AR (1) | AR034900A1 (es) |
BR (1) | BR0211450A (es) |
CA (1) | CA2455520A1 (es) |
CO (1) | CO5550426A2 (es) |
GB (1) | GB0118373D0 (es) |
HU (1) | HUP0401614A2 (es) |
IL (1) | IL160017A0 (es) |
MX (1) | MXPA04000793A (es) |
NO (1) | NO20040353L (es) |
PL (1) | PL368585A1 (es) |
RU (1) | RU2004105865A (es) |
WO (1) | WO2003011274A2 (es) |
ZA (1) | ZA200400410B (es) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2165768B1 (es) | 1999-07-14 | 2003-04-01 | Almirall Prodesfarma Sa | Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen. |
US7776315B2 (en) | 2000-10-31 | 2010-08-17 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Pharmaceutical compositions based on anticholinergics and additional active ingredients |
DE10230769A1 (de) * | 2002-07-09 | 2004-01-22 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Arzneimittelkompositionen auf der Basis neuer Anticholinergika und PDE-IV-Inhibitoren |
US20060189642A1 (en) * | 2003-03-28 | 2006-08-24 | Altana Pharma Ag | Synergistic combination comprising roflumilast and an anticholinergic agent selected from ipratropium, oxitropium and tiotropium salts for the treatment of respiratory diseases |
DK1610787T3 (da) * | 2003-03-28 | 2008-06-02 | Nycomed Gmbh | Synergistisk kombination der omfatter roflumilast og et antikolinergt middel der er valgt blandt tiotropiumsalte til behandling af respiratoriske sygdomme |
TWI328009B (en) | 2003-05-21 | 2010-08-01 | Glaxo Group Ltd | Quinoline derivatives as phosphodiesterase inhibitors |
US20050026883A1 (en) * | 2003-07-31 | 2005-02-03 | Robinson Cynthia B. | Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a PDE-4 inhibitor for treatment of asthma or chronic obstructive pulmonary disease |
EP1504756A1 (en) * | 2003-08-06 | 2005-02-09 | Kyowa Hakko Kogyo Co., Ltd | Medicament compositions comprising a heterocyclic compound and an anticholinergic |
WO2005074982A2 (en) * | 2004-02-06 | 2005-08-18 | Meda Pharma Gmbh & Co. Kg | Combination of anticholinergics and inhibitors of phosphodiesterase type 4 for the treatment of respiratory diseases |
JP4819699B2 (ja) | 2004-02-06 | 2011-11-24 | メダ ファーマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディト ゲゼルシャフト | 喘息及びcopdの長期間の治療のための抗コリン作用薬及びグルココルチコイドの組合せ剤 |
WO2005074983A2 (en) * | 2004-02-06 | 2005-08-18 | Meda Pharma Gmbh & Co. Kg | Treatment of rhinitis with anticholinergics alone in combination with antihistamines phosphodiesterase 4 inhibitors, or corticosteroids |
WO2005102344A1 (ja) * | 2004-04-27 | 2005-11-03 | Kyowa Hakko Kogyo Co., Ltd. | 医薬組成物 |
EP1616567A1 (en) * | 2004-07-16 | 2006-01-18 | Boehringer Ingelheim Pharma GmbH & Co.KG | Medicaments for inhalation comprising PDE IV inhibitors and glycopyrrolate salts |
NZ560206A (en) | 2005-03-16 | 2009-09-25 | Meda Pharma Gmbh & Co Kg | The combination of anticholinergics and leukotriene receptor antagonists for the treatment of respiratory diseases |
GB0521563D0 (en) | 2005-10-21 | 2005-11-30 | Glaxo Group Ltd | Novel compounds |
AU2006329042B2 (en) | 2005-12-21 | 2012-02-02 | Meda Pharma Gmbh & Co Kg | Combination of anticholinergics, glucocorticoids, beta2-agonists, PDE4 inhibitor and antileukotriene for the treatment of inflammatory diseases |
NZ574533A (en) | 2006-08-01 | 2011-05-27 | Glaxo Group Ltd | Pyrazolo[3,4-b]pyridine compounds, and their use as pde4 inhibitors |
AR066016A1 (es) * | 2007-04-11 | 2009-07-15 | Alcon Res Ltd | Uso de un inhibidor del tnf alfa junto con una antihistamina para tratar la rinitis alergica y la conjuntivitis alergica |
EP2100598A1 (en) | 2008-03-13 | 2009-09-16 | Laboratorios Almirall, S.A. | Inhalation composition containing aclidinium for treatment of asthma and chronic obstructive pulmonary disease |
EP2100599A1 (en) | 2008-03-13 | 2009-09-16 | Laboratorios Almirall, S.A. | Inhalation composition containing aclidinium for treatment of asthma and chronic obstructive pulmonary disease |
WO2010097248A1 (en) | 2009-01-13 | 2010-09-02 | Glaxo Group Limited | Pyrimidinecarboxamide derivatives as inhibitors of syk kinase |
CA2773483A1 (en) * | 2009-10-01 | 2011-04-07 | Alcon Research, Ltd. | Olopatadine compositions and uses thereof |
WO2012025474A1 (en) | 2010-08-24 | 2012-03-01 | Glaxo Group Limited | Indazole compounds |
WO2012025473A1 (en) | 2010-08-24 | 2012-03-01 | Glaxo Group Limited | Cc.chemokine receptor 4 antagonists |
EP2510928A1 (en) | 2011-04-15 | 2012-10-17 | Almirall, S.A. | Aclidinium for use in improving the quality of sleep in respiratory patients |
BR112015019276A2 (pt) | 2013-02-19 | 2017-07-18 | Pfizer | compostos de azabenzimidazol como inibidores de isoenzimas de pde4 para o tratamento de distúrbios do snc e outros distúrbios |
US10131669B2 (en) | 2014-07-24 | 2018-11-20 | Pfizer Inc. | Pyrazolopyrimidine compounds |
PL3177624T3 (pl) | 2014-08-06 | 2019-09-30 | Pfizer Inc. | Związki imidazopirydazynowe |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2000198734A (ja) * | 1998-12-30 | 2000-07-18 | Pfizer Inc | 胃運動性減弱および関連疾患の治療のための運動性増強薬 |
GEP20043302B (en) * | 2000-01-31 | 2004-02-10 | Pfizer Prod Inc | Nicotinamide Benzofused-Heterocyclyl Derivatives Useful as Selective Inhibitors of PDE4 Isozymes |
EP1270577B1 (en) * | 2000-03-23 | 2006-12-06 | Takeda Pharmaceutical Company Limited | Furoisoquinoline derivatives, process for producing the same and use thereof |
US20020052312A1 (en) * | 2000-05-30 | 2002-05-02 | Reiss Theodore F. | Combination therapy of chronic obstructive pulmonary disease using muscarinic receptor antagonists |
AR029984A1 (es) * | 2000-07-27 | 2003-07-23 | Smithkline Beecham Corp | Metodo para reducir las exacerbaciones asociadas copd ambito |
US20020137764A1 (en) * | 2000-10-31 | 2002-09-26 | Karin Drechsel | Inhalable formulation of a solution containing a tiotropium salt |
DE10110772A1 (de) * | 2001-03-07 | 2002-09-12 | Boehringer Ingelheim Pharma | Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren |
BR0116624A (pt) * | 2000-12-28 | 2003-12-23 | Almirall Prodesfarma Ag | Composto, processo para produzir o mesmo, composição farmacêutica, uso do composto ou da composição farmacêutica, e, produto de combinação |
-
2001
- 2001-07-27 GB GBGB0118373.0A patent/GB0118373D0/en not_active Ceased
-
2002
- 2002-07-25 AR ARP020102810A patent/AR034900A1/es unknown
- 2002-07-25 CA CA002455520A patent/CA2455520A1/en not_active Abandoned
- 2002-07-25 KR KR10-2004-7001218A patent/KR20040029384A/ko not_active Application Discontinuation
- 2002-07-25 RU RU2004105865/14A patent/RU2004105865A/ru not_active Application Discontinuation
- 2002-07-25 JP JP2003516505A patent/JP2004538302A/ja active Pending
- 2002-07-25 PL PL02368585A patent/PL368585A1/xx not_active Application Discontinuation
- 2002-07-25 BR BR0211450-0A patent/BR0211450A/pt not_active IP Right Cessation
- 2002-07-25 CN CNA028173961A patent/CN1551763A/zh active Pending
- 2002-07-25 IL IL16001702A patent/IL160017A0/xx unknown
- 2002-07-25 EP EP02754939A patent/EP1411914A2/en not_active Withdrawn
- 2002-07-25 WO PCT/EP2002/008322 patent/WO2003011274A2/en not_active Application Discontinuation
- 2002-07-25 HU HU0401614A patent/HUP0401614A2/hu unknown
- 2002-07-25 US US10/484,292 patent/US20040180918A1/en not_active Abandoned
- 2002-07-25 MX MXPA04000793A patent/MXPA04000793A/es not_active Application Discontinuation
-
2004
- 2004-01-20 ZA ZA200400410A patent/ZA200400410B/en unknown
- 2004-01-26 NO NO20040353A patent/NO20040353L/no not_active Application Discontinuation
- 2004-01-27 CO CO04005900A patent/CO5550426A2/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
RU2004105865A (ru) | 2005-02-20 |
CN1551763A (zh) | 2004-12-01 |
WO2003011274A2 (en) | 2003-02-13 |
JP2004538302A (ja) | 2004-12-24 |
KR20040029384A (ko) | 2004-04-06 |
EP1411914A2 (en) | 2004-04-28 |
IL160017A0 (en) | 2004-06-20 |
HUP0401614A2 (hu) | 2004-11-29 |
US20040180918A1 (en) | 2004-09-16 |
BR0211450A (pt) | 2004-07-20 |
CA2455520A1 (en) | 2003-02-13 |
CO5550426A2 (es) | 2005-08-31 |
WO2003011274A3 (en) | 2003-09-18 |
GB0118373D0 (en) | 2001-09-19 |
MXPA04000793A (es) | 2004-05-21 |
NO20040353L (no) | 2004-03-26 |
ZA200400410B (en) | 2004-10-13 |
PL368585A1 (en) | 2005-04-04 |
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Legal Events
Date | Code | Title | Description |
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FB | Suspension of granting procedure |