SU1327789A3 - Способ получени стероидных производных с замещенной 3-аминогруппой или их кислото-аддитивных солей - Google Patents

Способ получени стероидных производных с замещенной 3-аминогруппой или их кислото-аддитивных солей Download PDF

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Publication number
SU1327789A3
SU1327789A3 SU813355225A SU3355225A SU1327789A3 SU 1327789 A3 SU1327789 A3 SU 1327789A3 SU 813355225 A SU813355225 A SU 813355225A SU 3355225 A SU3355225 A SU 3355225A SU 1327789 A3 SU1327789 A3 SU 1327789A3
Authority
SU
USSR - Soviet Union
Prior art keywords
hydrogen
amino
acid
methyl
product
Prior art date
Application number
SU813355225A
Other languages
English (en)
Russian (ru)
Inventor
Дераедт Роже
Торелли Весперто
Бензони Жозетт
Original Assignee
Руссель-Юклаф (Фирма)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Руссель-Юклаф (Фирма) filed Critical Руссель-Юклаф (Фирма)
Application granted granted Critical
Publication of SU1327789A3 publication Critical patent/SU1327789A3/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/007—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 17 (20)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0027—Azides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SU813355225A 1980-11-21 1981-11-20 Способ получени стероидных производных с замещенной 3-аминогруппой или их кислото-аддитивных солей SU1327789A3 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8024750A FR2494698A1 (fr) 1980-11-21 1980-11-21 Nouveaux derives steroides 3-amino substitues, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant

Publications (1)

Publication Number Publication Date
SU1327789A3 true SU1327789A3 (ru) 1987-07-30

Family

ID=9248226

Family Applications (1)

Application Number Title Priority Date Filing Date
SU813355225A SU1327789A3 (ru) 1980-11-21 1981-11-20 Способ получени стероидных производных с замещенной 3-аминогруппой или их кислото-аддитивных солей

Country Status (23)

Country Link
JP (1) JPS57116099A (fi)
KR (1) KR880001239B1 (fi)
AT (1) AT389703B (fi)
AU (1) AU546100B2 (fi)
BE (1) BE891201A (fi)
CA (1) CA1175415A (fi)
CH (1) CH651056A5 (fi)
DE (1) DE3146117A1 (fi)
DK (1) DK161093C (fi)
ES (1) ES8207195A1 (fi)
FI (1) FI77871C (fi)
FR (1) FR2494698A1 (fi)
GB (1) GB2087894B (fi)
HU (1) HU184896B (fi)
IE (1) IE52188B1 (fi)
IL (1) IL64224A0 (fi)
IT (1) IT1172086B (fi)
LU (1) LU83781A1 (fi)
NL (1) NL8105260A (fi)
PT (1) PT74015B (fi)
SE (1) SE451456B (fi)
SU (1) SU1327789A3 (fi)
ZA (1) ZA817806B (fi)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9084800B2 (en) * 2011-11-07 2015-07-21 Natreon, Inc. Indolealkylamino-withasteroid conjugates and method of use

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2430467A (en) * 1944-02-11 1947-11-11 Glidden Co 3-amino-derivatives of steroids and method of making same
US2781342A (en) * 1952-05-17 1957-02-12 Upjohn Co Steroid enamines
DE1189074B (de) * 1959-09-12 1965-03-18 Clin Byla Ets Verfahren zur Herstellung von 3-Aminoverbindungen der Androstan- bzw. Pregnan-Reihe
FR1311761A (fr) * 1959-09-12 1962-12-14 Clin Byla Ets Composés aminés de la série des stéroïdes et procédé de préparation de tels composés
NL103735C (fi) * 1961-02-17
US3503959A (en) * 1962-03-30 1970-03-31 Sterling Drug Inc 3-amino steroids
US3196168A (en) * 1964-02-18 1965-07-20 American Home Prod Aminoaroyl aminosteroids
BE647858A (fi) * 1964-05-13
US3196169A (en) * 1964-11-03 1965-07-20 American Home Prod Aminoacyl aminosteroids
BE672238A (fi) * 1965-11-12 1966-03-01
BE811304R (fr) * 1973-10-24 1974-06-17 Pr0cede de preparation du (20 s) 3 beta -n-dimethylamino
FR2463777A1 (fr) * 1979-08-17 1981-02-27 Roussel Uclaf Nouveaux derives du 5a-pregnan-20-ol, leur procede de preparation et leur application comme medicaments

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
Патент DE № 1965431, кл. С 07 Н 19/16, 1978. Патент US № 3646007, кл. 260-211.5, 1972. Гр инштейн Дж., Виниц М. Хими ами- нокислот и пептидов. Мир, 1965, с. 440-445. : *

Also Published As

Publication number Publication date
DK161093B (da) 1991-05-27
FI813677L (fi) 1982-05-22
IT1172086B (it) 1987-06-18
LU83781A1 (fr) 1982-06-30
AT389703B (de) 1990-01-25
FI77871B (fi) 1989-01-31
FR2494698B1 (fi) 1983-06-24
SE451456B (sv) 1987-10-12
DE3146117A1 (de) 1982-06-16
KR830007716A (ko) 1983-11-04
IE52188B1 (en) 1987-08-05
IT8149746A0 (it) 1981-11-20
CH651056A5 (fr) 1985-08-30
GB2087894B (en) 1984-09-26
DK161093C (da) 1991-11-18
FI77871C (fi) 1989-05-10
SE8105995L (sv) 1982-05-22
PT74015B (fr) 1983-11-30
JPH0247479B2 (fi) 1990-10-19
NL8105260A (nl) 1982-06-16
IL64224A0 (en) 1982-02-28
ATA497081A (de) 1989-06-15
ZA817806B (en) 1982-10-27
GB2087894A (en) 1982-06-03
PT74015A (fr) 1981-12-01
AU546100B2 (en) 1985-08-15
HU184896B (en) 1984-10-29
ES507309A0 (es) 1982-09-01
ES8207195A1 (es) 1982-09-01
CA1175415A (fr) 1984-10-02
FR2494698A1 (fr) 1982-05-28
KR880001239B1 (ko) 1988-07-12
IE812732L (en) 1982-05-21
JPS57116099A (en) 1982-07-19
BE891201A (fr) 1982-05-21
AU7772381A (en) 1982-05-27
DK514981A (da) 1982-05-22

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