SK3502002A3 - Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists - Google Patents
Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists Download PDFInfo
- Publication number
- SK3502002A3 SK3502002A3 SK350-2002A SK3502002A SK3502002A3 SK 3502002 A3 SK3502002 A3 SK 3502002A3 SK 3502002 A SK3502002 A SK 3502002A SK 3502002 A3 SK3502002 A3 SK 3502002A3
- Authority
- SK
- Slovakia
- Prior art keywords
- compound
- thieno
- group
- isoxazol
- phenyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Psychology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US39615699A | 1999-09-14 | 1999-09-14 | |
PCT/US2000/024949 WO2001019832A2 (en) | 1999-09-14 | 2000-09-13 | Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
SK3502002A3 true SK3502002A3 (en) | 2002-09-10 |
Family
ID=23566087
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SK350-2002A SK3502002A3 (en) | 1999-09-14 | 2000-09-13 | Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists |
Country Status (23)
Country | Link |
---|---|
EP (1) | EP1216249B1 (xx) |
JP (1) | JP4717306B2 (xx) |
KR (1) | KR20020027644A (xx) |
AR (1) | AR032135A1 (xx) |
AT (1) | ATE254620T1 (xx) |
AU (1) | AU7577200A (xx) |
BR (1) | BR0014513A (xx) |
CA (1) | CA2383327C (xx) |
CZ (1) | CZ2002896A3 (xx) |
DE (1) | DE60006698T2 (xx) |
DK (1) | DK1216249T3 (xx) |
EA (1) | EA004177B1 (xx) |
EE (1) | EE200200133A (xx) |
ES (1) | ES2206305T3 (xx) |
HU (1) | HUP0202712A3 (xx) |
IL (1) | IL148522A0 (xx) |
MX (1) | MXPA02002690A (xx) |
NO (1) | NO20021249L (xx) |
PL (1) | PL354481A1 (xx) |
PT (1) | PT1216249E (xx) |
SK (1) | SK3502002A3 (xx) |
WO (1) | WO2001019832A2 (xx) |
ZA (1) | ZA200201760B (xx) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0207449D0 (en) * | 2002-03-28 | 2002-05-08 | Glaxo Group Ltd | Novel compounds |
WO2018166855A1 (en) | 2017-03-16 | 2018-09-20 | Basf Se | Heterobicyclic substituted dihydroisoxazoles |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4728651A (en) * | 1985-10-24 | 1988-03-01 | Hoechst-Roussel Pharmaceuticals Inc. | Antihypertensive thieno-isoxazoles and -pyrazoles |
US6187774B1 (en) * | 1996-03-04 | 2001-02-13 | Yoshitomi Pharmaceutical Industries, Ltd. | Fused heterocyclic compounds and pharmaceutical applications thereof |
HUP9603001A3 (en) * | 1996-10-30 | 1999-07-28 | Richter Gedeon Vegyeszet | Heterocycle compounds comprising nitrogen, process for producing them and pharmaceutical compositions containing the same |
ES2291023T3 (es) * | 1998-02-09 | 2008-02-16 | Duphar International Research B.V | Derivados de benzisoxazol que tienen actividad antagonista de d4. |
-
2000
- 2000-09-13 PT PT00964967T patent/PT1216249E/pt unknown
- 2000-09-13 AT AT00964967T patent/ATE254620T1/de not_active IP Right Cessation
- 2000-09-13 KR KR1020027003354A patent/KR20020027644A/ko not_active Application Discontinuation
- 2000-09-13 ES ES00964967T patent/ES2206305T3/es not_active Expired - Lifetime
- 2000-09-13 EP EP00964967A patent/EP1216249B1/en not_active Expired - Lifetime
- 2000-09-13 WO PCT/US2000/024949 patent/WO2001019832A2/en not_active Application Discontinuation
- 2000-09-13 DE DE60006698T patent/DE60006698T2/de not_active Expired - Lifetime
- 2000-09-13 CA CA002383327A patent/CA2383327C/en not_active Expired - Fee Related
- 2000-09-13 PL PL00354481A patent/PL354481A1/xx unknown
- 2000-09-13 EE EEP200200133A patent/EE200200133A/xx unknown
- 2000-09-13 IL IL14852200A patent/IL148522A0/xx unknown
- 2000-09-13 DK DK00964967T patent/DK1216249T3/da active
- 2000-09-13 CZ CZ2002896A patent/CZ2002896A3/cs unknown
- 2000-09-13 JP JP2001523409A patent/JP4717306B2/ja not_active Expired - Fee Related
- 2000-09-13 BR BR0014513-0A patent/BR0014513A/pt not_active IP Right Cessation
- 2000-09-13 HU HU0202712A patent/HUP0202712A3/hu unknown
- 2000-09-13 MX MXPA02002690A patent/MXPA02002690A/es active IP Right Grant
- 2000-09-13 EA EA200200357A patent/EA004177B1/ru not_active IP Right Cessation
- 2000-09-13 AU AU75772/00A patent/AU7577200A/en not_active Abandoned
- 2000-09-13 SK SK350-2002A patent/SK3502002A3/sk unknown
- 2000-09-13 AR ARP000104794A patent/AR032135A1/es not_active Application Discontinuation
-
2002
- 2002-03-01 ZA ZA200201760A patent/ZA200201760B/en unknown
- 2002-03-13 NO NO20021249A patent/NO20021249L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
PT1216249E (pt) | 2004-04-30 |
CA2383327C (en) | 2009-11-03 |
IL148522A0 (en) | 2002-09-12 |
DE60006698D1 (de) | 2003-12-24 |
KR20020027644A (ko) | 2002-04-13 |
DK1216249T3 (da) | 2004-03-15 |
CZ2002896A3 (cs) | 2002-08-14 |
JP2003509431A (ja) | 2003-03-11 |
EP1216249B1 (en) | 2003-11-19 |
WO2001019832A2 (en) | 2001-03-22 |
EA004177B1 (ru) | 2004-02-26 |
HUP0202712A3 (en) | 2004-12-28 |
ES2206305T3 (es) | 2004-05-16 |
EP1216249A2 (en) | 2002-06-26 |
WO2001019832A3 (en) | 2001-10-04 |
JP4717306B2 (ja) | 2011-07-06 |
PL354481A1 (en) | 2004-01-26 |
EE200200133A (et) | 2003-04-15 |
CA2383327A1 (en) | 2001-03-22 |
AU7577200A (en) | 2001-04-17 |
EA200200357A1 (ru) | 2002-10-31 |
ZA200201760B (en) | 2003-08-27 |
NO20021249L (no) | 2002-05-10 |
ATE254620T1 (de) | 2003-12-15 |
DE60006698T2 (de) | 2004-09-23 |
AR032135A1 (es) | 2003-10-29 |
MXPA02002690A (es) | 2004-09-10 |
HUP0202712A2 (hu) | 2002-12-28 |
NO20021249D0 (no) | 2002-03-13 |
BR0014513A (pt) | 2002-07-02 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NZ760006A (en) | Prodrugs of pyridone amides useful as modulators of sodium channels | |
TW201121977A (en) | Substituted dihydro benzocycloalkyloxymethyl oxazolopyrimidinones, preparation and use thereof | |
EP1216250B1 (en) | Thienoisoxazolyl and thienylpyrrazolyl phenoxy substituted propyl derivatives useful as d4 antagonists | |
US7511046B2 (en) | Thienoisoxazolyl- and thienylpyrrazolyl-phenoxy substituted propyl derivatives useful as D4 antagonists | |
EP1216244B1 (en) | Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists | |
CA2792918C (en) | Benzazepine compound | |
US7253165B2 (en) | Benzisoxazolyl-, pyridoisoxazolyl-and benzthienyl-phenoxy derivatives useful as D4 antagonists | |
CA3102458A1 (en) | Oga inhibitor compounds | |
SK3502002A3 (en) | Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists | |
US6696457B1 (en) | Morphinoid compounds | |
US7091199B1 (en) | Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists | |
MX2007011769A (es) | Ciclohexano-1,4-diaminas sustituidas con piperidinilo. | |
WO2012066486A1 (en) | Compound ethyl 8-oxo-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylate, salt, crystalline form, cocrystal, formulation, processes for preparation, application as medicaments, pharmaceutical compositions and new use particularly as inhibitor of aurora kinases |