EE200200133A - Asendamata tienoisoksasoolfenoksüetüül- ja propüülderivaadid ning nende kasutamine D4 antagonistidena - Google Patents
Asendamata tienoisoksasoolfenoksüetüül- ja propüülderivaadid ning nende kasutamine D4 antagonistidenaInfo
- Publication number
- EE200200133A EE200200133A EEP200200133A EEP200200133A EE200200133A EE 200200133 A EE200200133 A EE 200200133A EE P200200133 A EEP200200133 A EE P200200133A EE P200200133 A EEP200200133 A EE P200200133A EE 200200133 A EE200200133 A EE 200200133A
- Authority
- EE
- Estonia
- Prior art keywords
- thienoisoxazole
- phenoxyethyl
- antagonists
- unsubstituted
- propyl derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US39615699A | 1999-09-14 | 1999-09-14 | |
PCT/US2000/024949 WO2001019832A2 (en) | 1999-09-14 | 2000-09-13 | Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
EE200200133A true EE200200133A (et) | 2003-04-15 |
Family
ID=23566087
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EEP200200133A EE200200133A (et) | 1999-09-14 | 2000-09-13 | Asendamata tienoisoksasoolfenoksüetüül- ja propüülderivaadid ning nende kasutamine D4 antagonistidena |
Country Status (23)
Country | Link |
---|---|
EP (1) | EP1216249B1 (xx) |
JP (1) | JP4717306B2 (xx) |
KR (1) | KR20020027644A (xx) |
AR (1) | AR032135A1 (xx) |
AT (1) | ATE254620T1 (xx) |
AU (1) | AU7577200A (xx) |
BR (1) | BR0014513A (xx) |
CA (1) | CA2383327C (xx) |
CZ (1) | CZ2002896A3 (xx) |
DE (1) | DE60006698T2 (xx) |
DK (1) | DK1216249T3 (xx) |
EA (1) | EA004177B1 (xx) |
EE (1) | EE200200133A (xx) |
ES (1) | ES2206305T3 (xx) |
HU (1) | HUP0202712A3 (xx) |
IL (1) | IL148522A0 (xx) |
MX (1) | MXPA02002690A (xx) |
NO (1) | NO20021249L (xx) |
PL (1) | PL354481A1 (xx) |
PT (1) | PT1216249E (xx) |
SK (1) | SK3502002A3 (xx) |
WO (1) | WO2001019832A2 (xx) |
ZA (1) | ZA200201760B (xx) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0207449D0 (en) * | 2002-03-28 | 2002-05-08 | Glaxo Group Ltd | Novel compounds |
WO2018166855A1 (en) | 2017-03-16 | 2018-09-20 | Basf Se | Heterobicyclic substituted dihydroisoxazoles |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4728651A (en) * | 1985-10-24 | 1988-03-01 | Hoechst-Roussel Pharmaceuticals Inc. | Antihypertensive thieno-isoxazoles and -pyrazoles |
US6187774B1 (en) * | 1996-03-04 | 2001-02-13 | Yoshitomi Pharmaceutical Industries, Ltd. | Fused heterocyclic compounds and pharmaceutical applications thereof |
HUP9603001A3 (en) * | 1996-10-30 | 1999-07-28 | Richter Gedeon Vegyeszet | Heterocycle compounds comprising nitrogen, process for producing them and pharmaceutical compositions containing the same |
JP4627882B2 (ja) * | 1998-02-09 | 2011-02-09 | デユフアー・インターナシヨナル・リサーチ・ベー・ブイ | D4−アンタゴニスト活性を有するベンズイソキサゾール誘導体 |
-
2000
- 2000-09-13 AT AT00964967T patent/ATE254620T1/de not_active IP Right Cessation
- 2000-09-13 EP EP00964967A patent/EP1216249B1/en not_active Expired - Lifetime
- 2000-09-13 WO PCT/US2000/024949 patent/WO2001019832A2/en not_active Application Discontinuation
- 2000-09-13 HU HU0202712A patent/HUP0202712A3/hu unknown
- 2000-09-13 DK DK00964967T patent/DK1216249T3/da active
- 2000-09-13 EA EA200200357A patent/EA004177B1/ru not_active IP Right Cessation
- 2000-09-13 MX MXPA02002690A patent/MXPA02002690A/es active IP Right Grant
- 2000-09-13 SK SK350-2002A patent/SK3502002A3/sk unknown
- 2000-09-13 DE DE60006698T patent/DE60006698T2/de not_active Expired - Lifetime
- 2000-09-13 ES ES00964967T patent/ES2206305T3/es not_active Expired - Lifetime
- 2000-09-13 PL PL00354481A patent/PL354481A1/xx unknown
- 2000-09-13 AR ARP000104794A patent/AR032135A1/es not_active Application Discontinuation
- 2000-09-13 KR KR1020027003354A patent/KR20020027644A/ko not_active Application Discontinuation
- 2000-09-13 CA CA002383327A patent/CA2383327C/en not_active Expired - Fee Related
- 2000-09-13 AU AU75772/00A patent/AU7577200A/en not_active Abandoned
- 2000-09-13 JP JP2001523409A patent/JP4717306B2/ja not_active Expired - Fee Related
- 2000-09-13 EE EEP200200133A patent/EE200200133A/xx unknown
- 2000-09-13 CZ CZ2002896A patent/CZ2002896A3/cs unknown
- 2000-09-13 PT PT00964967T patent/PT1216249E/pt unknown
- 2000-09-13 BR BR0014513-0A patent/BR0014513A/pt not_active IP Right Cessation
- 2000-09-13 IL IL14852200A patent/IL148522A0/xx unknown
-
2002
- 2002-03-01 ZA ZA200201760A patent/ZA200201760B/en unknown
- 2002-03-13 NO NO20021249A patent/NO20021249L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EA004177B1 (ru) | 2004-02-26 |
CA2383327A1 (en) | 2001-03-22 |
WO2001019832A3 (en) | 2001-10-04 |
EP1216249B1 (en) | 2003-11-19 |
ATE254620T1 (de) | 2003-12-15 |
AR032135A1 (es) | 2003-10-29 |
JP4717306B2 (ja) | 2011-07-06 |
KR20020027644A (ko) | 2002-04-13 |
IL148522A0 (en) | 2002-09-12 |
HUP0202712A2 (hu) | 2002-12-28 |
CZ2002896A3 (cs) | 2002-08-14 |
EA200200357A1 (ru) | 2002-10-31 |
ES2206305T3 (es) | 2004-05-16 |
NO20021249D0 (no) | 2002-03-13 |
PL354481A1 (en) | 2004-01-26 |
JP2003509431A (ja) | 2003-03-11 |
MXPA02002690A (es) | 2004-09-10 |
BR0014513A (pt) | 2002-07-02 |
SK3502002A3 (en) | 2002-09-10 |
ZA200201760B (en) | 2003-08-27 |
EP1216249A2 (en) | 2002-06-26 |
DE60006698T2 (de) | 2004-09-23 |
DE60006698D1 (de) | 2003-12-24 |
PT1216249E (pt) | 2004-04-30 |
AU7577200A (en) | 2001-04-17 |
CA2383327C (en) | 2009-11-03 |
DK1216249T3 (da) | 2004-03-15 |
NO20021249L (no) | 2002-05-10 |
HUP0202712A3 (en) | 2004-12-28 |
WO2001019832A2 (en) | 2001-03-22 |
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