SK287811B6 - Glukopyranozyloxybenzylbenzénový derivát, farmaceutická kompozícia a ľudský SGLT2-inhibítor tento derivát obsahujúci a použitie tohto derivátu - Google Patents

Glukopyranozyloxybenzylbenzénový derivát, farmaceutická kompozícia a ľudský SGLT2-inhibítor tento derivát obsahujúci a použitie tohto derivátu Download PDF

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Publication number
SK287811B6
SK287811B6 SK334-2003A SK3342003A SK287811B6 SK 287811 B6 SK287811 B6 SK 287811B6 SK 3342003 A SK3342003 A SK 3342003A SK 287811 B6 SK287811 B6 SK 287811B6
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SK
Slovakia
Prior art keywords
group
straight
branched
carbon atoms
alkoxycarbonyl
Prior art date
Application number
SK334-2003A
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English (en)
Slovak (sk)
Other versions
SK3342003A3 (en
Inventor
Hideki Fujikura
Nobuhiko Fushimi
Toshihiro Nishimura
Kazuya Tatani
Masayuki Isaji
Original Assignee
Kissei Pharmaceutical Co., Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kissei Pharmaceutical Co., Ltd filed Critical Kissei Pharmaceutical Co., Ltd
Publication of SK3342003A3 publication Critical patent/SK3342003A3/sk
Publication of SK287811B6 publication Critical patent/SK287811B6/sk

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Genetics & Genomics (AREA)
  • Hematology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
SK334-2003A 2000-09-29 2001-09-21 Glukopyranozyloxybenzylbenzénový derivát, farmaceutická kompozícia a ľudský SGLT2-inhibítor tento derivát obsahujúci a použitie tohto derivátu SK287811B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000301523 2000-09-29
PCT/JP2001/008239 WO2002028872A1 (fr) 2000-09-29 2001-09-21 Derives de glucopyranosiloxybenzylbenzene et compositions therapeutiques contenant ces composes

Publications (2)

Publication Number Publication Date
SK3342003A3 SK3342003A3 (en) 2003-08-05
SK287811B6 true SK287811B6 (sk) 2011-10-04

Family

ID=18783054

Family Applications (1)

Application Number Title Priority Date Filing Date
SK334-2003A SK287811B6 (sk) 2000-09-29 2001-09-21 Glukopyranozyloxybenzylbenzénový derivát, farmaceutická kompozícia a ľudský SGLT2-inhibítor tento derivát obsahujúci a použitie tohto derivátu

Country Status (33)

Country Link
US (2) US6872706B2 (xx)
EP (1) EP1329456B1 (xx)
JP (1) JP3798375B2 (xx)
KR (1) KR100647204B1 (xx)
CN (1) CN1293087C (xx)
AR (1) AR030816A1 (xx)
AT (1) ATE335753T1 (xx)
AU (2) AU2001290257B2 (xx)
BG (1) BG66015B1 (xx)
BR (1) BR0114310A (xx)
CA (1) CA2423568C (xx)
CY (1) CY1106076T1 (xx)
CZ (1) CZ303544B6 (xx)
DE (1) DE60122193T2 (xx)
DK (1) DK1329456T3 (xx)
EA (1) EA005994B1 (xx)
ES (1) ES2269456T3 (xx)
HK (1) HK1061037A1 (xx)
HU (1) HUP0301178A3 (xx)
IL (2) IL155071A0 (xx)
MX (1) MXPA03002779A (xx)
MY (1) MY129023A (xx)
NO (1) NO327182B1 (xx)
NZ (1) NZ524917A (xx)
PE (1) PE20020476A1 (xx)
PL (1) PL205607B1 (xx)
PT (1) PT1329456E (xx)
SI (1) SI1329456T1 (xx)
SK (1) SK287811B6 (xx)
TW (1) TWI284641B (xx)
UA (1) UA73606C2 (xx)
WO (1) WO2002028872A1 (xx)
ZA (1) ZA200302283B (xx)

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Publication number Publication date
WO2002028872A1 (fr) 2002-04-11
CZ303544B6 (cs) 2012-11-28
BG66015B1 (bg) 2010-10-29
DE60122193T2 (de) 2007-07-05
US20040018998A1 (en) 2004-01-29
DE60122193D1 (de) 2006-09-21
PL362177A1 (en) 2004-10-18
ES2269456T3 (es) 2007-04-01
MXPA03002779A (es) 2004-05-04
AR030816A1 (es) 2003-09-03
NO20031407D0 (no) 2003-03-27
IL155071A (en) 2010-04-15
NO327182B1 (no) 2009-05-04
CN1293087C (zh) 2007-01-03
AU2001290257B2 (en) 2007-08-30
EP1329456A4 (en) 2005-03-30
DK1329456T3 (da) 2006-12-04
CA2423568A1 (en) 2002-04-11
US20050065098A1 (en) 2005-03-24
AU9025701A (en) 2002-04-15
NZ524917A (en) 2005-01-28
NO20031407L (no) 2003-04-30
JPWO2002028872A1 (ja) 2004-02-12
CA2423568C (en) 2011-03-15
EA005994B1 (ru) 2005-08-25
US6872706B2 (en) 2005-03-29
HK1061037A1 (en) 2004-09-03
ATE335753T1 (de) 2006-09-15
HUP0301178A2 (hu) 2003-11-28
KR20030036867A (ko) 2003-05-09
SK3342003A3 (en) 2003-08-05
CN1466590A (zh) 2004-01-07
CY1106076T1 (el) 2011-06-08
BG107674A (bg) 2004-01-30
ZA200302283B (en) 2005-05-27
IL155071A0 (en) 2003-10-31
PT1329456E (pt) 2006-12-29
TWI284641B (en) 2007-08-01
BR0114310A (pt) 2003-10-14
UA73606C2 (en) 2005-08-15
MY129023A (en) 2007-03-30
HUP0301178A3 (en) 2009-08-28
JP3798375B2 (ja) 2006-07-19
PL205607B1 (pl) 2010-05-31
EP1329456B1 (en) 2006-08-09
PE20020476A1 (es) 2002-07-04
KR100647204B1 (ko) 2006-11-17
EP1329456A1 (en) 2003-07-23
SI1329456T1 (sl) 2006-12-31
EA200300316A1 (ru) 2003-08-28

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