HUP0301178A3 - Glucopyranosyloxybenzylbenzene derivatives and pharmaceutical compositions containing the same - Google Patents

Glucopyranosyloxybenzylbenzene derivatives and pharmaceutical compositions containing the same

Info

Publication number
HUP0301178A3
HUP0301178A3 HU0301178A HUP0301178A HUP0301178A3 HU P0301178 A3 HUP0301178 A3 HU P0301178A3 HU 0301178 A HU0301178 A HU 0301178A HU P0301178 A HUP0301178 A HU P0301178A HU P0301178 A3 HUP0301178 A3 HU P0301178A3
Authority
HU
Hungary
Prior art keywords
same
pharmaceutical compositions
compositions containing
glucopyranosyloxybenzylbenzene derivatives
glucopyranosyloxybenzylbenzene
Prior art date
Application number
HU0301178A
Other languages
English (en)
Original Assignee
Kissei Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kissei Pharmaceutical filed Critical Kissei Pharmaceutical
Publication of HUP0301178A2 publication Critical patent/HUP0301178A2/hu
Publication of HUP0301178A3 publication Critical patent/HUP0301178A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
HU0301178A 2000-09-29 2001-09-21 Glucopyranosyloxybenzylbenzene derivatives and pharmaceutical compositions containing the same HUP0301178A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000301523 2000-09-29
PCT/JP2001/008239 WO2002028872A1 (fr) 2000-09-29 2001-09-21 Derives de glucopyranosiloxybenzylbenzene et compositions therapeutiques contenant ces composes

Publications (2)

Publication Number Publication Date
HUP0301178A2 HUP0301178A2 (hu) 2003-11-28
HUP0301178A3 true HUP0301178A3 (en) 2009-08-28

Family

ID=18783054

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0301178A HUP0301178A3 (en) 2000-09-29 2001-09-21 Glucopyranosyloxybenzylbenzene derivatives and pharmaceutical compositions containing the same

Country Status (33)

Country Link
US (2) US6872706B2 (hu)
EP (1) EP1329456B1 (hu)
JP (1) JP3798375B2 (hu)
KR (1) KR100647204B1 (hu)
CN (1) CN1293087C (hu)
AR (1) AR030816A1 (hu)
AT (1) ATE335753T1 (hu)
AU (2) AU9025701A (hu)
BG (1) BG66015B1 (hu)
BR (1) BR0114310A (hu)
CA (1) CA2423568C (hu)
CY (1) CY1106076T1 (hu)
CZ (1) CZ303544B6 (hu)
DE (1) DE60122193T2 (hu)
DK (1) DK1329456T3 (hu)
EA (1) EA005994B1 (hu)
ES (1) ES2269456T3 (hu)
HK (1) HK1061037A1 (hu)
HU (1) HUP0301178A3 (hu)
IL (2) IL155071A0 (hu)
MX (1) MXPA03002779A (hu)
MY (1) MY129023A (hu)
NO (1) NO327182B1 (hu)
NZ (1) NZ524917A (hu)
PE (1) PE20020476A1 (hu)
PL (1) PL205607B1 (hu)
PT (1) PT1329456E (hu)
SI (1) SI1329456T1 (hu)
SK (1) SK287811B6 (hu)
TW (1) TWI284641B (hu)
UA (1) UA73606C2 (hu)
WO (1) WO2002028872A1 (hu)
ZA (1) ZA200302283B (hu)

Families Citing this family (65)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1020944C (zh) 1990-01-30 1993-05-26 阿图尔-费希尔股份公司费希尔厂 紧固件
IL155071A0 (en) 2000-09-29 2003-10-31 Kissei Pharmaceutical Glucopyranosyloxybenzylbenzene derivatives and medical compositions containing the same
EP1344780A4 (en) * 2000-11-30 2004-01-28 Kissei Pharmaceutical GLUCOPYRANOSYLOXYBENZYLBENZOLE DERIVATIVES, MEDICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND INTERMEDIATE PRODUCTS FOR THEIR PREPARATION
TWI255817B (en) 2001-02-14 2006-06-01 Kissei Pharmaceutical Glucopyranosyloxybenzylbenzene derivatives and medicinal use thereof
MXPA04009229A (es) 2002-03-22 2004-11-26 Kissei Pharmaceutical Cristales derivados de glucopiranosiloxibencil benceno.
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CN1744916A (zh) * 2002-12-04 2006-03-08 橘生药品工业株式会社 预防和治疗高血糖所导致的疾病
JP4651934B2 (ja) * 2002-12-04 2011-03-16 キッセイ薬品工業株式会社 ベンジルフェノール誘導体、それを含有する医薬組成物およびその医薬用途
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DE10258008B4 (de) * 2002-12-12 2006-02-02 Sanofi-Aventis Deutschland Gmbh Heterocyclische Fluorglycosidderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zur Herstellung dieser Arzneimittel
UA86042C2 (en) * 2003-08-01 2009-03-25 Янссен Фармацевтика Н.В. Substituted indazole-o-glucosides
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JP5010918B2 (ja) * 2004-07-21 2012-08-29 キッセイ薬品工業株式会社 肝臓脂肪の異常蓄積に起因する疾患の進展抑制剤
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JP5073948B2 (ja) * 2005-01-31 2012-11-14 田辺三菱製薬株式会社 医薬組成物
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ATE453656T1 (de) * 2005-04-15 2010-01-15 Boehringer Ingelheim Int Glucopyranosyl-substituierte (heteroaryloxy- benzyl)-benzen-derivate als sglt-inhibitoren
US7723309B2 (en) * 2005-05-03 2010-05-25 Boehringer Ingelheim International Gmbh Crystalline forms of 1-chloro-4-(β-D-glucopyranos-1-yl)-2-[4-((R)-tetrahydrofuran-3-yloxy)-benzyl]-benzene, a method for its preparation and the use thereof for preparing medicaments
UA91546C2 (uk) * 2005-05-03 2010-08-10 Бьорінгер Інгельхайм Інтернаціональ Гмбх КРИСТАЛІЧНА ФОРМА 1-ХЛОР-4-(β-D-ГЛЮКОПІРАНОЗ-1-ИЛ)-2-[4-((S)-ТЕТРАГІДРОФУРАН-3-ІЛОКСИ)-БЕНЗИЛ]-БЕНЗОЛУ, СПОСІБ ЇЇ ОДЕРЖАННЯ ТА ЇЇ ЗАСТОСУВАННЯ ПРИ ПРИГОТУВАННІ ЛІКАРСЬКИХ ЗАСОБІВ
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DE102006028862A1 (de) 2006-06-23 2007-12-27 Merck Patent Gmbh 3-Amino-imidazo[1,2-a]pyridinderivate
TW200817424A (en) 2006-08-04 2008-04-16 Daiichi Sankyo Co Ltd Benzylphenyl glucopyranoside derivatives
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JP5330260B2 (ja) 2006-12-06 2013-10-30 スミスクライン ビーチャム コーポレーション 二環式化合物ならびに抗糖尿病薬としての使用
DE102007008420A1 (de) 2007-02-21 2008-08-28 Merck Patent Gmbh Benzimidazolderivate
CL2008002427A1 (es) * 2007-08-16 2009-09-11 Boehringer Ingelheim Int Composicion farmaceutica que comprende 1-cloro-4-(b-d-glucopiranos-1-il)-2-[4-((s)-tetrahidrofurano-3-iloxi)bencil]-benceno combinado con 1-[(4-metilquinazolin-2-il)metil]-3-metil-7-(2-butin-1-il)-8-(3-(r)-aminopiperidin-1-il)xantina; y su uso para tratar diabetes mellitus tipo 2.
DE102007048716A1 (de) 2007-10-11 2009-04-23 Merck Patent Gmbh Imidazo[1,2-a]pyrimidinderivate
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Family Cites Families (6)

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FR2549476B1 (fr) * 1983-07-20 1986-04-25 Rech Ind Benzyl-phenyl-osides, procede de preparation et utilisation en therapeutique
US5731292A (en) * 1992-11-12 1998-03-24 Tanabe Seiyaku Co., Ltd. Dihydrochalcone derivatives which are hypoglycemic agents
CA2102591C (en) * 1992-11-12 2000-12-26 Kenji Tsujihara Hypoglycemic agent
KR100660738B1 (ko) 2000-03-17 2006-12-22 깃세이 야쿠힌 고교 가부시키가이샤 글루코피라노실록시 벤질벤젠 유도체, 그것을 함유하는의약조성물 및 그 제조중간체
US6683056B2 (en) * 2000-03-30 2004-01-27 Bristol-Myers Squibb Company O-aryl glucoside SGLT2 inhibitors and method
IL155071A0 (en) 2000-09-29 2003-10-31 Kissei Pharmaceutical Glucopyranosyloxybenzylbenzene derivatives and medical compositions containing the same

Also Published As

Publication number Publication date
AU9025701A (en) 2002-04-15
MXPA03002779A (es) 2004-05-04
BG66015B1 (bg) 2010-10-29
US20050065098A1 (en) 2005-03-24
PE20020476A1 (es) 2002-07-04
CY1106076T1 (el) 2011-06-08
NZ524917A (en) 2005-01-28
UA73606C2 (en) 2005-08-15
IL155071A (en) 2010-04-15
NO20031407D0 (no) 2003-03-27
AR030816A1 (es) 2003-09-03
MY129023A (en) 2007-03-30
JPWO2002028872A1 (ja) 2004-02-12
DE60122193D1 (de) 2006-09-21
NO327182B1 (no) 2009-05-04
JP3798375B2 (ja) 2006-07-19
CA2423568C (en) 2011-03-15
EP1329456A4 (en) 2005-03-30
SK287811B6 (sk) 2011-10-04
ATE335753T1 (de) 2006-09-15
ZA200302283B (en) 2005-05-27
CN1466590A (zh) 2004-01-07
AU2001290257B2 (en) 2007-08-30
PL362177A1 (en) 2004-10-18
CA2423568A1 (en) 2002-04-11
EP1329456B1 (en) 2006-08-09
HUP0301178A2 (hu) 2003-11-28
SI1329456T1 (sl) 2006-12-31
WO2002028872A1 (fr) 2002-04-11
US20040018998A1 (en) 2004-01-29
KR100647204B1 (ko) 2006-11-17
US6872706B2 (en) 2005-03-29
KR20030036867A (ko) 2003-05-09
PT1329456E (pt) 2006-12-29
EA200300316A1 (ru) 2003-08-28
SK3342003A3 (en) 2003-08-05
CZ303544B6 (cs) 2012-11-28
TWI284641B (en) 2007-08-01
PL205607B1 (pl) 2010-05-31
BR0114310A (pt) 2003-10-14
EA005994B1 (ru) 2005-08-25
IL155071A0 (en) 2003-10-31
HK1061037A1 (en) 2004-09-03
CN1293087C (zh) 2007-01-03
ES2269456T3 (es) 2007-04-01
DE60122193T2 (de) 2007-07-05
EP1329456A1 (en) 2003-07-23
DK1329456T3 (da) 2006-12-04
BG107674A (bg) 2004-01-30
NO20031407L (no) 2003-04-30

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Legal Events

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FD9A Lapse of provisional protection due to non-payment of fees