SK15282001A3 - Perorálny farmaceutický prípravok na aplikáciu do ilea, obsahujúci inhibítor transportu žlčových kyselín - Google Patents

Perorálny farmaceutický prípravok na aplikáciu do ilea, obsahujúci inhibítor transportu žlčových kyselín Download PDF

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Publication number
SK15282001A3
SK15282001A3 SK1528-2001A SK15282001A SK15282001A3 SK 15282001 A3 SK15282001 A3 SK 15282001A3 SK 15282001 A SK15282001 A SK 15282001A SK 15282001 A3 SK15282001 A3 SK 15282001A3
Authority
SK
Slovakia
Prior art keywords
ibat inhibitor
ileum
ibat
composition
bile acid
Prior art date
Application number
SK1528-2001A
Other languages
English (en)
Slovak (sk)
Inventor
Bertil Abrahamsson
Ann-Margret Lindqvist
Anna-Lena Ungell
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of SK15282001A3 publication Critical patent/SK15282001A3/sk

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
SK1528-2001A 1999-04-19 2000-04-19 Perorálny farmaceutický prípravok na aplikáciu do ilea, obsahujúci inhibítor transportu žlčových kyselín SK15282001A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9901387A SE9901387D0 (sv) 1999-04-19 1999-04-19 New pharmaceutical foromaulations
PCT/SE2000/000755 WO2000062810A1 (en) 1999-04-19 2000-04-19 An oral formulation for ileum administering comprising an inhibitor compound of the ileal bile acid transport

Publications (1)

Publication Number Publication Date
SK15282001A3 true SK15282001A3 (sk) 2002-04-04

Family

ID=20415263

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1528-2001A SK15282001A3 (sk) 1999-04-19 2000-04-19 Perorálny farmaceutický prípravok na aplikáciu do ilea, obsahujúci inhibítor transportu žlčových kyselín

Country Status (27)

Country Link
EP (1) EP1173205B1 (sl)
JP (1) JP2002542208A (sl)
KR (1) KR20010108516A (sl)
CN (1) CN1348384A (sl)
AT (1) ATE296641T1 (sl)
AU (1) AU767425B2 (sl)
BR (1) BR0009835A (sl)
CA (1) CA2379105A1 (sl)
CZ (1) CZ20013743A3 (sl)
DE (1) DE60020551T2 (sl)
DK (1) DK1173205T3 (sl)
EE (1) EE04607B1 (sl)
ES (1) ES2241603T3 (sl)
HK (1) HK1042850A1 (sl)
HU (1) HUP0200793A3 (sl)
IL (1) IL145871A0 (sl)
IS (1) IS2161B (sl)
NO (1) NO20015063D0 (sl)
NZ (1) NZ514264A (sl)
PL (1) PL351186A1 (sl)
PT (1) PT1173205E (sl)
SE (1) SE9901387D0 (sl)
SI (1) SI1173205T1 (sl)
SK (1) SK15282001A3 (sl)
TR (1) TR200103033T2 (sl)
WO (1) WO2000062810A1 (sl)
ZA (1) ZA200108539B (sl)

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GB0121337D0 (en) 2001-09-04 2001-10-24 Astrazeneca Ab Chemical compounds
GB0121621D0 (en) 2001-09-07 2001-10-31 Astrazeneca Ab Chemical compounds
GB0121622D0 (en) 2001-09-07 2001-10-31 Astrazeneca Ab Chemical compounds
ATE349214T1 (de) 2001-09-08 2007-01-15 Astrazeneca Ab Benzothiazepin und benzothiadiazepin derivative mit hemmender wirkung auf den säuretransport in den gallengängen zur behandlung von hyperlipidaemia
GB0209467D0 (en) 2002-04-25 2002-06-05 Astrazeneca Ab Chemical compounds
GB0213669D0 (en) 2002-06-14 2002-07-24 Astrazeneca Ab Chemical compounds
GB0216321D0 (en) * 2002-07-13 2002-08-21 Astrazeneca Ab Therapeutic treatment
GB0304194D0 (en) 2003-02-25 2003-03-26 Astrazeneca Ab Chemical compounds
GB0307918D0 (en) 2003-04-05 2003-05-14 Astrazeneca Ab Therapeutic use
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EP4137137A1 (en) 2010-05-26 2023-02-22 Satiogen Pharmaceuticals, Inc. Bile acid recycling inhibitors and satiogens for treatment of diabetes, obesity, and inflammatory gastrointestinal conditions
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AU2011326872C1 (en) * 2010-11-08 2015-02-19 Albireo Ab A pharmaceutical combination comprising an IBAT inhibitor and a bile acid binder
US20130108573A1 (en) 2011-10-28 2013-05-02 Lumena Pharmaceuticals, Inc. Bile Acid Recycling Inhibitors for Treatment of Hypercholemia and Cholestatic Liver Disease
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US10441605B2 (en) 2016-02-09 2019-10-15 Albireo Ab Oral cholestyramine formulation and use thereof
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CN108601745B (zh) 2016-02-09 2021-12-07 阿尔比里奥公司 口服考来烯胺制剂及其用途
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US10722457B2 (en) 2018-08-09 2020-07-28 Albireo Ab Oral cholestyramine formulation and use thereof
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US11549878B2 (en) 2018-08-09 2023-01-10 Albireo Ab In vitro method for determining the adsorbing capacity of an insoluble adsorbant
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WO2021110884A1 (en) 2019-12-04 2021-06-10 Albireo Ab Benzothia(di)azepine compounds and their use as bile acid modulators
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TW202134218A (zh) 2019-12-04 2021-09-16 瑞典商艾爾比瑞歐公司 苯并噻氮呯化合物及其作為膽酸調節劑之用途
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JP2023537285A (ja) 2020-08-03 2023-08-31 アルビレオ・アクチボラグ ベンゾチア(ジ)アゼピン化合物及び胆汁酸モジュレータとしてのそれらの使用
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Also Published As

Publication number Publication date
EP1173205A1 (en) 2002-01-23
HUP0200793A3 (en) 2004-07-28
ES2241603T3 (es) 2005-11-01
PT1173205E (pt) 2005-10-31
EP1173205B1 (en) 2005-06-01
AU767425B2 (en) 2003-11-13
EE04607B1 (et) 2006-04-17
IS2161B (is) 2006-11-15
HUP0200793A2 (hu) 2002-07-29
NZ514264A (en) 2003-10-31
SI1173205T1 (sl) 2005-10-31
SE9901387D0 (sv) 1999-04-19
DE60020551D1 (de) 2005-07-07
CA2379105A1 (en) 2000-10-26
WO2000062810A1 (en) 2000-10-26
JP2002542208A (ja) 2002-12-10
BR0009835A (pt) 2002-01-08
ZA200108539B (en) 2003-01-17
AU4633500A (en) 2000-11-02
NO20015063L (no) 2001-10-18
CN1348384A (zh) 2002-05-08
TR200103033T2 (tr) 2002-03-21
CZ20013743A3 (cs) 2002-01-16
KR20010108516A (ko) 2001-12-07
IL145871A0 (en) 2002-07-25
NO20015063D0 (no) 2001-10-18
IS6109A (is) 2001-10-16
EE200100545A (et) 2003-02-17
HK1042850A1 (en) 2002-08-30
PL351186A1 (en) 2003-03-24
DK1173205T3 (da) 2005-08-08
DE60020551T2 (de) 2006-03-23
ATE296641T1 (de) 2005-06-15

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