SK12682003A3 - Prípravky obsahujúce imidazotriazinón na nazálnu aplikáciu - Google Patents

Prípravky obsahujúce imidazotriazinón na nazálnu aplikáciu Download PDF

Info

Publication number
SK12682003A3
SK12682003A3 SK1268-2003A SK12682003A SK12682003A3 SK 12682003 A3 SK12682003 A3 SK 12682003A3 SK 12682003 A SK12682003 A SK 12682003A SK 12682003 A3 SK12682003 A3 SK 12682003A3
Authority
SK
Slovakia
Prior art keywords
group
hydrochloride
carbon atoms
alkyl
optionally
Prior art date
Application number
SK1268-2003A
Other languages
English (en)
Slovak (sk)
Inventor
Peter Serno
Andreas Ohm
Wolfgang Barth
Richard-Josef Bauer
Hans-Martin Siefert
Dieter Zimmer
Original Assignee
Bayer Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft
Publication of SK12682003A3 publication Critical patent/SK12682003A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0043—Nose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/007—Pulmonary tract; Aromatherapy
    • A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A61P23/02—Local anaesthetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Otolaryngology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pulmonology (AREA)
  • Anesthesiology (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SK1268-2003A 2001-04-12 2002-04-03 Prípravky obsahujúce imidazotriazinón na nazálnu aplikáciu SK12682003A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10118306A DE10118306A1 (de) 2001-04-12 2001-04-12 Imidazotriazinonhaltige Zusammensetzungen zur nasalen Applikation
PCT/EP2002/003663 WO2002083674A2 (de) 2001-04-12 2002-04-03 Imidazotriazinonhaltige zusammensetzungen zur nasalen applikation

Publications (1)

Publication Number Publication Date
SK12682003A3 true SK12682003A3 (sk) 2004-03-02

Family

ID=7681379

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1268-2003A SK12682003A3 (sk) 2001-04-12 2002-04-03 Prípravky obsahujúce imidazotriazinón na nazálnu aplikáciu

Country Status (25)

Country Link
US (2) US6740306B2 (bg)
EP (1) EP1381368A2 (bg)
JP (1) JP2004525968A (bg)
KR (1) KR20030087072A (bg)
CN (1) CN1537004A (bg)
AR (1) AR035821A1 (bg)
BG (1) BG108245A (bg)
BR (1) BR0208813A (bg)
CA (1) CA2443639A1 (bg)
CZ (1) CZ20032752A3 (bg)
DE (1) DE10118306A1 (bg)
DO (1) DOP2002000373A (bg)
EC (1) ECSP034795A (bg)
EE (1) EE200300501A (bg)
GT (1) GT200200070A (bg)
HU (1) HUP0303877A3 (bg)
IL (1) IL158255A0 (bg)
MX (1) MXPA03009314A (bg)
NO (1) NO20034556L (bg)
PE (1) PE20021035A1 (bg)
PL (1) PL363033A1 (bg)
RU (1) RU2003133143A (bg)
SK (1) SK12682003A3 (bg)
UY (1) UY27256A1 (bg)
WO (1) WO2002083674A2 (bg)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0209541A (pt) * 2001-05-09 2004-04-20 Bayer Healthcare Ag Uso das imidazotriazinonas 2-fenil-substituìdas
DE102004023069A1 (de) * 2004-05-11 2005-12-08 Bayer Healthcare Ag Neue Darreichungsformen des PDE 5-Inhibitors Vardenafil
AU2005322305B2 (en) * 2004-12-23 2010-09-16 Roxro Pharma, Inc. Therapeutic compositions for intranasal administration of ketorolac
DE102005001989A1 (de) * 2005-01-15 2006-07-20 Bayer Healthcare Ag Intravenöse Formulierungen von PDE-Inhibitoren
DE102005009240A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften
DE102005009241A1 (de) * 2005-03-01 2006-09-07 Bayer Healthcare Ag Arzneiformen mit kontrollierter Bioverfügbarkeit
CA2612917A1 (en) * 2005-06-23 2007-01-04 Schering Corporation Rapidly absorbing oral formulations of pde5 inhibitors
KR20080056250A (ko) * 2005-09-29 2008-06-20 바이엘 헬스케어 아게 비뇨기 장애의 치료를 위한 ｐｄｅ 억제제 및 이들의 조합
US20100184769A1 (en) * 2007-06-13 2010-07-22 Bayer Schering Pharma Aktiengesellschaft Pde inhibitors for the treatment of hearing impairment
AU2009257385A1 (en) * 2008-06-13 2009-12-17 Roxro Pharma, Inc. Pharmaceutical formulation of ketorolac for intranasal administration
US8551454B2 (en) * 2009-03-13 2013-10-08 Luitpold Pharmaceuticals, Inc. Device for intranasal administration
US8277781B2 (en) * 2009-03-13 2012-10-02 Luitpold Pharmaceuticals, Inc. Device for intranasal administration
WO2017168174A1 (en) 2016-04-02 2017-10-05 N4 Pharma Uk Limited New pharmaceutical forms of sildenafil
WO2020006606A1 (en) * 2018-07-05 2020-01-09 Helium 3 Resources Pty Ltd A pharmaceutical composition and method of use of same
SE542968C2 (en) * 2018-10-26 2020-09-22 Lindahl Anders Treatment of osteoarthritis
AU2021280285A1 (en) * 2020-05-26 2023-02-02 Strategic Drug Solutions, Inc. Formulations and methods for treating erectile dysfunction

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4602099A (en) * 1973-04-02 1986-07-22 Merrell Dow Pharmaceuticals Inc. Antirhinovirus agents
GB9013750D0 (en) 1990-06-20 1990-08-08 Pfizer Ltd Therapeutic agents
GB9301192D0 (en) 1993-06-09 1993-06-09 Trott Francis W Flower shaped mechanised table
GB9514465D0 (en) 1995-07-14 1995-09-13 Glaxo Lab Sa Chemical compounds
GB9514473D0 (en) 1995-07-14 1995-09-13 Glaxo Lab Sa Chemical compounds
ATE236156T1 (de) 1996-05-31 2003-04-15 Mochida Pharm Co Ltd Pyridocarbazol derivate die einen cgmp-pde inhibilierenden effekt haben
GB2315673A (en) * 1996-08-01 1998-02-11 Merck & Co Inc Treatment of migraine
BR9809508A (pt) * 1997-05-29 2000-06-20 Mochida Pharm Co Ltd Agente terapêutico para disfunção de ereção
AU9214498A (en) 1997-09-23 1999-04-12 Eli Lilly And Company Treatment of attention-deficit/hyperactivity disorder
DE59803108D1 (de) 1997-11-12 2002-03-21 Bayer Ag 2-phenyl-substituierte imidazotriazinone als phosphodiesterase inhibitoren
TWI223598B (en) * 1998-06-22 2004-11-11 Pfizer Ireland Pharmaceuticals An intranasal pharmaceutical composition for the treatment of male erectile dysfunction or female sexual disorders, an intranasal delivery system or device and sildenafil mesylate
AU4717299A (en) * 1998-06-26 2000-01-17 Nastech Pharmaceutical Company, Inc Nasal delivery of sildenafil citrate
JP2002542147A (ja) * 1998-12-14 2002-12-10 セレジィ ファーマシューティカルス， インコーポレイテッド 肛門直腸障害の処置のための組成物および方法

Also Published As

Publication number Publication date
PE20021035A1 (es) 2002-11-29
CZ20032752A3 (cs) 2004-01-14
GT200200070A (es) 2003-01-31
BG108245A (bg) 2005-01-31
JP2004525968A (ja) 2004-08-26
US6740306B2 (en) 2004-05-25
CN1537004A (zh) 2004-10-13
UY27256A1 (es) 2002-11-29
ECSP034795A (es) 2003-12-01
HUP0303877A2 (hu) 2004-03-29
WO2002083674A3 (de) 2003-01-09
US20040248891A1 (en) 2004-12-09
EP1381368A2 (de) 2004-01-21
NO20034556D0 (no) 2003-10-10
IL158255A0 (en) 2004-05-12
RU2003133143A (ru) 2005-04-10
AR035821A1 (es) 2004-07-14
EE200300501A (et) 2003-12-15
DE10118306A1 (de) 2002-10-17
HUP0303877A3 (en) 2005-05-30
US20030022894A1 (en) 2003-01-30
MXPA03009314A (es) 2004-03-10
DOP2002000373A (es) 2002-11-30
NO20034556L (no) 2003-12-10
WO2002083674A2 (de) 2002-10-24
PL363033A1 (en) 2004-11-15
KR20030087072A (ko) 2003-11-12
CA2443639A1 (en) 2002-10-24
BR0208813A (pt) 2004-03-09

Similar Documents

Publication Publication Date Title
US11717571B2 (en) Intranasal epinephrine formulations and methods for the treatment of disease
AP1178A (en) Intranasal formulations for treating sexual disorders
EP2522365B1 (en) Compositions comprising azelastine and methods of use thereof
SK12682003A3 (sk) Prípravky obsahujúce imidazotriazinón na nazálnu aplikáciu
US20070065366A1 (en) Pharmaceutical formulations comprising a long-acting beta2-agonist for administration by nebulisation
US7220767B2 (en) Pharmaceutical formulations containing zolmitriptan
KR20020016831A (ko) 비내용 모르핀을 함유하는 의약 조성물 및 그 제조방법
AU2005281736A1 (en) Roflumilast and syk inhibitor combination and methods of use thereof
SK15112002A3 (sk) Liečivo na liečenie sexuálnej dysfunkcie pacienta
US20040142944A1 (en) Compositions for nasal application
JP2011524366A (ja) 鼻内投与のためのケトロラクの薬学的処方物
ES2791775B2 (es) Formulaciones de epinefrina intranasal y metodos para el tratamiento de enfermedades
GB2114001A (en) Nasal pharmaceutical compositions
FI81258C (fi) Foerfarande foer framstaellning av en farmaceutisk komposition foer nasal administration.