SK12452001A3 - Zlúčenina vytvárajúca inhibítor metaloproteinázy, farmaceutický prostriedok, spôsob prípravy liečiva a liečivo - Google Patents

Zlúčenina vytvárajúca inhibítor metaloproteinázy, farmaceutický prostriedok, spôsob prípravy liečiva a liečivo Download PDF

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SK12452001A3
SK12452001A3 SK1245-2001A SK12452001A SK12452001A3 SK 12452001 A3 SK12452001 A3 SK 12452001A3 SK 12452001 A SK12452001 A SK 12452001A SK 12452001 A3 SK12452001 A3 SK 12452001A3
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Slovakia
Prior art keywords
amino
aryl
heteroaryl
alkyl
cycloalkyl
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SK1245-2001A
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English (en)
Slovak (sk)
Inventor
Michael George Natchus
Roger Gunnard Bookland
Neil Gregory Almstead
Stanislaw Pikul
Biswanath De
Menyan Cheng
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The Procter & Gamble Company
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Publication of SK12452001A3 publication Critical patent/SK12452001A3/sk

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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/337—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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SK1245-2001A 1999-03-03 2000-03-01 Zlúčenina vytvárajúca inhibítor metaloproteinázy, farmaceutický prostriedok, spôsob prípravy liečiva a liečivo SK12452001A3 (sk)

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CO5150219A1 (es) 2002-04-29
IL145089A0 (en) 2002-06-30
AU3386000A (en) 2000-09-21
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WO2000051975A1 (fr) 2000-09-08
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AU764051B2 (en) 2003-08-07
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PE20001565A1 (es) 2001-02-02
TR200102523T2 (tr) 2002-02-21
HUP0202199A2 (en) 2002-10-28
US6197770B1 (en) 2001-03-06
PL350340A1 (en) 2002-12-02
JP2002538136A (ja) 2002-11-12
NO20014242D0 (no) 2001-08-31
MA25391A1 (fr) 2002-04-01
KR20010102486A (ko) 2001-11-15
CZ20013176A3 (cs) 2002-04-17
MXPA01008855A (es) 2002-07-02

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